ATE377603T1 - Tetracyklische arylsulfonylindole mit affinität zum serotonin rezeptor - Google Patents
Tetracyklische arylsulfonylindole mit affinität zum serotonin rezeptorInfo
- Publication number
- ATE377603T1 ATE377603T1 AT03760857T AT03760857T ATE377603T1 AT E377603 T1 ATE377603 T1 AT E377603T1 AT 03760857 T AT03760857 T AT 03760857T AT 03760857 T AT03760857 T AT 03760857T AT E377603 T1 ATE377603 T1 AT E377603T1
- Authority
- AT
- Austria
- Prior art keywords
- pharmaceutically acceptable
- tetracyclic
- compound
- arylsulfonylindoles
- affinity
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Addiction (AREA)
- Anesthesiology (AREA)
- Obesity (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Indole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN478CH2002 | 2002-06-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE377603T1 true ATE377603T1 (de) | 2007-11-15 |
Family
ID=29798513
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT03760857T ATE377603T1 (de) | 2002-06-21 | 2003-06-19 | Tetracyklische arylsulfonylindole mit affinität zum serotonin rezeptor |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US7649097B2 (de) |
| EP (1) | EP1523486B1 (de) |
| JP (1) | JP4473120B2 (de) |
| CN (1) | CN100378108C (de) |
| AT (1) | ATE377603T1 (de) |
| AU (1) | AU2003249582B2 (de) |
| BR (1) | BR0312176A (de) |
| CA (1) | CA2490254C (de) |
| DE (1) | DE60317333T2 (de) |
| DK (1) | DK1523486T3 (de) |
| ES (1) | ES2297216T3 (de) |
| HK (1) | HK1074843A1 (de) |
| MX (1) | MXPA04012832A (de) |
| NZ (1) | NZ537770A (de) |
| RU (1) | RU2340619C2 (de) |
| WO (1) | WO2004000849A2 (de) |
| ZA (1) | ZA200409886B (de) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0315958B8 (pt) * | 2002-11-28 | 2021-05-25 | Suven Life Sciences Ltd | composto, composição farmacêutica, processo para a preparação de um composto, novos intermediários e uso do composto |
| PT1581538E (pt) * | 2002-12-18 | 2007-05-31 | Suven Life Sciences Ltd | Indolos tetracíclicos substituidos na posição 3 que possuem afinidade pelo receptor de serotonina. |
| DK1704154T3 (da) * | 2004-01-02 | 2009-08-31 | Suven Life Sciences Ltd | Nye indeno(2,1-A)indener og isoindol(2,1-A)indoler |
| CA2561733A1 (en) * | 2004-04-01 | 2005-10-13 | Cardiome Pharma Corp. | Pegylated ion channel modulating compounds |
| WO2006095360A1 (en) * | 2005-03-08 | 2006-09-14 | Suven Life Sciences Limited | Process for preparing substituted benzothiazinoindoles |
| JP2023508469A (ja) | 2019-12-26 | 2023-03-02 | ギルガメッシュ・ファーマシューティカルズ・インコーポレイテッド | アリールシクロヘキシルアミン誘導体及び精神障害の処置におけるそれらの使用 |
| MX2022010082A (es) | 2020-02-18 | 2022-11-14 | Gilgamesh Pharmaceuticals Inc | Triptaminas especificas para usarse en el tratamiento de trastornos de estado de animo. |
| EP4153564A4 (de) | 2020-05-19 | 2024-06-19 | Cybin IRL Limited | Deuterierte tryptaminderivate und verfahren zur verwendung |
| CN116056762A (zh) | 2020-06-12 | 2023-05-02 | 贝克利心理科技有限公司 | 包含5-甲氧基-n,n-二甲基色胺的苯甲酸盐的组合物 |
| GB202212116D0 (en) | 2022-08-19 | 2022-10-05 | Beckley Psytech Ltd | Pharmaceutically acceptable salts and Compositions thereof |
Family Cites Families (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3487091A (en) * | 1967-12-18 | 1969-12-30 | American Home Prod | 1-(benzyl- or substituted-benzyl)-3-(2-substituted-ethyl) indoles |
| ZA795239B (en) | 1978-10-12 | 1980-11-26 | Glaxo Group Ltd | Heterocyclic compounds |
| BE889931A (fr) | 1980-08-12 | 1982-02-11 | Glaxo Group Ltd | Derives indoliques, leur preparation et leurs applications en tant que medicaments |
| GB8600397D0 (en) | 1986-01-08 | 1986-02-12 | Glaxo Group Ltd | Chemical compounds |
| GB8719167D0 (en) | 1987-08-13 | 1987-09-23 | Glaxo Group Ltd | Chemical compounds |
| GB8724912D0 (en) | 1987-10-23 | 1987-11-25 | Wellcome Found | Indole derivatives |
| GB8819024D0 (en) | 1988-08-10 | 1988-09-14 | Glaxo Group Ltd | Chemical compounds |
| IL96891A0 (en) | 1990-01-17 | 1992-03-29 | Merck Sharp & Dohme | Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them |
| CA2042295A1 (fr) | 1990-05-15 | 1991-11-16 | Jacques Chauveau | Derives de mediateurs endogenes, leurs sels, procede de preparation, applications, et compositions les renfermant |
| RU2160736C2 (ru) | 1990-06-07 | 2000-12-20 | Зенека Лимитед | Производные индола и их физиологически приемлемые соли и сольваты, способы их получения, лекарственное средство для лечения или профилактики клинических состояний, для которых показан прием агониста "5-нт1-подобного" рецептора, и способ его получения |
| CZ283018B6 (cs) | 1991-02-01 | 1997-12-17 | Merck Sharp And Dohme Limited | Deriváty imidazolu, triazolu a tetrazolu a farmaceutické přípravky na jejich bázi |
| GB9113802D0 (en) | 1991-06-26 | 1991-08-14 | Smithkline Beecham Plc | Medicaments |
| GB9210400D0 (en) | 1992-05-15 | 1992-07-01 | Merck Sharp & Dohme | Therapeutic agents |
| KR940007001A (ko) | 1992-09-16 | 1994-04-26 | 최승주 | 새로운 n-신나모일-2-메틸-5-메톡시-3-인돌 아세트산 에스테르, 그 제조방법 및 이를 함유하는 약학적 제제 |
| JP2000026471A (ja) * | 1998-07-10 | 2000-01-25 | Nippon Soda Co Ltd | １１−ホルミル−インドロ［１，２−ｂ］［１，２］ベンズイソチアゾールおよび農園芸用殺菌剤 |
| GB9820113D0 (en) | 1998-09-15 | 1998-11-11 | Merck Sharp & Dohme | Therapeutic agents |
| ES2260958T3 (es) | 1998-12-11 | 2006-11-01 | Virginia Commonwealth University | Ligandos selectivos del receptor 5 - ht 6. |
| MXPA03008726A (es) | 2001-03-29 | 2003-12-12 | Lilly Co Eli | N-(2-ariletil)benzilaminas como antagonistas del receptor 5-ht6. |
-
2003
- 2003-06-19 CA CA2490254A patent/CA2490254C/en not_active Expired - Fee Related
- 2003-06-19 US US10/519,219 patent/US7649097B2/en not_active Expired - Fee Related
- 2003-06-19 AT AT03760857T patent/ATE377603T1/de active
- 2003-06-19 BR BR0312176-3A patent/BR0312176A/pt not_active IP Right Cessation
- 2003-06-19 RU RU2005101344/04A patent/RU2340619C2/ru not_active IP Right Cessation
- 2003-06-19 NZ NZ537770A patent/NZ537770A/en not_active IP Right Cessation
- 2003-06-19 AU AU2003249582A patent/AU2003249582B2/en not_active Ceased
- 2003-06-19 WO PCT/IN2003/000222 patent/WO2004000849A2/en active IP Right Grant
- 2003-06-19 EP EP03760857A patent/EP1523486B1/de not_active Expired - Lifetime
- 2003-06-19 JP JP2004515418A patent/JP4473120B2/ja not_active Expired - Fee Related
- 2003-06-19 DK DK03760857T patent/DK1523486T3/da active
- 2003-06-19 DE DE60317333T patent/DE60317333T2/de not_active Expired - Lifetime
- 2003-06-19 MX MXPA04012832A patent/MXPA04012832A/es active IP Right Grant
- 2003-06-19 ES ES03760857T patent/ES2297216T3/es not_active Expired - Lifetime
- 2003-06-19 CN CNB038146029A patent/CN100378108C/zh not_active Expired - Fee Related
-
2004
- 2004-12-07 ZA ZA200409886A patent/ZA200409886B/en unknown
-
2005
- 2005-10-06 HK HK05108865A patent/HK1074843A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ES2297216T3 (es) | 2008-05-01 |
| WO2004000849A2 (en) | 2003-12-31 |
| RU2340619C2 (ru) | 2008-12-10 |
| DE60317333D1 (de) | 2007-12-20 |
| AU2003249582A1 (en) | 2004-01-06 |
| MXPA04012832A (es) | 2005-05-27 |
| NZ537770A (en) | 2007-03-30 |
| AU2003249582B2 (en) | 2006-08-03 |
| CN100378108C (zh) | 2008-04-02 |
| JP4473120B2 (ja) | 2010-06-02 |
| DE60317333T2 (de) | 2008-08-28 |
| CA2490254C (en) | 2011-11-01 |
| JP2005535621A (ja) | 2005-11-24 |
| CN1662544A (zh) | 2005-08-31 |
| BR0312176A (pt) | 2005-04-05 |
| EP1523486A2 (de) | 2005-04-20 |
| DK1523486T3 (da) | 2008-03-03 |
| CA2490254A1 (en) | 2003-12-31 |
| US20050203154A1 (en) | 2005-09-15 |
| RU2005101344A (ru) | 2005-08-20 |
| HK1074843A1 (en) | 2005-11-25 |
| ZA200409886B (en) | 2006-07-26 |
| WO2004000849A3 (en) | 2004-03-25 |
| US7649097B2 (en) | 2010-01-19 |
| EP1523486B1 (de) | 2007-11-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
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