EE03263B1 - Erütromütsiini derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja vaheühendid - Google Patents

Erütromütsiini derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja vaheühendid

Info

Publication number
EE03263B1
EE03263B1 EE9600151A EE9600151A EE03263B1 EE 03263 B1 EE03263 B1 EE 03263B1 EE 9600151 A EE9600151 A EE 9600151A EE 9600151 A EE9600151 A EE 9600151A EE 03263 B1 EE03263 B1 EE 03263B1
Authority
EE
Estonia
Prior art keywords
intermediates
preparation
pharmaceutical composition
erythromycin derivatives
erythromycin
Prior art date
Application number
EE9600151A
Other languages
English (en)
Estonian (et)
Inventor
Agouridas Constantin
Chantot Jean-Fran�Ois
Denis Alexis
Gouin D'ambrieres Solange
Le Martret Odile
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of EE03263B1 publication Critical patent/EE03263B1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Indole Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
EE9600151A 1994-05-03 1995-05-02 Erütromütsiini derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja vaheühendid EE03263B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9405368A FR2719587B1 (fr) 1994-05-03 1994-05-03 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
PCT/FR1995/000565 WO1995029929A1 (fr) 1994-05-03 1995-05-02 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
EE03263B1 true EE03263B1 (et) 2000-04-17

Family

ID=9462785

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9600151A EE03263B1 (et) 1994-05-03 1995-05-02 Erütromütsiini derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja vaheühendid

Country Status (42)

Country Link
US (2) US5635485A (ro)
EP (1) EP0680967B1 (ro)
JP (4) JP2992540B2 (ro)
KR (1) KR100312267B1 (ro)
CN (2) CN1052984C (ro)
AP (1) AP558A (ro)
AT (1) ATE172203T1 (ro)
AU (1) AU684027B2 (ro)
BG (1) BG63087B1 (ro)
BR (1) BR9507700A (ro)
CA (1) CA2189271C (ro)
CZ (1) CZ293455B6 (ro)
DE (2) DE69505296T2 (ro)
DK (1) DK0680967T3 (ro)
DZ (1) DZ1878A1 (ro)
EE (1) EE03263B1 (ro)
ES (1) ES2122472T3 (ro)
FI (1) FI111263B (ro)
FR (1) FR2719587B1 (ro)
GE (1) GEP19991538B (ro)
HU (2) HU219599B (ro)
IL (1) IL113245A (ro)
LU (1) LU90872I2 (ro)
LV (1) LV11739B (ro)
MA (1) MA23534A1 (ro)
MD (1) MD1233C2 (ro)
NL (1) NL300077I1 (ro)
NO (2) NO308853B1 (ro)
NZ (1) NZ285416A (ro)
OA (1) OA10319A (ro)
PL (1) PL182034B1 (ro)
RO (1) RO113350B1 (ro)
RU (1) RU2144036C1 (ro)
SI (1) SI0680967T1 (ro)
SK (1) SK281707B6 (ro)
TJ (1) TJ313B (ro)
TN (1) TNSN95049A1 (ro)
TW (1) TW341573B (ro)
UA (1) UA51618C2 (ro)
WO (1) WO1995029929A1 (ro)
YU (1) YU49235B (ro)
ZA (1) ZA953501B (ro)

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FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
US5780605A (en) * 1997-09-08 1998-07-14 Abbott Laboratories 6,9-bridged erythromycin derivatives
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
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Also Published As

Publication number Publication date
MD1233C2 (ro) 2000-10-31
FI964395L (fi) 1996-10-31
HUT75698A (en) 1997-05-28
JP3998828B2 (ja) 2007-10-31
NO308853B1 (no) 2000-11-06
CN1229082A (zh) 1999-09-22
DE10299001I2 (de) 2012-07-05
JPH11152296A (ja) 1999-06-08
MX9605208A (es) 1997-09-30
NO2001027I1 (no) 2002-01-28
WO1995029929A1 (fr) 1995-11-09
CA2189271C (fr) 2005-12-27
JP2992540B2 (ja) 1999-12-20
HU219599B (hu) 2001-05-28
FR2719587A1 (fr) 1995-11-10
OA10319A (fr) 1997-10-07
ATE172203T1 (de) 1998-10-15
FR2719587B1 (fr) 1996-07-12
US5635485A (en) 1997-06-03
NO964654D0 (no) 1996-11-04
DE69505296T2 (de) 1999-04-22
NL300077I1 (nl) 2002-03-01
US6100404A (en) 2000-08-08
EP0680967A1 (fr) 1995-11-08
UA51618C2 (uk) 2002-12-16
FI111263B (fi) 2003-06-30
SK140296A3 (en) 1998-04-08
GEP19991538B (en) 1999-03-05
HU9904687D0 (en) 2000-03-28
SK281707B6 (sk) 2001-07-10
JP2007269810A (ja) 2007-10-18
AU2449995A (en) 1995-11-29
CN1052984C (zh) 2000-05-31
TNSN95049A1 (fr) 1996-02-06
SI0680967T1 (en) 1999-02-28
CZ321496A3 (en) 1997-08-13
BG63087B1 (bg) 2001-03-30
DZ1878A1 (fr) 2002-02-17
AP558A (en) 1996-11-07
YU27095A (sh) 1998-05-15
CN1151746A (zh) 1997-06-11
JPH0853489A (ja) 1996-02-27
HU227493B1 (en) 2011-07-28
HU9603038D0 (en) 1997-01-28
DE10299001I1 (de) 2012-07-05
PL317071A1 (en) 1997-03-03
AU684027B2 (en) 1997-11-27
LU90872I2 (fr) 2002-03-12
CA2189271A1 (fr) 1995-11-09
JP4750755B2 (ja) 2011-08-17
CZ293455B6 (cs) 2004-05-12
EP0680967B1 (fr) 1998-10-14
FI964395A0 (fi) 1996-10-31
BG100951A (en) 1997-08-29
TW341573B (en) 1998-10-01
NZ285416A (en) 1997-07-27
DK0680967T3 (da) 1999-06-23
PL182034B1 (pl) 2001-10-31
NO964654L (no) 1996-11-04
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JP4658902B2 (ja) 2011-03-23
RU2144036C1 (ru) 2000-01-10
MD1233B1 (ro) 1999-05-31
YU49235B (sh) 2004-12-31
HK1010732A1 (en) 1999-06-25
JP2007045847A (ja) 2007-02-22
AP9500744A0 (en) 1995-07-31
LV11739B (en) 1997-08-20
CN1088709C (zh) 2002-08-07
KR100312267B1 (ko) 2002-06-22
LV11739A (lv) 1997-04-20
IL113245A (en) 1999-11-30
BR9507700A (pt) 1997-08-19
ZA953501B (en) 1996-05-02
IL113245A0 (en) 1995-07-31
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DE69505296D1 (de) 1998-11-19
MA23534A1 (fr) 1995-12-31

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