NO308853B1 - Nye erytromycinderivater, farmasøytiske preparater som inneholder dem, samt mellomprodukter for deres fremstilling - Google Patents
Nye erytromycinderivater, farmasøytiske preparater som inneholder dem, samt mellomprodukter for deres fremstillingInfo
- Publication number
- NO308853B1 NO308853B1 NO964654A NO964654A NO308853B1 NO 308853 B1 NO308853 B1 NO 308853B1 NO 964654 A NO964654 A NO 964654A NO 964654 A NO964654 A NO 964654A NO 308853 B1 NO308853 B1 NO 308853B1
- Authority
- NO
- Norway
- Prior art keywords
- intermediates
- preparation
- pharmaceuticals containing
- erythromycin derivatives
- new erythromycin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Quinoline Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyrrole Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9405368A FR2719587B1 (fr) | 1994-05-03 | 1994-05-03 | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
PCT/FR1995/000565 WO1995029929A1 (fr) | 1994-05-03 | 1995-05-02 | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
Publications (3)
Publication Number | Publication Date |
---|---|
NO964654L NO964654L (no) | 1996-11-04 |
NO964654D0 NO964654D0 (no) | 1996-11-04 |
NO308853B1 true NO308853B1 (no) | 2000-11-06 |
Family
ID=9462785
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO964654A NO308853B1 (no) | 1994-05-03 | 1996-11-04 | Nye erytromycinderivater, farmasøytiske preparater som inneholder dem, samt mellomprodukter for deres fremstilling |
NO2001027C NO2001027I1 (no) | 1994-05-03 | 2001-12-28 | Telitromycin |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO2001027C NO2001027I1 (no) | 1994-05-03 | 2001-12-28 | Telitromycin |
Country Status (43)
Country | Link |
---|---|
US (2) | US5635485A (no) |
EP (1) | EP0680967B1 (no) |
JP (4) | JP2992540B2 (no) |
KR (1) | KR100312267B1 (no) |
CN (2) | CN1052984C (no) |
AP (1) | AP558A (no) |
AT (1) | ATE172203T1 (no) |
AU (1) | AU684027B2 (no) |
BG (1) | BG63087B1 (no) |
BR (1) | BR9507700A (no) |
CA (1) | CA2189271C (no) |
CZ (1) | CZ293455B6 (no) |
DE (2) | DE69505296T2 (no) |
DK (1) | DK0680967T3 (no) |
DZ (1) | DZ1878A1 (no) |
EE (1) | EE03263B1 (no) |
ES (1) | ES2122472T3 (no) |
FI (1) | FI111263B (no) |
FR (1) | FR2719587B1 (no) |
GE (1) | GEP19991538B (no) |
HK (1) | HK1010732A1 (no) |
HU (2) | HU219599B (no) |
IL (1) | IL113245A (no) |
LU (1) | LU90872I2 (no) |
LV (1) | LV11739B (no) |
MA (1) | MA23534A1 (no) |
MD (1) | MD1233C2 (no) |
NL (1) | NL300077I1 (no) |
NO (2) | NO308853B1 (no) |
NZ (1) | NZ285416A (no) |
OA (1) | OA10319A (no) |
PL (1) | PL182034B1 (no) |
RO (1) | RO113350B1 (no) |
RU (1) | RU2144036C1 (no) |
SI (1) | SI0680967T1 (no) |
SK (1) | SK281707B6 (no) |
TJ (1) | TJ313B (no) |
TN (1) | TNSN95049A1 (no) |
TW (1) | TW341573B (no) |
UA (1) | UA51618C2 (no) |
WO (1) | WO1995029929A1 (no) |
YU (1) | YU49235B (no) |
ZA (1) | ZA953501B (no) |
Families Citing this family (85)
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US5708005A (en) * | 1995-06-27 | 1998-01-13 | Takeda Chemical Industries, Ltd. | Quinolines, their production and use |
FR2742757B1 (fr) * | 1995-12-22 | 1998-01-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
IL128681A0 (en) * | 1996-09-04 | 2000-01-31 | Abbott Lab | 6-O substituted ketolides having antibacterial activity |
UA51730C2 (uk) * | 1996-09-04 | 2002-12-16 | Ебботт Лабораторіз | 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців |
FR2757168B1 (fr) * | 1996-12-12 | 1999-06-11 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2760017B1 (fr) * | 1997-02-27 | 1999-04-30 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments |
US5780605A (en) * | 1997-09-08 | 1998-07-14 | Abbott Laboratories | 6,9-bridged erythromycin derivatives |
FR2771008B1 (fr) * | 1997-11-17 | 2000-04-28 | Hoechst Marion Roussel Inc | Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose |
JP4573925B2 (ja) * | 1998-07-09 | 2010-11-04 | アベンティス・ファーマ・ソシエテ・アノニム | 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用 |
FR2781484B1 (fr) * | 1998-07-21 | 2001-08-10 | Hoechst Marion Roussel Inc | Nouveaux derives de la 6-deoxy erythromycine, leur procede de preparation et leur application comme medicaments |
EP1115732B1 (en) * | 1998-09-22 | 2005-06-29 | Pfizer Products Inc. | Carbamate and carbazate ketolide antibiotics |
FR2785612A1 (fr) * | 1998-11-10 | 2000-05-12 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
FR2786188B1 (fr) * | 1998-11-24 | 2002-10-31 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments |
TW526202B (en) | 1998-11-27 | 2003-04-01 | Shionogi & Amp Co | Broad spectrum cephem having benzo[4,5-b]pyridium methyl group of antibiotic activity |
ATE344269T1 (de) | 1998-12-10 | 2006-11-15 | Pfizer Prod Inc | Carbamat und carbazat ketolid antibiotika |
BR9916969A (pt) * | 1999-01-27 | 2001-11-06 | Pfizer Prod Inc | Antibióticos cetólidos |
FR2789392B1 (fr) * | 1999-02-04 | 2001-10-05 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
US6054435A (en) * | 1999-03-19 | 2000-04-25 | Abbott Laboratories | 6-O-substituted macrolides having antibacterial activity |
US6399582B1 (en) | 1999-04-16 | 2002-06-04 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
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US6590083B1 (en) | 1999-04-16 | 2003-07-08 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
KR100710605B1 (ko) | 1999-04-16 | 2007-04-24 | 코산 바이오사이언시즈, 인코포레이티드 | 매크롤라이드 항감염제 |
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US6946446B2 (en) | 2000-02-24 | 2005-09-20 | Abbott Laboratories | Anti-infective agents useful against multidrug-resistant strains of bacteria |
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US8063021B2 (en) * | 2002-01-17 | 2011-11-22 | Kosan Biosciences Incorporated | Ketolide anti-infective compounds |
US6995143B2 (en) | 2002-02-28 | 2006-02-07 | Basilea Pharmaceutica Ag | Macrolides with antibacterial activity |
JP4530851B2 (ja) | 2002-07-08 | 2010-08-25 | グラクソスミスクライン・イストラジヴァッキ・センタル・ザグレブ・ドルズバ・ゼー・オメイェノ・オドゴヴォルノスティオ | ステロイド/非ステロイド抗炎症活性分子、抗新生物活性分子および抗ウイルス活性分子用担体としての新規な化合物、組成物 |
CN100577681C (zh) | 2002-07-08 | 2010-01-06 | 葛兰素伊斯特拉齐瓦基森塔萨格勒布公司 | 用于治疗炎性疾病和病症的新化合物、组合物和方法 |
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AR085286A1 (es) | 2011-02-21 | 2013-09-18 | Taisho Pharmaceutical Co Ltd | Derivado de macrolido sustituido en la posicion c-4 |
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CN105524132B (zh) * | 2014-09-30 | 2019-07-02 | 中国医学科学院药物研究所 | 含有喹啉取代基的红霉素a酮内酯类抗生素衍生物、其制备方法及应用 |
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FR2692579B1 (fr) * | 1992-06-19 | 1995-06-02 | Roussel Uclaf | Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments. |
FR2697524B1 (fr) * | 1992-11-05 | 1994-12-23 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
US5527780A (en) * | 1992-11-05 | 1996-06-18 | Roussel Uclaf | Erythromycin derivatives |
TW370529B (en) * | 1992-12-17 | 1999-09-21 | Pfizer | Pyrazolopyrimidines |
HRP930014A2 (en) * | 1993-01-08 | 1994-08-31 | Pliva Pharm & Chem Works | 9-deoxo-9a-aza-11-deoxy-9a-homoeritromycin a 9a, 11-cyclic carbamates |
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1994
- 1994-05-03 FR FR9405368A patent/FR2719587B1/fr not_active Expired - Lifetime
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1995
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- 1995-05-01 JP JP7128791A patent/JP2992540B2/ja not_active Expired - Lifetime
- 1995-05-02 DZ DZ950049A patent/DZ1878A1/fr active
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- 1995-05-02 CN CN95193911A patent/CN1052984C/zh not_active Expired - Lifetime
- 1995-05-02 SI SI9530184T patent/SI0680967T1/xx unknown
- 1995-05-02 TN TNTNSN95049A patent/TNSN95049A1/fr unknown
- 1995-05-02 KR KR1019960706191A patent/KR100312267B1/ko not_active IP Right Cessation
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- 1995-05-02 AU AU24499/95A patent/AU684027B2/en not_active Expired
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- 1995-05-02 GE GEAP19953425A patent/GEP19991538B/en unknown
- 1995-05-02 RU RU96123129A patent/RU2144036C1/ru active
- 1995-05-02 AT AT95400987T patent/ATE172203T1/de active
- 1995-05-02 MD MD97-0010A patent/MD1233C2/ro unknown
- 1995-05-02 EE EE9600151A patent/EE03263B1/xx active Protection Beyond IP Right Term
- 1995-05-02 RO RO96-02081A patent/RO113350B1/ro unknown
- 1995-05-02 CZ CZ19963214A patent/CZ293455B6/cs not_active IP Right Cessation
- 1995-05-02 NZ NZ285416A patent/NZ285416A/en not_active IP Right Cessation
- 1995-05-02 DE DE2002199001 patent/DE10299001I1/de active Granted
- 1995-05-02 AP APAP/P/1995/000744A patent/AP558A/en active
- 1995-05-02 WO PCT/FR1995/000565 patent/WO1995029929A1/fr active IP Right Grant
- 1995-05-02 PL PL95317071A patent/PL182034B1/pl unknown
- 1995-05-02 EP EP95400987A patent/EP0680967B1/fr not_active Expired - Lifetime
- 1995-06-29 TW TW084106692A patent/TW341573B/zh not_active IP Right Cessation
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1996
- 1996-10-31 FI FI964395A patent/FI111263B/fi not_active IP Right Cessation
- 1996-11-01 OA OA60917A patent/OA10319A/fr unknown
- 1996-11-01 LV LVP-96-421A patent/LV11739B/lv unknown
- 1996-11-01 TJ TJ96000417A patent/TJ313B/xx unknown
- 1996-11-01 BG BG100951A patent/BG63087B1/bg unknown
- 1996-11-04 NO NO964654A patent/NO308853B1/no not_active IP Right Cessation
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1997
- 1997-01-09 US US08/780,861 patent/US6100404A/en not_active Expired - Lifetime
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1998
- 1998-08-24 JP JP25181798A patent/JP3998828B2/ja not_active Expired - Lifetime
- 1998-11-05 HK HK98111758A patent/HK1010732A1/xx not_active IP Right Cessation
- 1998-12-07 CN CN98123072A patent/CN1088709C/zh not_active Expired - Lifetime
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2001
- 2001-12-28 NL NL300077C patent/NL300077I1/nl unknown
- 2001-12-28 NO NO2001027C patent/NO2001027I1/no unknown
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2002
- 2002-01-08 LU LU90872C patent/LU90872I2/xx unknown
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2006
- 2006-11-21 JP JP2006314281A patent/JP4658902B2/ja not_active Expired - Lifetime
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2007
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Legal Events
Date | Code | Title | Description |
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SPCG | Granted supplementary protection certificate |
Spc suppl protection certif: SPC/NO 2001 027 Filing date: 20011228 Extension date: 20160709 |
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MK1K | Patent expired |