AP558A - New erythromycin derivatives, their preparation process and their use as medicaments. - Google Patents

New erythromycin derivatives, their preparation process and their use as medicaments. Download PDF

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Publication number
AP558A
AP558A APAP/P/1995/000744A AP9500744A AP558A AP 558 A AP558 A AP 558A AP 9500744 A AP9500744 A AP 9500744A AP 558 A AP558 A AP 558A
Authority
AP
ARIPO
Prior art keywords
butanamine
methyl
dideoxy
oxy
formula
Prior art date
Application number
APAP/P/1995/000744A
Other languages
English (en)
Other versions
AP9500744A0 (en
Inventor
Constantin Agouridas
Jean-Francis Chantot (Deceased)
Alexis Denis
Solange Gouin D'ambrieres
Martret Odile Le
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of AP9500744A0 publication Critical patent/AP9500744A0/xx
Application granted granted Critical
Publication of AP558A publication Critical patent/AP558A/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/16Otologicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pulmonology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pyrrole Compounds (AREA)
APAP/P/1995/000744A 1994-05-03 1995-05-02 New erythromycin derivatives, their preparation process and their use as medicaments. AP558A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9405368A FR2719587B1 (fr) 1994-05-03 1994-05-03 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Publications (2)

Publication Number Publication Date
AP9500744A0 AP9500744A0 (en) 1995-07-31
AP558A true AP558A (en) 1996-11-07

Family

ID=9462785

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1995/000744A AP558A (en) 1994-05-03 1995-05-02 New erythromycin derivatives, their preparation process and their use as medicaments.

Country Status (43)

Country Link
US (2) US5635485A (no)
EP (1) EP0680967B1 (no)
JP (4) JP2992540B2 (no)
KR (1) KR100312267B1 (no)
CN (2) CN1052984C (no)
AP (1) AP558A (no)
AT (1) ATE172203T1 (no)
AU (1) AU684027B2 (no)
BG (1) BG63087B1 (no)
BR (1) BR9507700A (no)
CA (1) CA2189271C (no)
CZ (1) CZ293455B6 (no)
DE (2) DE10299001I2 (no)
DK (1) DK0680967T3 (no)
DZ (1) DZ1878A1 (no)
EE (1) EE03263B1 (no)
ES (1) ES2122472T3 (no)
FI (1) FI111263B (no)
FR (1) FR2719587B1 (no)
GE (1) GEP19991538B (no)
HK (1) HK1010732A1 (no)
HU (2) HU227493B1 (no)
IL (1) IL113245A (no)
LU (1) LU90872I2 (no)
LV (1) LV11739B (no)
MA (1) MA23534A1 (no)
MD (1) MD1233C2 (no)
NL (1) NL300077I1 (no)
NO (2) NO308853B1 (no)
NZ (1) NZ285416A (no)
OA (1) OA10319A (no)
PL (1) PL182034B1 (no)
RO (1) RO113350B1 (no)
RU (1) RU2144036C1 (no)
SI (1) SI0680967T1 (no)
SK (1) SK281707B6 (no)
TJ (1) TJ313B (no)
TN (1) TNSN95049A1 (no)
TW (1) TW341573B (no)
UA (1) UA51618C2 (no)
WO (1) WO1995029929A1 (no)
YU (1) YU49235B (no)
ZA (1) ZA953501B (no)

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UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
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FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
US5780605A (en) * 1997-09-08 1998-07-14 Abbott Laboratories 6,9-bridged erythromycin derivatives
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
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FR2785612A1 (fr) * 1998-11-10 2000-05-12 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
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EP0487411A1 (fr) * 1990-11-21 1992-05-27 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation, les nouveaux intermédiaires obtenus et leur application comme médicaments
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Also Published As

Publication number Publication date
JP4658902B2 (ja) 2011-03-23
LV11739B (en) 1997-08-20
AU2449995A (en) 1995-11-29
ZA953501B (en) 1996-05-02
NO2001027I1 (no) 2002-01-28
CA2189271C (fr) 2005-12-27
MD1233B1 (en) 1999-05-31
EE03263B1 (et) 2000-04-17
RU2144036C1 (ru) 2000-01-10
CZ293455B6 (cs) 2004-05-12
CN1151746A (zh) 1997-06-11
HUT75698A (en) 1997-05-28
FI964395A0 (fi) 1996-10-31
DE10299001I1 (de) 2012-07-05
IL113245A0 (en) 1995-07-31
ATE172203T1 (de) 1998-10-15
HK1010732A1 (en) 1999-06-25
EP0680967A1 (fr) 1995-11-08
DE10299001I2 (de) 2012-07-05
HU227493B1 (en) 2011-07-28
HU9603038D0 (en) 1997-01-28
MA23534A1 (fr) 1995-12-31
SK281707B6 (sk) 2001-07-10
MD1233C2 (ro) 2000-10-31
FR2719587B1 (fr) 1996-07-12
RO113350B1 (ro) 1998-06-30
JP4750755B2 (ja) 2011-08-17
JPH0853489A (ja) 1996-02-27
HU9904687D0 (en) 2000-03-28
US5635485A (en) 1997-06-03
JP2007045847A (ja) 2007-02-22
YU27095A (sh) 1998-05-15
NZ285416A (en) 1997-07-27
US6100404A (en) 2000-08-08
NO964654L (no) 1996-11-04
JP3998828B2 (ja) 2007-10-31
JP2007269810A (ja) 2007-10-18
MX9605208A (es) 1997-09-30
FI111263B (fi) 2003-06-30
NO308853B1 (no) 2000-11-06
CA2189271A1 (fr) 1995-11-09
DZ1878A1 (fr) 2002-02-17
DK0680967T3 (da) 1999-06-23
DE69505296D1 (de) 1998-11-19
SK140296A3 (en) 1998-04-08
CN1229082A (zh) 1999-09-22
KR100312267B1 (ko) 2002-06-22
WO1995029929A1 (fr) 1995-11-09
BG63087B1 (bg) 2001-03-30
IL113245A (en) 1999-11-30
NO964654D0 (no) 1996-11-04
PL317071A1 (en) 1997-03-03
FR2719587A1 (fr) 1995-11-10
AU684027B2 (en) 1997-11-27
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AP9500744A0 (en) 1995-07-31
GEP19991538B (en) 1999-03-05
LU90872I2 (fr) 2002-03-12
YU49235B (sh) 2004-12-31
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HU219599B (hu) 2001-05-28
JP2992540B2 (ja) 1999-12-20
BR9507700A (pt) 1997-08-19
EP0680967B1 (fr) 1998-10-14
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CN1052984C (zh) 2000-05-31
DE69505296T2 (de) 1999-04-22
PL182034B1 (pl) 2001-10-31
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BG100951A (en) 1997-08-29
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UA51618C2 (uk) 2002-12-16
CZ321496A3 (en) 1997-08-13
SI0680967T1 (en) 1999-02-28
ES2122472T3 (es) 1998-12-16
LV11739A (lv) 1997-04-20
OA10319A (fr) 1997-10-07
JPH11152296A (ja) 1999-06-08

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