EA019741B1 - Пиррольные соединения - Google Patents

Пиррольные соединения Download PDF

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Publication number
EA019741B1
EA019741B1 EA201170384A EA201170384A EA019741B1 EA 019741 B1 EA019741 B1 EA 019741B1 EA 201170384 A EA201170384 A EA 201170384A EA 201170384 A EA201170384 A EA 201170384A EA 019741 B1 EA019741 B1 EA 019741B1
Authority
EA
Eurasian Patent Office
Prior art keywords
compound
acid
group
ulcers
ulcer
Prior art date
Application number
EA201170384A
Other languages
English (en)
Russian (ru)
Other versions
EA201170384A1 (ru
Inventor
Харуюки Нисида
Ясуеси Арикава
Икуо Фудзимори
Original Assignee
Такеда Фармасьютикал Компани Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41508823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA019741(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Такеда Фармасьютикал Компани Лимитед filed Critical Такеда Фармасьютикал Компани Лимитед
Publication of EA201170384A1 publication Critical patent/EA201170384A1/ru
Publication of EA019741B1 publication Critical patent/EA019741B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
EA201170384A 2008-08-27 2009-08-26 Пиррольные соединения EA019741B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2008218851 2008-08-27
JP2008269099 2008-10-17
PCT/JP2009/065279 WO2010024451A1 (en) 2008-08-27 2009-08-26 Pyrrole compounds

Publications (2)

Publication Number Publication Date
EA201170384A1 EA201170384A1 (ru) 2011-10-31
EA019741B1 true EA019741B1 (ru) 2014-05-30

Family

ID=41508823

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201170384A EA019741B1 (ru) 2008-08-27 2009-08-26 Пиррольные соединения

Country Status (38)

Country Link
US (3) US8592597B2 (enExample)
EP (1) EP2318390B1 (enExample)
JP (1) JP5638515B2 (enExample)
KR (1) KR101629181B1 (enExample)
CN (1) CN102197033B (enExample)
AR (1) AR073136A1 (enExample)
AU (1) AU2009284867B2 (enExample)
BR (1) BRPI0917705A2 (enExample)
CA (1) CA2735162C (enExample)
CL (1) CL2011000402A1 (enExample)
CO (1) CO6321166A2 (enExample)
CR (1) CR20110169A (enExample)
CY (1) CY1114452T1 (enExample)
DK (1) DK2318390T3 (enExample)
DO (1) DOP2011000061A (enExample)
EA (1) EA019741B1 (enExample)
EC (1) ECSP11010912A (enExample)
ES (1) ES2423289T3 (enExample)
GE (1) GEP20135786B (enExample)
HR (1) HRP20130653T1 (enExample)
IL (1) IL211335A (enExample)
JO (1) JO2871B1 (enExample)
MA (1) MA32647B1 (enExample)
ME (1) ME01598B (enExample)
MX (1) MX2011001955A (enExample)
MY (1) MY152008A (enExample)
NZ (1) NZ591793A (enExample)
PE (2) PE20110300A1 (enExample)
PL (1) PL2318390T3 (enExample)
PT (1) PT2318390E (enExample)
RS (1) RS52872B (enExample)
SI (1) SI2318390T1 (enExample)
SM (1) SMT201300085B (enExample)
TW (1) TWI473798B (enExample)
UA (1) UA105185C2 (enExample)
UY (1) UY32074A (enExample)
WO (1) WO2010024451A1 (enExample)
ZA (1) ZA201101774B (enExample)

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PL2318390T3 (pl) 2008-08-27 2013-09-30 Takeda Pharmaceuticals Co Związki pirolowe
US20110229879A1 (en) * 2010-03-19 2011-09-22 University Of Rochester Methods and compositions for nuclear staining
CN102452979B (zh) * 2010-11-03 2015-04-01 天津药明康德新药开发有限公司 5-氟-3-吡啶磺酰氯的合成方法
CN102863371B (zh) * 2011-07-06 2016-04-13 中国科学院上海有机化学研究所 氟代二氢吡咯或氟代吡咯
US10039813B2 (en) 2012-02-07 2018-08-07 Massachusetts Institute Of Technology Use of antagonists of ghrelin or ghrelin receptor to prevent or treat stress-sensitive psychiatric illness
CN110917130A (zh) 2012-06-27 2020-03-27 武田药品工业株式会社 用盐稳定的胺和有机酸的液体制剂
WO2014133059A1 (ja) * 2013-02-28 2014-09-04 武田薬品工業株式会社 スルホニルクロライド化合物の製造法
WO2014144231A1 (en) 2013-03-15 2014-09-18 Massachusetts Institute Of Technology Use of antagonists of growth hormone or growth hormone receptor to prevent or treat stress-sensitive psychiatric illness
KR102084185B1 (ko) 2013-08-29 2020-03-04 주식회사 대웅제약 테트라히드로사이클로펜타피롤 유도체 및 이의 제조방법
CN105367550A (zh) * 2014-08-11 2016-03-02 江苏柯菲平医药股份有限公司 四氢环戊二烯并[c]吡咯类衍生物、其制备方法及其在医药上的应用
UY36547A (es) 2015-02-05 2016-06-01 Bayer Cropscience Ag Derivados heterocíclicos condensados bicíclicos sustituidos por 2-(het)arilo como pesticidas
US10317418B2 (en) 2015-02-24 2019-06-11 Massachusetts Institute Of Technology Use of ghrelin or functional ghrelin receptor agonists to prevent and treat stress-sensitive psychiatric illness
TWI710379B (zh) 2015-07-30 2020-11-21 日商武田藥品工業股份有限公司 錠劑
ES2882667T3 (es) 2015-08-07 2021-12-02 Bayer Cropscience Ag Derivados heterocíclicos condensados sustituidos por 2-(het)arilo como pesticidas
CN106430006B (zh) * 2016-08-18 2018-06-12 国网湖南省电力公司带电作业中心 配电线路移动式绝缘登高作业装置及方法
CN108203430A (zh) * 2016-12-16 2018-06-26 天地人和生物科技有限公司 一种新型可逆性质子泵抑制剂及其制备方法和用途
PE20200442A1 (es) 2017-07-10 2020-02-28 Takeda Pharmaceuticals Co Preparacion que comprende vonoprazan
KR102126576B1 (ko) 2018-09-19 2020-06-24 주식회사 대웅제약 4-메톡시 피롤 유도체의 제조 방법
CN113527536B (zh) * 2020-04-21 2024-03-22 杭州德柯医疗科技有限公司 一种含氟多糖高分子化合物及其制备方法
ES3014815T3 (en) * 2020-06-17 2025-04-25 Ildong Pharmaceutical Co Ltd Novel acid secretion inhibitor and use thereof
EP4074317A1 (en) 2021-04-14 2022-10-19 Bayer AG Phosphorus derivatives as novel sos1 inhibitors
CN113620930B (zh) * 2021-07-12 2022-08-16 南京烁慧医药科技有限公司 一种含磺酰胺结构的化合物及其制备方法和应用、一种药物组合物及应用
KR20240119083A (ko) * 2021-12-15 2024-08-06 일동제약(주) 1-설포닐 피롤 유도체의 신규 염, 이의 제조 방법 및 이를 포함하는 약학 조성물
KR102802551B1 (ko) * 2021-12-15 2025-05-07 유노비아 주식회사 1-설포닐 피롤 유도체의 신규 염, 이의 제조 방법 및 이를 포함하는 약학 조성물
KR20230102353A (ko) * 2021-12-30 2023-07-07 주식회사 대웅제약 삼중음성유방암의 예방 또는 치료용 약학적 조성물

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EP1803709A1 (en) * 2004-09-30 2007-07-04 Takeda Pharmaceutical Company Limited Proton pump inhibitors
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Also Published As

Publication number Publication date
US20140031393A1 (en) 2014-01-30
WO2010024451A1 (en) 2010-03-04
EP2318390A1 (en) 2011-05-11
US8969387B2 (en) 2015-03-03
MY152008A (en) 2014-08-15
MX2011001955A (es) 2011-03-29
CO6321166A2 (es) 2011-09-20
CA2735162A1 (en) 2010-03-04
PE20110300A1 (es) 2011-06-16
TW201010993A (en) 2010-03-16
DK2318390T3 (da) 2013-07-08
RS52872B (sr) 2013-12-31
CN102197033B (zh) 2014-07-16
CN102197033A (zh) 2011-09-21
UY32074A (es) 2010-03-26
UA105185C2 (uk) 2014-04-25
CY1114452T1 (el) 2016-10-05
DOP2011000061A (es) 2011-04-15
TWI473798B (zh) 2015-02-21
ME01598B (me) 2014-09-20
EA201170384A1 (ru) 2011-10-31
AU2009284867B2 (en) 2014-08-28
HRP20130653T1 (en) 2013-08-31
HK1157756A1 (en) 2012-07-06
ECSP11010912A (es) 2011-04-29
PT2318390E (pt) 2013-07-10
CL2011000402A1 (es) 2011-07-29
JP5638515B2 (ja) 2014-12-10
AR073136A1 (es) 2010-10-13
IL211335A0 (en) 2011-04-28
CR20110169A (es) 2011-05-16
JO2871B1 (en) 2015-03-15
IL211335A (en) 2013-12-31
KR101629181B1 (ko) 2016-06-13
US8592597B2 (en) 2013-11-26
NZ591793A (en) 2012-11-30
BRPI0917705A2 (pt) 2016-02-16
EP2318390B1 (en) 2013-05-01
US8993598B2 (en) 2015-03-31
MA32647B1 (fr) 2011-09-01
SI2318390T1 (sl) 2013-08-30
PL2318390T3 (pl) 2013-09-30
PE20141174A1 (es) 2014-09-19
ES2423289T3 (es) 2013-09-19
US20110172275A1 (en) 2011-07-14
CA2735162C (en) 2015-06-23
JP2012501296A (ja) 2012-01-19
AU2009284867A1 (en) 2010-03-04
KR20110071067A (ko) 2011-06-28
GEP20135786B (en) 2013-03-11
AU2009284867A2 (en) 2011-04-21
SMT201300085B (it) 2013-09-06
ZA201101774B (en) 2012-06-27
US20100056577A1 (en) 2010-03-04

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Designated state(s): AM AZ BY KZ KG MD TJ TM RU