MA32647B1 - Composés pyrrole - Google Patents

Composés pyrrole

Info

Publication number
MA32647B1
MA32647B1 MA33715A MA33715A MA32647B1 MA 32647 B1 MA32647 B1 MA 32647B1 MA 33715 A MA33715 A MA 33715A MA 33715 A MA33715 A MA 33715A MA 32647 B1 MA32647 B1 MA 32647B1
Authority
MA
Morocco
Prior art keywords
pyrrole compounds
pyrrole
compounds
pyruidyl
substitute
Prior art date
Application number
MA33715A
Other languages
Arabic (ar)
English (en)
Inventor
Haruyuki Nishida
Yasuyoshi Arikawa
Ikuo Fujimori
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41508823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA32647(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of MA32647B1 publication Critical patent/MA32647B1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

L'invention concerne un composé représenté par la formule: dans laquelle A représente un groupe pyridyle ayant au moins un substituant dans lequel R
MA33715A 2008-08-27 2011-03-18 Composés pyrrole MA32647B1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2008218851 2008-08-27
JP2008269099 2008-10-17
PCT/JP2009/065279 WO2010024451A1 (fr) 2008-08-27 2009-08-26 Composés pyrrole

Publications (1)

Publication Number Publication Date
MA32647B1 true MA32647B1 (fr) 2011-09-01

Family

ID=41508823

Family Applications (1)

Application Number Title Priority Date Filing Date
MA33715A MA32647B1 (fr) 2008-08-27 2011-03-18 Composés pyrrole

Country Status (38)

Country Link
US (3) US8592597B2 (fr)
EP (1) EP2318390B1 (fr)
JP (1) JP5638515B2 (fr)
KR (1) KR101629181B1 (fr)
CN (1) CN102197033B (fr)
AR (1) AR073136A1 (fr)
AU (1) AU2009284867B2 (fr)
BR (1) BRPI0917705A2 (fr)
CA (1) CA2735162C (fr)
CL (1) CL2011000402A1 (fr)
CO (1) CO6321166A2 (fr)
CR (1) CR20110169A (fr)
CY (1) CY1114452T1 (fr)
DK (1) DK2318390T3 (fr)
DO (1) DOP2011000061A (fr)
EA (1) EA019741B1 (fr)
EC (1) ECSP11010912A (fr)
ES (1) ES2423289T3 (fr)
GE (1) GEP20135786B (fr)
HR (1) HRP20130653T1 (fr)
IL (1) IL211335A (fr)
JO (1) JO2871B1 (fr)
MA (1) MA32647B1 (fr)
ME (1) ME01598B (fr)
MX (1) MX2011001955A (fr)
MY (1) MY152008A (fr)
NZ (1) NZ591793A (fr)
PE (2) PE20110300A1 (fr)
PL (1) PL2318390T3 (fr)
PT (1) PT2318390E (fr)
RS (1) RS52872B (fr)
SI (1) SI2318390T1 (fr)
SM (1) SMT201300085B (fr)
TW (1) TWI473798B (fr)
UA (1) UA105185C2 (fr)
UY (1) UY32074A (fr)
WO (1) WO2010024451A1 (fr)
ZA (1) ZA201101774B (fr)

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US20110229879A1 (en) * 2010-03-19 2011-09-22 University Of Rochester Methods and compositions for nuclear staining
CN102452979B (zh) * 2010-11-03 2015-04-01 天津药明康德新药开发有限公司 5-氟-3-吡啶磺酰氯的合成方法
CN102863371B (zh) * 2011-07-06 2016-04-13 中国科学院上海有机化学研究所 氟代二氢吡咯或氟代吡咯
US10039813B2 (en) 2012-02-07 2018-08-07 Massachusetts Institute Of Technology Use of antagonists of ghrelin or ghrelin receptor to prevent or treat stress-sensitive psychiatric illness
AR091567A1 (es) 2012-06-27 2015-02-11 Takeda Pharmaceutical Preparacion liquida, metodo, kit de inyeccion
US9487485B2 (en) 2013-02-28 2016-11-08 Takeda Pharmaceutical Company Limited Method for producing sulfonyl chloride compound
WO2014144231A1 (fr) 2013-03-15 2014-09-18 Massachusetts Institute Of Technology Utilisation d'antagonistes de l'hormone de croissance ou de recepteur de l'hormone de croissance pour empecher ou traiter une maladie psychiatrique sensible au stress
KR102084185B1 (ko) * 2013-08-29 2020-03-04 주식회사 대웅제약 테트라히드로사이클로펜타피롤 유도체 및 이의 제조방법
CN105367550A (zh) * 2014-08-11 2016-03-02 江苏柯菲平医药股份有限公司 四氢环戊二烯并[c]吡咯类衍生物、其制备方法及其在医药上的应用
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WO2016138099A1 (fr) 2015-02-24 2016-09-01 Massachusetts Institute Of Technology Utilisation de ghréline ou d'agonistes fonctionnels des récepteurs de la ghréline pour prévenir et traiter une maladie psychiatrique sensible au stress
US10835541B2 (en) 2015-07-30 2020-11-17 Takeda Pharmaceutical Company Limited Tablet
EP3331870B1 (fr) 2015-08-07 2021-06-16 Bayer CropScience Aktiengesellschaft Derives d'heterocyclene condenses 2-(het)aryl-substitues en tant que pesticides
CN106430006B (zh) * 2016-08-18 2018-06-12 国网湖南省电力公司带电作业中心 配电线路移动式绝缘登高作业装置及方法
CN108203430A (zh) * 2016-12-16 2018-06-26 天地人和生物科技有限公司 一种新型可逆性质子泵抑制剂及其制备方法和用途
CA3069563A1 (fr) 2017-07-10 2019-01-17 Takeda Pharmaceutical Company Limited Preparation comprenant du vonoprazan
KR102126576B1 (ko) 2018-09-19 2020-06-24 주식회사 대웅제약 4-메톡시 피롤 유도체의 제조 방법
CN113527536B (zh) * 2020-04-21 2024-03-22 杭州德柯医疗科技有限公司 一种含氟多糖高分子化合物及其制备方法
AU2021293694B2 (en) * 2020-06-17 2023-12-21 Ildong Pharmaceutical Co., Ltd. Novel Acid Secretion Inhibitor and use thereof
EP4074317A1 (fr) 2021-04-14 2022-10-19 Bayer AG Dérivés de phosphore en tant que nouveaux inhibiteurs de sos1
CN113620930B (zh) * 2021-07-12 2022-08-16 南京烁慧医药科技有限公司 一种含磺酰胺结构的化合物及其制备方法和应用、一种药物组合物及应用
CN118541361A (zh) * 2021-12-15 2024-08-23 日东制药株式会社 1-磺酰基吡咯衍生物的新型盐、其制备方法和包括其的药物组合物
WO2023113458A1 (fr) * 2021-12-15 2023-06-22 Ildong Pharmaceutical Co., Ltd. Nouveau sel de dérivé de 1-sulfonyle pyrrole, son procédé de préparation et composition pharmaceutique le comprenant
KR20230102353A (ko) * 2021-12-30 2023-07-07 주식회사 대웅제약 삼중음성유방암의 예방 또는 치료용 약학적 조성물

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Also Published As

Publication number Publication date
CY1114452T1 (el) 2016-10-05
CL2011000402A1 (es) 2011-07-29
ME01598B (me) 2014-09-20
US8993598B2 (en) 2015-03-31
UY32074A (es) 2010-03-26
US20100056577A1 (en) 2010-03-04
DK2318390T3 (da) 2013-07-08
EP2318390B1 (fr) 2013-05-01
SMT201300085B (it) 2013-09-06
DOP2011000061A (es) 2011-04-15
IL211335A (en) 2013-12-31
US8592597B2 (en) 2013-11-26
KR101629181B1 (ko) 2016-06-13
PE20110300A1 (es) 2011-06-16
CN102197033B (zh) 2014-07-16
ZA201101774B (en) 2012-06-27
US20140031393A1 (en) 2014-01-30
PT2318390E (pt) 2013-07-10
UA105185C2 (uk) 2014-04-25
CO6321166A2 (es) 2011-09-20
TW201010993A (en) 2010-03-16
AU2009284867A2 (en) 2011-04-21
BRPI0917705A2 (pt) 2016-02-16
CA2735162A1 (fr) 2010-03-04
CN102197033A (zh) 2011-09-21
AU2009284867A1 (en) 2010-03-04
CA2735162C (fr) 2015-06-23
ECSP11010912A (es) 2011-04-29
ES2423289T3 (es) 2013-09-19
TWI473798B (zh) 2015-02-21
AR073136A1 (es) 2010-10-13
AU2009284867B2 (en) 2014-08-28
WO2010024451A1 (fr) 2010-03-04
US20110172275A1 (en) 2011-07-14
PE20141174A1 (es) 2014-09-19
SI2318390T1 (sl) 2013-08-30
RS52872B (sr) 2013-12-31
GEP20135786B (en) 2013-03-11
HRP20130653T1 (en) 2013-08-31
NZ591793A (en) 2012-11-30
JO2871B1 (en) 2015-03-15
EP2318390A1 (fr) 2011-05-11
HK1157756A1 (en) 2012-07-06
PL2318390T3 (pl) 2013-09-30
JP2012501296A (ja) 2012-01-19
JP5638515B2 (ja) 2014-12-10
MY152008A (en) 2014-08-15
EA019741B1 (ru) 2014-05-30
US8969387B2 (en) 2015-03-03
IL211335A0 (en) 2011-04-28
CR20110169A (es) 2011-05-16
KR20110071067A (ko) 2011-06-28
MX2011001955A (es) 2011-03-29
EA201170384A1 (ru) 2011-10-31

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