AU2001258784A1 - Tyrosine phosphatase inhibitors - Google Patents
Tyrosine phosphatase inhibitorsInfo
- Publication number
- AU2001258784A1 AU2001258784A1 AU2001258784A AU5878401A AU2001258784A1 AU 2001258784 A1 AU2001258784 A1 AU 2001258784A1 AU 2001258784 A AU2001258784 A AU 2001258784A AU 5878401 A AU5878401 A AU 5878401A AU 2001258784 A1 AU2001258784 A1 AU 2001258784A1
- Authority
- AU
- Australia
- Prior art keywords
- tyrosine phosphatase
- phosphatase inhibitors
- inhibitors
- tyrosine
- phosphatase
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C07D207/333—Radicals substituted by oxygen or sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/402—1-aryl substituted, e.g. piretanide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2000154441 | 2000-05-22 | ||
JP2000-154441 | 2000-05-22 | ||
JP2000-247954 | 2000-08-10 | ||
JP2000247954 | 2000-08-10 | ||
PCT/JP2001/004201 WO2001090067A1 (en) | 2000-05-22 | 2001-05-21 | Tyrosine phosphatase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
AU2001258784A1 true AU2001258784A1 (en) | 2001-12-03 |
Family
ID=26592561
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2001258784A Abandoned AU2001258784A1 (en) | 2000-05-22 | 2001-05-21 | Tyrosine phosphatase inhibitors |
Country Status (5)
Country | Link |
---|---|
US (1) | US6911468B2 (en) |
EP (1) | EP1284260A4 (en) |
AU (1) | AU2001258784A1 (en) |
CA (1) | CA2410338A1 (en) |
WO (1) | WO2001090067A1 (en) |
Families Citing this family (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6569853B1 (en) * | 2000-11-06 | 2003-05-27 | Combinatorx, Incorporated | Combinations of chlorpromazine and pentamidine for the treatment of neoplastic disorders |
US7220773B2 (en) | 2001-04-19 | 2007-05-22 | Dainippon Sumitomo Pharma Co., Ltd. | Pyrrole derivative |
GB0212785D0 (en) * | 2002-05-31 | 2002-07-10 | Glaxo Group Ltd | Compounds |
WO2004018455A1 (en) * | 2002-08-23 | 2004-03-04 | Chiron Corporation | Pyrrole based inhibitors of glycogen synthase kinase 3 |
US20040186151A1 (en) * | 2003-02-12 | 2004-09-23 | Mjalli Adnan M.M. | Substituted azole derivatives as therapeutic agents |
CA2514363A1 (en) * | 2003-02-12 | 2004-08-26 | Transtech Pharma, Inc. | Substituted azole derivatives as therapeutic agents |
MXPA06000539A (en) * | 2003-07-15 | 2006-03-30 | Dainippon Sumitomo Pharma Co | Novel heteroaryl derivative. |
US20050054708A1 (en) * | 2003-07-28 | 2005-03-10 | Nichols Matthew James | Combinations of drugs for the treatment of neoplasms |
WO2005020913A2 (en) * | 2003-08-25 | 2005-03-10 | Combinatorx, Incorporated | Formulations, conjugates, and combinations of drugs for the treatment of neoplasms |
US20050100508A1 (en) * | 2003-11-12 | 2005-05-12 | Nichols M. J. | Methods for identifying drug combinations for the treatment of proliferative diseases |
US20050158320A1 (en) * | 2003-11-12 | 2005-07-21 | Nichols M. J. | Combinations for the treatment of proliferative diseases |
ZA200605526B (en) * | 2004-02-12 | 2007-11-28 | Transtech Pharma Inc | Substituted azole derivatives, compositions and methods of use |
ATE493973T1 (en) | 2004-06-04 | 2011-01-15 | Teva Pharma | PHARMACEUTICAL COMPOSITION CONTAINING IRBESARTAN |
EP1803709B1 (en) | 2004-09-30 | 2013-01-02 | Takeda Pharmaceutical Company Limited | Proton pump inhibitors |
EP1837329A4 (en) * | 2005-01-14 | 2009-08-05 | Dainippon Sumitomo Pharma Co | Novel heteroaryl derivative |
WO2006092449A2 (en) * | 2005-03-02 | 2006-09-08 | Metanomics Gmbh | Process for the production of fine chemicals |
CA2617557A1 (en) * | 2005-08-04 | 2007-02-15 | Sirtris Pharmaceuticals, Inc. | Benzimidazole derivatives as sirtuin modulators |
EP1919865B1 (en) | 2005-08-30 | 2011-04-06 | Takeda Pharmaceutical Company Limited | 1-heterocyclylsulfonyl, 2-aminomethyl, 5- (hetero-) aryl substituted 1-h-pyrrole derivatives as acid secretion inhibitors |
US20070161006A1 (en) * | 2006-01-10 | 2007-07-12 | Vita Genomics, Inc. | Single nucleotide polymorphisms in protein-tyrosine phosphatase receptor-type delta for the diagnosis of susceptibility to infection and asthma |
WO2007089857A2 (en) | 2006-01-30 | 2007-08-09 | Transtech Pharma, Inc. | Substituted imidazole derivatives and their use as ptpase inhibitors |
US8933105B2 (en) | 2007-02-28 | 2015-01-13 | Takeda Pharmaceutical Company Limited | Pyrrole compounds |
TW200916472A (en) | 2007-06-20 | 2009-04-16 | Sirtris Pharmaceuticals Inc | Sirtuin modulating compounds |
US8969387B2 (en) | 2008-08-27 | 2015-03-03 | Takeda Pharmaceutical Company Limited | Pyrrole compounds |
CN102648183B (en) * | 2009-10-07 | 2015-12-02 | 卡罗生物股份公司 | As the substituted pyrazolecarboxylic of estrogen receptor ligands |
US20120225846A1 (en) | 2011-03-02 | 2012-09-06 | Bioenergenix | Heterocyclic compounds for the inhibition of pask |
GB201113538D0 (en) | 2011-08-04 | 2011-09-21 | Karobio Ab | Novel estrogen receptor ligands |
US9073881B2 (en) | 2011-09-23 | 2015-07-07 | Hoffmann-La Roche Inc. | Benzoic acid derivatives |
WO2016074696A1 (en) * | 2014-11-10 | 2016-05-19 | Givaudan Ag | Perfume ingredients and perfume preparations containing same |
GB201706806D0 (en) | 2017-04-28 | 2017-06-14 | Sentinel Oncology Ltd | Pharmaceutical compounds |
CN107935863A (en) * | 2017-11-30 | 2018-04-20 | 厦门海乐景生化有限公司 | The synthetic method of the critical materials compound C of Elagolix |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3168529A (en) * | 1962-06-14 | 1965-02-02 | Parke Davis & Co | 1-(p-lower alkanoylphenyl)-5-arylpyrrole-2-propionic acid compounds |
DK148576A (en) * | 1975-04-18 | 1976-10-19 | Boehringer Mannheim Gmbh | PHENYLALCANCARBONIC ACID DERIVATIVES AND PROCEDURE FOR THEIR PREPARATION |
IL92915A0 (en) | 1989-01-05 | 1990-09-17 | Ciba Geigy Ag | Certain pyrrolylphenyl-substituted hydroxamic acid derivatives |
US5096919A (en) * | 1989-01-05 | 1992-03-17 | Ciba-Geigy Corporation | Pyrrolylphenyl-substituted hydroxamic acid derivatives |
US5385929A (en) * | 1994-05-04 | 1995-01-31 | Warner-Lambert Company | [(Hydroxyphenylamino) carbonyl] pyrroles |
ATE255090T1 (en) * | 1996-08-01 | 2003-12-15 | Merckle Gmbh | ACYLPYRROLDICARBONONIC ACIDS AND ACYLINDOLICARBONONIC ACIDS AND THEIR DERIVATIVES AS INHIBITORS OF CYTOSOLIC PHOSPHOLIPASE A2 |
AU2713799A (en) | 1998-03-12 | 1999-09-27 | Novo Nordisk A/S | Modulators of protein tyrosine phosphatases (ptpases) |
ATE228120T1 (en) | 1998-05-12 | 2002-12-15 | Wyeth Corp | BIPHENYLSULFONYLARYL CARBOXYLIC ACIDS USED FOR TREATING INSULIN RESISTANCE AND HYPERGLYCEMIA |
AU4072799A (en) * | 1998-05-12 | 1999-12-13 | American Home Products Corporation | 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia |
JP2002514635A (en) | 1998-05-12 | 2002-05-21 | アメリカン・ホーム・プロダクツ・コーポレイション | Biphenyloxo-acetic acid useful for treating insulin resistance and hyperglycemia |
US7314888B1 (en) * | 1998-11-05 | 2008-01-01 | Toyama Chemical Co., Ltd. | Compounds and medicinal use thereof |
US7220773B2 (en) | 2001-04-19 | 2007-05-22 | Dainippon Sumitomo Pharma Co., Ltd. | Pyrrole derivative |
-
2001
- 2001-05-21 AU AU2001258784A patent/AU2001258784A1/en not_active Abandoned
- 2001-05-21 US US10/276,674 patent/US6911468B2/en not_active Expired - Fee Related
- 2001-05-21 EP EP01932153A patent/EP1284260A4/en not_active Withdrawn
- 2001-05-21 CA CA002410338A patent/CA2410338A1/en not_active Abandoned
- 2001-05-21 WO PCT/JP2001/004201 patent/WO2001090067A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
US20030144338A1 (en) | 2003-07-31 |
EP1284260A4 (en) | 2004-03-31 |
EP1284260A1 (en) | 2003-02-19 |
CA2410338A1 (en) | 2001-11-29 |
WO2001090067A1 (en) | 2001-11-29 |
US6911468B2 (en) | 2005-06-28 |
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