AR073136A1 - Compuestos de pirrol - Google Patents

Compuestos de pirrol

Info

Publication number
AR073136A1
AR073136A1 ARP090103278A ARP090103278A AR073136A1 AR 073136 A1 AR073136 A1 AR 073136A1 AR P090103278 A ARP090103278 A AR P090103278A AR P090103278 A ARP090103278 A AR P090103278A AR 073136 A1 AR073136 A1 AR 073136A1
Authority
AR
Argentina
Prior art keywords
halogen
optionally substituted
group optionally
hydrogen atom
alkyl group
Prior art date
Application number
ARP090103278A
Other languages
English (en)
Inventor
Yasuyoshi Arikawa
Haruyuki Nishida
Ikuo Fujimori
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41508823&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR073136(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of AR073136A1 publication Critical patent/AR073136A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente se refiere a un compuesto representado por la formula (1) en donde A es grupo piridilo que tiene al menos un sustituyente de formula (2) o (3) en donde R1, R2 y R3 son cada uno un átomo de hidrogeno, de halogeno, un grupo alquilo C1-6 opcionalmente sustituido con halogeno o un grupo alcoxi C1-6 opcionalmente sustituido con halogeno; R4 y R6 son cada uno un átomo de hidrogeno, de halogeno o un grupo alquilo C1-6, opcionalmente sustituido con halogeno; R5 es un átomo de hidrogeno, de halogeno, un grupo alquilo C1-6 opcionalmente sustituido con halogeno o un grupo alcoxi C1-6 opcionalmente sustituido con halogeno; y R7 es un átomo de hidrogeno o un grupo alquilo C1-6 opcionalmente sustituido con halogeno; o una de sus sales o una composicion farmacéutica que los contiene, utiles para suprimir la secrecion ácida.
ARP090103278A 2008-08-27 2009-08-26 Compuestos de pirrol AR073136A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2008218851 2008-08-27
JP2008269099 2008-10-17

Publications (1)

Publication Number Publication Date
AR073136A1 true AR073136A1 (es) 2010-10-13

Family

ID=41508823

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090103278A AR073136A1 (es) 2008-08-27 2009-08-26 Compuestos de pirrol

Country Status (39)

Country Link
US (3) US8969387B2 (es)
EP (1) EP2318390B1 (es)
JP (1) JP5638515B2 (es)
KR (1) KR101629181B1 (es)
CN (1) CN102197033B (es)
AR (1) AR073136A1 (es)
AU (1) AU2009284867B2 (es)
BR (1) BRPI0917705A2 (es)
CA (1) CA2735162C (es)
CL (1) CL2011000402A1 (es)
CO (1) CO6321166A2 (es)
CR (1) CR20110169A (es)
CY (1) CY1114452T1 (es)
DK (1) DK2318390T3 (es)
DO (1) DOP2011000061A (es)
EA (1) EA019741B1 (es)
EC (1) ECSP11010912A (es)
ES (1) ES2423289T3 (es)
GE (1) GEP20135786B (es)
HK (1) HK1157756A1 (es)
HR (1) HRP20130653T1 (es)
IL (1) IL211335A (es)
JO (1) JO2871B1 (es)
MA (1) MA32647B1 (es)
ME (1) ME01598B (es)
MX (1) MX2011001955A (es)
MY (1) MY152008A (es)
NZ (1) NZ591793A (es)
PE (2) PE20141174A1 (es)
PL (1) PL2318390T3 (es)
PT (1) PT2318390E (es)
RS (1) RS52872B (es)
SI (1) SI2318390T1 (es)
SM (1) SMT201300085B (es)
TW (1) TWI473798B (es)
UA (1) UA105185C2 (es)
UY (1) UY32074A (es)
WO (1) WO2010024451A1 (es)
ZA (1) ZA201101774B (es)

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CN102452979B (zh) * 2010-11-03 2015-04-01 天津药明康德新药开发有限公司 5-氟-3-吡啶磺酰氯的合成方法
CN102863371B (zh) * 2011-07-06 2016-04-13 中国科学院上海有机化学研究所 氟代二氢吡咯或氟代吡咯
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US9724396B2 (en) 2013-03-15 2017-08-08 Massachusetts Institute Of Technology Use of antagonists of growth hormone or growth hormone receptor to prevent or treat stress-sensitive psychiatric illness
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WO2016138099A1 (en) 2015-02-24 2016-09-01 Massachusetts Institute Of Technology Use of ghrelin or functional ghrelin receptor agonists to prevent and treat stress-sensitive psychiatric illness
TWI710379B (zh) 2015-07-30 2020-11-21 日商武田藥品工業股份有限公司 錠劑
AU2016307233B2 (en) 2015-08-07 2020-12-24 Bayer Cropscience Aktiengesellschaft 2-(het)aryl-substituted condensed heterocyclic derivatives as pest control agents
CN106430006B (zh) * 2016-08-18 2018-06-12 国网湖南省电力公司带电作业中心 配电线路移动式绝缘登高作业装置及方法
CN108203430A (zh) * 2016-12-16 2018-06-26 天地人和生物科技有限公司 一种新型可逆性质子泵抑制剂及其制备方法和用途
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CN113527536B (zh) * 2020-04-21 2024-03-22 杭州德柯医疗科技有限公司 一种含氟多糖高分子化合物及其制备方法
CN115884968B (zh) * 2020-06-17 2024-06-21 日东制药株式会社 新型酸分泌抑制剂及其用途
EP4074317A1 (en) 2021-04-14 2022-10-19 Bayer AG Phosphorus derivatives as novel sos1 inhibitors
CN113620930B (zh) * 2021-07-12 2022-08-16 南京烁慧医药科技有限公司 一种含磺酰胺结构的化合物及其制备方法和应用、一种药物组合物及应用
CN118401510A (zh) * 2021-12-15 2024-07-26 日东制药株式会社 1-磺酰基吡咯衍生物的新颖盐类、其制备方法及包含其的药物组合物
WO2023113474A1 (ko) * 2021-12-15 2023-06-22 일동제약(주) 1-설포닐 피롤 유도체의 신규 염, 이의 제조 방법 및 이를 포함하는 약학 조성물
KR20230102353A (ko) * 2021-12-30 2023-07-07 주식회사 대웅제약 삼중음성유방암의 예방 또는 치료용 약학적 조성물

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Also Published As

Publication number Publication date
KR20110071067A (ko) 2011-06-28
MX2011001955A (es) 2011-03-29
MA32647B1 (fr) 2011-09-01
UA105185C2 (uk) 2014-04-25
JP2012501296A (ja) 2012-01-19
NZ591793A (en) 2012-11-30
US8993598B2 (en) 2015-03-31
ZA201101774B (en) 2012-06-27
SI2318390T1 (sl) 2013-08-30
CA2735162C (en) 2015-06-23
US20100056577A1 (en) 2010-03-04
CA2735162A1 (en) 2010-03-04
ME01598B (me) 2014-09-20
CL2011000402A1 (es) 2011-07-29
IL211335A0 (en) 2011-04-28
IL211335A (en) 2013-12-31
CN102197033B (zh) 2014-07-16
EA019741B1 (ru) 2014-05-30
JP5638515B2 (ja) 2014-12-10
ES2423289T3 (es) 2013-09-19
TWI473798B (zh) 2015-02-21
PT2318390E (pt) 2013-07-10
EP2318390A1 (en) 2011-05-11
MY152008A (en) 2014-08-15
GEP20135786B (en) 2013-03-11
CR20110169A (es) 2011-05-16
UY32074A (es) 2010-03-26
JO2871B1 (en) 2015-03-15
ECSP11010912A (es) 2011-04-29
US20140031393A1 (en) 2014-01-30
AU2009284867A2 (en) 2011-04-21
US8592597B2 (en) 2013-11-26
DK2318390T3 (da) 2013-07-08
TW201010993A (en) 2010-03-16
PE20110300A1 (es) 2011-06-16
AU2009284867A1 (en) 2010-03-04
EA201170384A1 (ru) 2011-10-31
BRPI0917705A2 (pt) 2016-02-16
HRP20130653T1 (en) 2013-08-31
CO6321166A2 (es) 2011-09-20
AU2009284867B2 (en) 2014-08-28
CY1114452T1 (el) 2016-10-05
PE20141174A1 (es) 2014-09-19
EP2318390B1 (en) 2013-05-01
US20110172275A1 (en) 2011-07-14
HK1157756A1 (en) 2012-07-06
SMT201300085B (it) 2013-09-06
PL2318390T3 (pl) 2013-09-30
WO2010024451A1 (en) 2010-03-04
DOP2011000061A (es) 2011-04-15
RS52872B (en) 2013-12-31
US8969387B2 (en) 2015-03-03
CN102197033A (zh) 2011-09-21
KR101629181B1 (ko) 2016-06-13

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