DE69930328T2 - Dimere Pyrrolobenzodiazepine - Google Patents
Dimere Pyrrolobenzodiazepine Download PDFInfo
- Publication number
- DE69930328T2 DE69930328T2 DE69930328T DE69930328T DE69930328T2 DE 69930328 T2 DE69930328 T2 DE 69930328T2 DE 69930328 T DE69930328 T DE 69930328T DE 69930328 T DE69930328 T DE 69930328T DE 69930328 T2 DE69930328 T2 DE 69930328T2
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- Prior art keywords
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- mmol
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- mice
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- Expired - Lifetime
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Classifications
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- C—CHEMISTRY; METALLURGY
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- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
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| GBGB9818733.9A GB9818733D0 (en) | 1998-08-27 | 1998-08-27 | Compounds |
| HN9818733 | 1998-08-27 | ||
| GBGB9901929.1A GB9901929D0 (en) | 1999-01-28 | 1999-01-28 | Compounds |
| GB9901929 | 1999-01-28 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE69930328D1 DE69930328D1 (de) | 2006-05-11 |
| DE69930328T2 true DE69930328T2 (de) | 2006-12-14 |
Family
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| Application Number | Title | Priority Date | Filing Date |
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| DE69907977T Expired - Lifetime DE69907977T2 (de) | 1998-08-27 | 1999-08-27 | Pyrrolobenzodiazepine |
| DE69925133T Expired - Lifetime DE69925133T2 (de) | 1998-08-27 | 1999-08-27 | Pyrrolobenzodiazepine |
| DE69930328T Expired - Lifetime DE69930328T2 (de) | 1998-08-27 | 1999-08-27 | Dimere Pyrrolobenzodiazepine |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE69907977T Expired - Lifetime DE69907977T2 (de) | 1998-08-27 | 1999-08-27 | Pyrrolobenzodiazepine |
| DE69925133T Expired - Lifetime DE69925133T2 (de) | 1998-08-27 | 1999-08-27 | Pyrrolobenzodiazepine |
Country Status (12)
| Country | Link |
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| US (3) | US7049311B1 (enExample) |
| EP (3) | EP1109812B1 (enExample) |
| JP (1) | JP4824165B2 (enExample) |
| AT (3) | ATE294803T1 (enExample) |
| AU (1) | AU757510C (enExample) |
| CA (1) | CA2341471C (enExample) |
| DE (3) | DE69907977T2 (enExample) |
| DK (3) | DK1413582T3 (enExample) |
| ES (3) | ES2199200T3 (enExample) |
| NZ (1) | NZ510493A (enExample) |
| PT (3) | PT1109812E (enExample) |
| WO (1) | WO2000012508A2 (enExample) |
Families Citing this family (196)
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| GB9818731D0 (en) * | 1998-08-27 | 1998-10-21 | Univ Portsmouth | Compounds |
| GB0226593D0 (en) * | 2002-11-14 | 2002-12-24 | Consultants Ltd | Compounds |
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