TWI316930B - 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands - Google Patents

3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands Download PDF

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TWI316930B
TWI316930B TW091107670A TW91107670A TWI316930B TW I316930 B TWI316930 B TW I316930B TW 091107670 A TW091107670 A TW 091107670A TW 91107670 A TW91107670 A TW 91107670A TW I316930 B TWI316930 B TW I316930B
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Chinese (zh)
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G Taveras Arthur
J Aki Cynthia
W Bond Richard
Chao Jianping
Dwyer Michael
A Ferreira Johan
Chao Jianhua
Yu Younong
J Baldwin John
Kaiser Bernd
Li Ge
j merritt Robert
H Nelson Kingsley Jr
L Rokosz Laura
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Schering Corp
Pharmacopeia Drug Discovery
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TW091107670A 2001-04-16 2002-04-16 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands TWI316930B (en)

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US28402601P 2001-04-16 2001-04-16

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TW096102669A TW200736196A (en) 2001-04-16 2002-04-16 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands

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US20040106794A1 (en) 2001-04-16 2004-06-03 Schering Corporation 3,4-Di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands
JP2005505595A (ja) 2001-10-12 2005-02-24 シェーリング　コーポレイション Ｃｘｃ−ケモカインレセプターアンタゴニストとしての３，４−二置換マレイミド化合物
US8246969B2 (en) 2001-11-16 2012-08-21 Skinmedica, Inc. Compositions containing aromatic aldehydes and their use in treatments
US6878709B2 (en) 2002-01-04 2005-04-12 Schering Corporation 3,4-di-substituted pyridazinediones as CXC chemokine receptor antagonists
JP4733350B2 (ja) * 2002-03-18 2011-07-27 シェーリング コーポレイション ケモカイン媒介疾患の併用治療
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ATE422203T1 (de) 2002-10-09 2009-02-15 Schering Corp Thiadiazoldioxide und thiadiazoloxide als cxc- und cc-chemokinrezeptor liganden
GB0302094D0 (en) 2003-01-29 2003-02-26 Pharmagene Lab Ltd EP4 receptor antagonists
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DE602004025458D1 (de) 2003-04-18 2010-03-25 Schering Corp SYNTHESE VON 2-HYDROXY-N,N-DIMETHYL-3-ii2-i1(R)-(5-METHYL-2-FURANYL)PROPYL AMINO -3,4-DIOXO-1-CYCLOBUTEN-1-YL AMINO BENZAMID
PL1651612T3 (pl) 2003-07-22 2012-09-28 Astex Therapeutics Ltd Związki 3,4-pochodne 1h-pirazolu i ich zastosowanie jako kinazy zależne od cyklin (cdk) i modulatory kinazy syntazy glikogenu-3 (gsk-3)
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