TW200745045A - Imidazole based LXR modulators - Google Patents
Imidazole based LXR modulatorsInfo
- Publication number
- TW200745045A TW200745045A TW095123162A TW95123162A TW200745045A TW 200745045 A TW200745045 A TW 200745045A TW 095123162 A TW095123162 A TW 095123162A TW 95123162 A TW95123162 A TW 95123162A TW 200745045 A TW200745045 A TW 200745045A
- Authority
- TW
- Taiwan
- Prior art keywords
- compounds
- lxr modulators
- imidazole based
- based lxr
- modulators
- Prior art date
Links
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- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
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- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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US69437205P | 2005-06-27 | 2005-06-27 | |
US73612005P | 2005-11-10 | 2005-11-10 |
Publications (1)
Publication Number | Publication Date |
---|---|
TW200745045A true TW200745045A (en) | 2007-12-16 |
Family
ID=37309323
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW095123162A TW200745045A (en) | 2005-06-27 | 2006-06-27 | Imidazole based LXR modulators |
TW095123212A TWI388323B (zh) | 2005-06-27 | 2006-06-27 | 基於吡唑之肝x受體(lxr)調節劑 |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
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TW095123212A TWI388323B (zh) | 2005-06-27 | 2006-06-27 | 基於吡唑之肝x受體(lxr)調節劑 |
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US (3) | US8703805B2 (zh) |
EP (2) | EP1910307A1 (zh) |
JP (2) | JP5244589B2 (zh) |
KR (2) | KR101363278B1 (zh) |
AR (2) | AR054521A1 (zh) |
AU (2) | AU2006261845C1 (zh) |
BR (1) | BRPI0612287A8 (zh) |
CA (2) | CA2613522A1 (zh) |
ES (1) | ES2525217T3 (zh) |
IL (1) | IL188239A0 (zh) |
MX (1) | MX2008000141A (zh) |
MY (1) | MY152162A (zh) |
NO (1) | NO20080391L (zh) |
NZ (1) | NZ564916A (zh) |
PE (2) | PE20070105A1 (zh) |
SG (1) | SG162804A1 (zh) |
TW (2) | TW200745045A (zh) |
WO (2) | WO2007002559A1 (zh) |
Families Citing this family (122)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE602004000260T2 (de) | 2003-07-22 | 2006-08-24 | Arena Pharmaceuticals, Inc., San Diego | Diaryl- und arylheteroarylharnstoffderivate als modulatoren des 5-ht2a-serotoninrezeptors, die sich zur prophylaxe und behandlung von damit im zusammenhang stehenden erkrankungen eignen |
PE20061130A1 (es) | 2004-11-19 | 2007-01-05 | Arena Pharm Inc | Derivados de 3-fenil-pirazol como moduladores del receptor de serotonina 5-ht2a |
CA2613522A1 (en) | 2005-06-27 | 2007-01-04 | Exelixis, Inc. | Imidazole based lxr modulators |
AU2013200480B2 (en) * | 2006-02-28 | 2016-06-09 | Dart Neuroscience (Cayman) Ltd. | Therapeutic compounds |
ES2462240T3 (es) | 2006-02-28 | 2014-05-22 | Dart Neuroscience (Cayman) Ltd | Piperazinas terapéuticas como inhibidores de PDE4 |
AU2007221020B9 (en) * | 2006-02-28 | 2013-04-04 | Dart Neuroscience (Cayman) Ltd. | Therapeutic compounds |
EP3395816A1 (en) | 2006-05-18 | 2018-10-31 | Arena Pharmaceuticals, Inc. | Ethers, secondary amines and derivatives thereof as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto |
CA2646081C (en) | 2006-05-18 | 2017-06-27 | Arena Pharmaceuticals, Inc. | Crystalline forms and processes for the preparation of phenyl-pyrazoles useful as modulators of the 5-ht2a serotonin receptor |
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2006
- 2006-06-26 CA CA002613522A patent/CA2613522A1/en not_active Abandoned
- 2006-06-26 SG SG201004273-7A patent/SG162804A1/en unknown
- 2006-06-26 EP EP06785558A patent/EP1910307A1/en not_active Withdrawn
- 2006-06-26 KR KR1020087001879A patent/KR101363278B1/ko not_active IP Right Cessation
- 2006-06-26 ES ES06785562.7T patent/ES2525217T3/es active Active
- 2006-06-26 US US11/993,806 patent/US8703805B2/en active Active
- 2006-06-26 US US11/993,529 patent/US8569352B2/en active Active
- 2006-06-26 KR KR1020087001957A patent/KR20080028964A/ko not_active Application Discontinuation
- 2006-06-26 JP JP2008519445A patent/JP5244589B2/ja active Active
- 2006-06-26 WO PCT/US2006/024749 patent/WO2007002559A1/en active Application Filing
- 2006-06-26 EP EP06785562.7A patent/EP1910308B1/en active Active
- 2006-06-26 WO PCT/US2006/024757 patent/WO2007002563A1/en active Application Filing
- 2006-06-26 BR BRPI0612287A patent/BRPI0612287A8/pt not_active IP Right Cessation
- 2006-06-26 AU AU2006261845A patent/AU2006261845C1/en not_active Ceased
- 2006-06-26 MX MX2008000141A patent/MX2008000141A/es active IP Right Grant
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- 2006-06-26 AU AU2006261841A patent/AU2006261841B8/en not_active Ceased
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