SK287869B6 - Beta-carboline pharmaceutical compositions - Google Patents

Beta-carboline pharmaceutical compositions Download PDF

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Publication number
SK287869B6
SK287869B6 SK173-2002A SK1732002A SK287869B6 SK 287869 B6 SK287869 B6 SK 287869B6 SK 1732002 A SK1732002 A SK 1732002A SK 287869 B6 SK287869 B6 SK 287869B6
Authority
SK
Slovakia
Prior art keywords
formulation
amount
active compound
weight
present
Prior art date
Application number
SK173-2002A
Other languages
English (en)
Slovak (sk)
Other versions
SK1732002A3 (en
Inventor
Peter L. Oren
Neil R. Anderson
Martha A. Kral
Original Assignee
Icos Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22519593&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK287869(B6) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Icos Corporation filed Critical Icos Corporation
Publication of SK1732002A3 publication Critical patent/SK1732002A3/sk
Publication of SK287869B6 publication Critical patent/SK287869B6/sk

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SK173-2002A 1999-08-03 2000-04-26 Beta-carboline pharmaceutical compositions SK287869B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14692499P 1999-08-03 1999-08-03
PCT/US2000/011130 WO2001008686A1 (en) 1999-08-03 2000-04-26 Beta-carboline pharmaceutical compositions

Publications (2)

Publication Number Publication Date
SK1732002A3 SK1732002A3 (en) 2002-05-09
SK287869B6 true SK287869B6 (sk) 2012-02-03

Family

ID=22519593

Family Applications (1)

Application Number Title Priority Date Filing Date
SK173-2002A SK287869B6 (sk) 1999-08-03 2000-04-26 Beta-carboline pharmaceutical compositions

Country Status (29)

Country Link
US (2) US7182958B1 (cs)
EP (3) EP1200091B1 (cs)
JP (2) JP2003505509A (cs)
KR (2) KR100738861B1 (cs)
CN (1) CN1213754C (cs)
AT (1) ATE399554T1 (cs)
AU (2) AU4491200A (cs)
BR (1) BR0012863A (cs)
CA (1) CA2379948C (cs)
CZ (1) CZ304624B6 (cs)
DE (1) DE60039357D1 (cs)
DK (1) DK1200090T3 (cs)
DZ (1) DZ3179A1 (cs)
EA (1) EA004872B1 (cs)
ES (2) ES2310166T3 (cs)
HK (1) HK1044277B (cs)
HR (1) HRP20020090B1 (cs)
HU (1) HU230660B1 (cs)
IL (2) IL147641A0 (cs)
MX (1) MXPA02001196A (cs)
NO (1) NO321649B1 (cs)
NZ (1) NZ516616A (cs)
PL (1) PL199137B1 (cs)
PT (1) PT1200090E (cs)
SI (1) SI1200090T1 (cs)
SK (1) SK287869B6 (cs)
UA (1) UA72922C2 (cs)
WO (2) WO2001008686A1 (cs)
ZA (1) ZA200200823B (cs)

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Also Published As

Publication number Publication date
CZ2002386A3 (cs) 2002-07-17
CZ304624B6 (cs) 2014-08-13
HK1044277B (en) 2014-02-28
PL199137B1 (pl) 2008-08-29
JP2010163464A (ja) 2010-07-29
EA004872B1 (ru) 2004-08-26
HRP20020090B1 (hr) 2014-03-28
NO20020532D0 (no) 2002-02-01
ATE399554T1 (de) 2008-07-15
PL353304A1 (en) 2003-11-03
US6841167B1 (en) 2005-01-11
CA2379948A1 (en) 2001-02-08
HU230660B1 (hu) 2017-06-28
WO2001008687A1 (en) 2001-02-08
EP1200091A1 (en) 2002-05-02
CN1213754C (zh) 2005-08-10
EP1200090B1 (en) 2013-09-11
SK1732002A3 (en) 2002-05-09
DE60039357D1 (de) 2008-08-14
HUP0202513A3 (en) 2004-06-28
EP1200091B1 (en) 2008-07-02
AU4490900A (en) 2001-02-19
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WO2001008686A1 (en) 2001-02-08
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BR0012863A (pt) 2002-04-16
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IL147641A (en) 2007-12-03
DZ3179A1 (fr) 2001-02-08
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UA72922C2 (uk) 2005-05-16
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NO321649B1 (no) 2006-06-19
PT1200090E (pt) 2013-11-25
CN1365282A (zh) 2002-08-21
ZA200200823B (en) 2003-04-30
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EP2338491A2 (en) 2011-06-29
AU4491200A (en) 2001-02-19
SI1200090T1 (sl) 2013-12-31
HRP20020090A2 (en) 2003-12-31
KR20020014843A (ko) 2002-02-25
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NO20020532L (no) 2002-03-26
EP1200090A1 (en) 2002-05-02

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Effective date: 20091214

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Expiry date: 20200426