SI9010243B - Substituirani 1,3-oksatiolani z antivirusnimi lastnostmi - Google Patents

Substituirani 1,3-oksatiolani z antivirusnimi lastnostmi Download PDF

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Publication number
SI9010243B
SI9010243B SI9010243A SI9010243A SI9010243B SI 9010243 B SI9010243 B SI 9010243B SI 9010243 A SI9010243 A SI 9010243A SI 9010243 A SI9010243 A SI 9010243A SI 9010243 B SI9010243 B SI 9010243B
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SI
Slovenia
Prior art keywords
oxathiolane
compound
formula
group
hydroxymethyl
Prior art date
Application number
SI9010243A
Other languages
English (en)
Slovenian (sl)
Other versions
SI9010243A (en
Inventor
Bernard Belleau
Pierette Belleau
Nghe Nguyen-Ba
Original Assignee
Biochem Pharma Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25678044&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI9010243(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Biochem Pharma Inc. filed Critical Biochem Pharma Inc.
Priority claimed from CA002152269A external-priority patent/CA2152269C/en
Publication of SI9010243A publication Critical patent/SI9010243A/sl
Publication of SI9010243B publication Critical patent/SI9010243B/sl

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D327/02—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
    • C07D327/04—Five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
    • C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D411/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/40—Heterocyclic compounds containing purine ring systems with halogen atoms or perhalogeno-alkyl radicals directly attached in position 2 or 6
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Saccharide Compounds (AREA)
SI9010243A 1989-02-08 1990-02-08 Substituirani 1,3-oksatiolani z antivirusnimi lastnostmi SI9010243B (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US07/308,101 US5047407A (en) 1989-02-08 1989-02-08 2-substituted-5-substituted-1,3-oxathiolanes with antiviral properties
YU24390A YU48840B (sh) 1989-02-08 1990-02-08 Postupak za dobijanje substituisanih 1,3-oksatiolana sa antivirusnim osobinama
CA002152269A CA2152269C (en) 1989-02-08 1992-12-21 Process for preparing substituted 1,3-oxathiolanes with antiviral properties

Publications (2)

Publication Number Publication Date
SI9010243A SI9010243A (en) 1996-10-31
SI9010243B true SI9010243B (sl) 1998-08-31

Family

ID=25678044

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9010243A SI9010243B (sl) 1989-02-08 1990-02-08 Substituirani 1,3-oksatiolani z antivirusnimi lastnostmi

Country Status (35)

Country Link
US (1) US5047407A (de)
EP (2) EP0711771B1 (de)
JP (4) JP2644357B2 (de)
KR (1) KR960007531B1 (de)
CN (1) CN1033640C (de)
AP (1) AP136A (de)
AT (2) ATE254125T1 (de)
AU (1) AU630913B2 (de)
CA (1) CA2009637C (de)
CY (1) CY2036A (de)
CZ (1) CZ282720B6 (de)
DE (3) DE69034119T2 (de)
DK (2) DK0711771T3 (de)
ES (2) ES2206476T3 (de)
FI (1) FI98065C (de)
GR (1) GR3019919T3 (de)
HK (1) HK51997A (de)
HR (1) HRP940040B1 (de)
HU (2) HU208134B (de)
IE (1) IE72184B1 (de)
IL (1) IL93318A (de)
LU (1) LU88809I2 (de)
MX (1) MX19437A (de)
NL (1) NL960025I2 (de)
NO (2) NO179518C (de)
NZ (1) NZ232421A (de)
OA (1) OA09193A (de)
PL (1) PL164785B1 (de)
PT (1) PT93094B (de)
RU (1) RU2092485C1 (de)
SG (2) SG77215A1 (de)
SI (1) SI9010243B (de)
SK (1) SK279175B6 (de)
YU (1) YU48840B (de)
ZA (1) ZA90943B (de)

Families Citing this family (151)

* Cited by examiner, † Cited by third party
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CN1044817A (zh) 1990-08-22
HU208134B (en) 1993-08-30
ATE254125T1 (de) 2003-11-15
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ZA90943B (en) 1990-10-31
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FI98065B (fi) 1996-12-31
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