NO330424B1 - Nukleosidderivater, fremstilling av slike, farmasoytiske preparater omfattende slike, slike forbindelser for behandling av sykdommer samt anvendelse av slike for fremstilling av preparater for behandling av sykdom - Google Patents
Nukleosidderivater, fremstilling av slike, farmasoytiske preparater omfattende slike, slike forbindelser for behandling av sykdommer samt anvendelse av slike for fremstilling av preparater for behandling av sykdom Download PDFInfo
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- NO330424B1 NO330424B1 NO20052304A NO20052304A NO330424B1 NO 330424 B1 NO330424 B1 NO 330424B1 NO 20052304 A NO20052304 A NO 20052304A NO 20052304 A NO20052304 A NO 20052304A NO 330424 B1 NO330424 B1 NO 330424B1
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- HZCAHMRRMINHDJ-DBRKOABJSA-N ribavirin Natural products O[C@@H]1[C@H](O)[C@@H](CO)O[C@H]1N1N=CN=C1 HZCAHMRRMINHDJ-DBRKOABJSA-N 0.000 description 1
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- HPALAKNZSZLMCH-UHFFFAOYSA-M sodium;chloride;hydrate Chemical compound O.[Na+].[Cl-] HPALAKNZSZLMCH-UHFFFAOYSA-M 0.000 description 1
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- YLQBMQCUIZJEEH-UHFFFAOYSA-N tetrahydrofuran Natural products C=1C=COC=1 YLQBMQCUIZJEEH-UHFFFAOYSA-N 0.000 description 1
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- VZCYOOQTPOCHFL-UHFFFAOYSA-N trans-butenedioic acid Natural products OC(=O)C=CC(O)=O VZCYOOQTPOCHFL-UHFFFAOYSA-N 0.000 description 1
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- CYRMSUTZVYGINF-UHFFFAOYSA-N trichlorofluoromethane Chemical compound FC(Cl)(Cl)Cl CYRMSUTZVYGINF-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/06—Pyrimidine radicals
- C07H19/073—Pyrimidine radicals with 2-deoxyribosyl as the saccharide radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
- C07H19/167—Purine radicals with ribosyl as the saccharide radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Gastroenterology & Hepatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US42744702P | 2002-11-19 | 2002-11-19 | |
| US48397003P | 2003-07-01 | 2003-07-01 | |
| PCT/EP2003/012733 WO2004046159A1 (en) | 2002-11-19 | 2003-11-14 | Antiviral nucleoside derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20052304L NO20052304L (no) | 2005-06-23 |
| NO330424B1 true NO330424B1 (no) | 2011-04-11 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| NO20052304A NO330424B1 (no) | 2002-11-19 | 2005-05-11 | Nukleosidderivater, fremstilling av slike, farmasoytiske preparater omfattende slike, slike forbindelser for behandling av sykdommer samt anvendelse av slike for fremstilling av preparater for behandling av sykdom |
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| US (1) | US6846810B2 (de) |
| EP (1) | EP1565481B1 (de) |
| JP (1) | JP4362450B2 (de) |
| KR (1) | KR100676662B1 (de) |
| AR (1) | AR042192A1 (de) |
| AT (1) | ATE335755T1 (de) |
| AU (1) | AU2003288064B2 (de) |
| BR (1) | BR0316407A (de) |
| CA (1) | CA2504846C (de) |
| CO (1) | CO5550501A2 (de) |
| CY (1) | CY1106207T1 (de) |
| DE (1) | DE60307503T2 (de) |
| DK (1) | DK1565481T3 (de) |
| ES (1) | ES2270136T3 (de) |
| HR (1) | HRP20050417B1 (de) |
| IL (1) | IL168266A (de) |
| JO (1) | JO2403B1 (de) |
| MX (1) | MXPA05005282A (de) |
| MY (1) | MY136229A (de) |
| NO (1) | NO330424B1 (de) |
| NZ (1) | NZ539644A (de) |
| PA (1) | PA8588501A1 (de) |
| PE (1) | PE20040836A1 (de) |
| PL (1) | PL210967B1 (de) |
| PT (1) | PT1565481E (de) |
| RU (1) | RU2327701C2 (de) |
| TW (1) | TWI332507B (de) |
| UY (1) | UY28084A1 (de) |
| WO (1) | WO2004046159A1 (de) |
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| WO2003084518A2 (fr) | 2002-04-09 | 2003-10-16 | Flamel Technologies | Suspension orale de microcapsules de principes actifs |
| CA2480824A1 (fr) * | 2002-04-09 | 2003-10-16 | Flamel Technologies | Formulation pharmaceutique orale sous forme de suspension aqueuse de microcapsules permettant la liberation modifiee d'amoxicilline |
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| EP1536804A4 (de) * | 2002-06-28 | 2007-10-31 | Idenix Cayman Ltd | 2'-c-methyl-3'-o-l-valinester-ribofuranosylcytidin zur behandlung von flaviviridae-infektionen |
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| RU2005123395A (ru) * | 2002-12-23 | 2006-01-27 | Айденикс (Кайман) Лимитед (Ky) | Способ получения 3-нуклеозидных пролекарств |
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