NO316377B1 - Kinolin- og kinoksalinforbindelser som inhiberer blodplateavledet vekstfaktor og/eller P56<O>lck</O>-tyrosinkinase, farmas degree ytisk blandinginneholdende detsamme samt anvendelse derav - Google Patents
Kinolin- og kinoksalinforbindelser som inhiberer blodplateavledet vekstfaktor og/eller P56<O>lck</O>-tyrosinkinase, farmas degree ytisk blandinginneholdende detsamme samt anvendelse derav Download PDFInfo
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- NO316377B1 NO316377B1 NO19995817A NO995817A NO316377B1 NO 316377 B1 NO316377 B1 NO 316377B1 NO 19995817 A NO19995817 A NO 19995817A NO 995817 A NO995817 A NO 995817A NO 316377 B1 NO316377 B1 NO 316377B1
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- Norway
- Prior art keywords
- ylamino
- cyclohexanol
- dimethoxyquinoxalin
- compound according
- trans
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A61P17/06—Antipsoriatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
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- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
- C07D241/40—Benzopyrazines
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- C07D241/50—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to ring nitrogen atoms
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- C07D241/50—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to ring nitrogen atoms
- C07D241/54—Nitrogen atoms
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/06—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing isoquinuclidine ring systems
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
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US86445597A | 1997-05-28 | 1997-05-28 | |
US97261497A | 1997-11-18 | 1997-11-18 | |
PCT/US1998/011000 WO1998054157A1 (en) | 1997-05-28 | 1998-05-28 | QUINOLINE AND QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR p561ck TYROSINE KINASES |
Publications (3)
Publication Number | Publication Date |
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NO995817D0 NO995817D0 (no) | 1999-11-26 |
NO995817L NO995817L (no) | 1999-11-26 |
NO316377B1 true NO316377B1 (no) | 2004-01-19 |
Family
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Application Number | Title | Priority Date | Filing Date |
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NO19995818A NO323720B1 (no) | 1997-05-28 | 1999-11-26 | Kinolin- og kinoksalinforbindelser som inhiberer blodplateavledet vekstfaktor og/eller P561ck-tyrosinkinase |
NO19995817A NO316377B1 (no) | 1997-05-28 | 1999-11-26 | Kinolin- og kinoksalinforbindelser som inhiberer blodplateavledet vekstfaktor og/eller P56<O>lck</O>-tyrosinkinase, farmas degree ytisk blandinginneholdende detsamme samt anvendelse derav |
NO19995819A NO323721B1 (no) | 1997-05-28 | 1999-11-26 | Kinolin- og kinoksalinforbindelser som inhiberer blodplateavledet vekstfaktor og/eller P56lck-tyrosinkinase og farmasoytisk formulering inneholdende det samme, samt anvendelse derav |
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NO19995818A NO323720B1 (no) | 1997-05-28 | 1999-11-26 | Kinolin- og kinoksalinforbindelser som inhiberer blodplateavledet vekstfaktor og/eller P561ck-tyrosinkinase |
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Application Number | Title | Priority Date | Filing Date |
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NO19995819A NO323721B1 (no) | 1997-05-28 | 1999-11-26 | Kinolin- og kinoksalinforbindelser som inhiberer blodplateavledet vekstfaktor og/eller P56lck-tyrosinkinase og farmasoytisk formulering inneholdende det samme, samt anvendelse derav |
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EP (3) | EP1001945B1 (de) |
JP (3) | JP2002500676A (de) |
KR (2) | KR100425638B1 (de) |
CN (3) | CN1280572A (de) |
AP (3) | AP1362A (de) |
AT (3) | ATE493389T1 (de) |
AU (3) | AU742739B2 (de) |
BG (3) | BG64419B1 (de) |
BR (3) | BR9809172A (de) |
CA (3) | CA2291728A1 (de) |
CZ (3) | CZ298521B6 (de) |
DE (3) | DE69842077D1 (de) |
DK (1) | DK0991628T3 (de) |
EA (4) | EA008136B1 (de) |
ES (1) | ES2235331T3 (de) |
HK (1) | HK1028042A1 (de) |
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SI (1) | SI0991628T1 (de) |
SK (4) | SK286084B6 (de) |
UA (1) | UA57790C2 (de) |
WO (3) | WO1998054156A1 (de) |
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AU5574798A (en) * | 1997-01-21 | 1998-08-07 | Nissan Chemical Industries Ltd. | Industrial antimicrobial/mildew-proofing agents, algicides and antifouling agents containing n-quinoxalylanilines |
EP1001945B1 (de) * | 1997-05-28 | 2011-03-02 | Aventis Pharmaceuticals Inc. | CHINOLIN UND CHINOXALINVERBINDUNGEN DIE DEN VON BLUTPLÄTTCHEN ABSTAMMENDEN FAKTOR UND/ODER p56Ick-TYROSINKINASE HEMMEN |
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1998
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- 1998-05-28 DK DK98925022T patent/DK0991628T3/da active
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1999
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2000
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