MY130622A - Naphthyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors - Google Patents

Naphthyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors

Info

Publication number
MY130622A
MY130622A MYPI20024102A MYPI20024102A MY130622A MY 130622 A MY130622 A MY 130622A MY PI20024102 A MYPI20024102 A MY PI20024102A MY PI20024102 A MYPI20024102 A MY PI20024102A MY 130622 A MY130622 A MY 130622A
Authority
MY
Malaysia
Prior art keywords
preparation
pde4
inhibitors
naphthyridine derivatives
phosphodiesterase isoenzyme
Prior art date
Application number
MYPI20024102A
Other languages
English (en)
Inventor
Denholm Alastair
Hugo Keller Thomas
Mccarthy Clive
John Press Neil
John Taylor Roger
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0126511A external-priority patent/GB0126511D0/en
Priority claimed from GB0209882A external-priority patent/GB0209882D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of MY130622A publication Critical patent/MY130622A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Endocrinology (AREA)
  • Hospice & Palliative Care (AREA)
  • Emergency Medicine (AREA)
  • Psychology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Transplantation (AREA)
  • Otolaryngology (AREA)
  • Ophthalmology & Optometry (AREA)
MYPI20024102A 2001-11-05 2002-11-01 Naphthyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors MY130622A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0126511A GB0126511D0 (en) 2001-11-05 2001-11-05 Organic compounds
GB0209882A GB0209882D0 (en) 2002-04-30 2002-04-30 Organic compounds

Publications (1)

Publication Number Publication Date
MY130622A true MY130622A (en) 2007-07-31

Family

ID=26246741

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI20024102A MY130622A (en) 2001-11-05 2002-11-01 Naphthyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors

Country Status (25)

Country Link
US (1) US7273875B2 (cg-RX-API-DMAC7.html)
EP (1) EP1443925B8 (cg-RX-API-DMAC7.html)
JP (1) JP4150672B2 (cg-RX-API-DMAC7.html)
KR (1) KR100623548B1 (cg-RX-API-DMAC7.html)
CN (1) CN1298324C (cg-RX-API-DMAC7.html)
AR (1) AR037517A1 (cg-RX-API-DMAC7.html)
AT (1) ATE349209T1 (cg-RX-API-DMAC7.html)
BR (1) BR0213877A (cg-RX-API-DMAC7.html)
CA (1) CA2462211C (cg-RX-API-DMAC7.html)
CY (1) CY1107532T1 (cg-RX-API-DMAC7.html)
DE (1) DE60217160T2 (cg-RX-API-DMAC7.html)
DK (1) DK1443925T3 (cg-RX-API-DMAC7.html)
ES (1) ES2275935T3 (cg-RX-API-DMAC7.html)
HU (1) HUP0402311A3 (cg-RX-API-DMAC7.html)
IL (2) IL161257A0 (cg-RX-API-DMAC7.html)
MX (1) MXPA04004264A (cg-RX-API-DMAC7.html)
MY (1) MY130622A (cg-RX-API-DMAC7.html)
NO (1) NO329093B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ532586A (cg-RX-API-DMAC7.html)
PE (1) PE20030535A1 (cg-RX-API-DMAC7.html)
PL (1) PL368286A1 (cg-RX-API-DMAC7.html)
PT (1) PT1443925E (cg-RX-API-DMAC7.html)
RU (1) RU2296764C2 (cg-RX-API-DMAC7.html)
TW (1) TWI320784B (cg-RX-API-DMAC7.html)
WO (1) WO2003039544A1 (cg-RX-API-DMAC7.html)

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US8247436B2 (en) 2010-03-19 2012-08-21 Novartis Ag Pyridine and pyrazine derivative for the treatment of CF
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