DE60217160D1 - Naphthyridine derivate, ihre herstellung und ihre anwendung als phosphodiesterase isoenzyme 4 (pde4) inhibitoren - Google Patents

Naphthyridine derivate, ihre herstellung und ihre anwendung als phosphodiesterase isoenzyme 4 (pde4) inhibitoren

Info

Publication number
DE60217160D1
DE60217160D1 DE60217160T DE60217160T DE60217160D1 DE 60217160 D1 DE60217160 D1 DE 60217160D1 DE 60217160 T DE60217160 T DE 60217160T DE 60217160 T DE60217160 T DE 60217160T DE 60217160 D1 DE60217160 D1 DE 60217160D1
Authority
DE
Germany
Prior art keywords
pde4
inhibitors
preparation
naphthyridine derivatives
phosphodiesterase isoenzyme
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60217160T
Other languages
English (en)
Other versions
DE60217160T2 (de
Inventor
Alastair Denholm
Thomas H Keller
Clive Mccarthy
Neil J Press
Roger J Taylor
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Novartis AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0126511A external-priority patent/GB0126511D0/en
Priority claimed from GB0209882A external-priority patent/GB0209882D0/en
Application filed by Novartis AG filed Critical Novartis AG
Publication of DE60217160D1 publication Critical patent/DE60217160D1/de
Application granted granted Critical
Publication of DE60217160T2 publication Critical patent/DE60217160T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
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DE60217160T 2001-11-05 2002-11-04 Naphthyridine derivate, ihre herstellung und ihre anwendung als phosphodiesterase isoenzyme 4 (pde4) inhibitoren Expired - Lifetime DE60217160T2 (de)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0126511 2001-11-05
GB0126511A GB0126511D0 (en) 2001-11-05 2001-11-05 Organic compounds
GB0209882A GB0209882D0 (en) 2002-04-30 2002-04-30 Organic compounds
GB0209882 2002-04-30
PCT/EP2002/012300 WO2003039544A1 (en) 2001-11-05 2002-11-04 Naphtyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors

Publications (2)

Publication Number Publication Date
DE60217160D1 true DE60217160D1 (de) 2007-02-08
DE60217160T2 DE60217160T2 (de) 2007-10-04

Family

ID=26246741

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60217160T Expired - Lifetime DE60217160T2 (de) 2001-11-05 2002-11-04 Naphthyridine derivate, ihre herstellung und ihre anwendung als phosphodiesterase isoenzyme 4 (pde4) inhibitoren

Country Status (26)

Country Link
US (1) US7273875B2 (de)
EP (1) EP1443925B8 (de)
JP (1) JP4150672B2 (de)
KR (1) KR100623548B1 (de)
CN (1) CN1298324C (de)
AR (1) AR037517A1 (de)
AT (1) ATE349209T1 (de)
BR (1) BR0213877A (de)
CA (1) CA2462211C (de)
CY (1) CY1107532T1 (de)
DE (1) DE60217160T2 (de)
DK (1) DK1443925T3 (de)
ES (1) ES2275935T3 (de)
HK (1) HK1069970A1 (de)
HU (1) HUP0402311A3 (de)
IL (2) IL161257A0 (de)
MX (1) MXPA04004264A (de)
MY (1) MY130622A (de)
NO (1) NO329093B1 (de)
NZ (1) NZ532586A (de)
PE (1) PE20030535A1 (de)
PL (1) PL368286A1 (de)
PT (1) PT1443925E (de)
RU (1) RU2296764C2 (de)
TW (1) TWI320784B (de)
WO (1) WO2003039544A1 (de)

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