MX370904B - Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il)ciclopropanocarboxamida. - Google Patents

Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il)ciclopropanocarboxamida.

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Publication number
MX370904B
MX370904B MX2017001548A MX2017001548A MX370904B MX 370904 B MX370904 B MX 370904B MX 2017001548 A MX2017001548 A MX 2017001548A MX 2017001548 A MX2017001548 A MX 2017001548A MX 370904 B MX370904 B MX 370904B
Authority
MX
Mexico
Prior art keywords
difluorobenzo
methylpropan
dioxol
indol
fluoro
Prior art date
Application number
MX2017001548A
Other languages
English (en)
Spanish (es)
Inventor
A Nugent William
Zhang Beili
Krawiec Mariusz
Chungmin Lee Elaine
Edward Alcacio Tim
Zhang Yuegang
Keshavarz-Shokri Ali
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43903962&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX370904(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of MX370904B publication Critical patent/MX370904B/es

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    • C—CHEMISTRY; METALLURGY
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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
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MX2017001548A 2010-03-25 2011-03-25 Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il)ciclopropanocarboxamida. MX370904B (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US31737610P 2010-03-25 2010-03-25
US31995310P 2010-04-01 2010-04-01
US32163610P 2010-04-07 2010-04-07
US32156110P 2010-04-07 2010-04-07
PCT/US2011/030032 WO2011119984A1 (en) 2010-03-25 2011-03-25 Solid forms of (r)-1(2,2-difluorobenzo[d][1,3]dioxol-5-yl)-n-(1-(2,3-dihyderoxypropyl)-6-fluoro-2-(1-hydroxy-2-methylpropan-2-yl)-1h-indol-5-yl) cyclopropanecarboxamide

Publications (1)

Publication Number Publication Date
MX370904B true MX370904B (es) 2020-01-09

Family

ID=43903962

Family Applications (3)

Application Number Title Priority Date Filing Date
MX2017001548A MX370904B (es) 2010-03-25 2011-03-25 Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il)ciclopropanocarboxamida.
MX2016001939A MX345541B (es) 2010-03-25 2011-03-25 Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il) ciclopropanocarboxamida.
MX2012011062A MX347804B (es) 2010-03-25 2011-03-25 Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il) ciclopropanocarboxamida.

Family Applications After (2)

Application Number Title Priority Date Filing Date
MX2016001939A MX345541B (es) 2010-03-25 2011-03-25 Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il) ciclopropanocarboxamida.
MX2012011062A MX347804B (es) 2010-03-25 2011-03-25 Formas solidas de (r)-1(2,2-difluorobenzo[d] [1,3]dioxol-5-il)-n-( 1-(2,3-dihidroxipropil)-6-fluoro-2-(1-hidroxi-2-metilpropan-2-il) -1h-indol-5-il) ciclopropanocarboxamida.

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US (1) US20110251253A1 (enExample)
EP (5) EP3181561B1 (enExample)
JP (5) JP5734410B2 (enExample)
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