LU90736I2 - Agenerase-amprenavir et ses d-riv-s pharmaceutiquement acceptables - Google Patents

Agenerase-amprenavir et ses d-riv-s pharmaceutiquement acceptables

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Publication number
LU90736I2
LU90736I2 LU90736C LU90736C LU90736I2 LU 90736 I2 LU90736 I2 LU 90736I2 LU 90736 C LU90736 C LU 90736C LU 90736 C LU90736 C LU 90736C LU 90736 I2 LU90736 I2 LU 90736I2
Authority
LU
Luxembourg
Prior art keywords
agenerase
amprenavir
pharmaceutically acceptable
acceptable derivatives
derivatives
Prior art date
Application number
LU90736C
Other languages
English (en)
French (fr)
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of LU90736I2 publication Critical patent/LU90736I2/fr

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    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
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    • C07C311/12—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing rings
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    • C07C311/18—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to hydrogen atoms or to an acyclic carbon atom to an acyclic carbon atom of a hydrocarbon radical substituted by nitrogen atoms, not being part of nitro or nitroso groups
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EP0659181B1 (en) 1999-04-07
EP0885887A2 (en) 1998-12-23
HK1012631A1 (en) 1999-08-06
NO303444B1 (no) 1998-07-13
CA2143208A1 (en) 1994-03-17
NO950876L (no) 1995-05-08
NZ256238A (en) 1997-04-24
AU4852093A (en) 1994-03-29
SG43862A1 (en) 1997-11-14
IL106927A (en) 2001-01-11
US20080293727A1 (en) 2008-11-27
US20030069222A1 (en) 2003-04-10
US20100210603A1 (en) 2010-08-19
HK1023561A1 (en) 2000-09-15
SK281360B6 (sk) 2001-02-12
NO950876D0 (no) 1995-03-07
PT885887E (pt) 2003-10-31
MXPA03010538A (es) 2011-12-16
CY2164B1 (en) 2002-08-23
BG62488B1 (bg) 1999-12-30
EP0885887A3 (en) 1999-02-03
DE69333012T2 (de) 2004-04-01
DE69324369D1 (de) 1999-05-12
AU691160B2 (en) 1998-05-14
TW254927B (OSRAM) 1995-08-21
IS4068A (is) 1994-03-09
HU228198B1 (en) 2013-01-28
AP9300572A0 (en) 1993-10-31
US7608632B2 (en) 2009-10-27
ES2200243T3 (es) 2004-03-01
CA2143208C (en) 2003-01-07
DK0885887T3 (da) 2003-09-22
DE69324369T2 (de) 1999-08-26
NO2001012I1 (no) 2001-07-23
FI951059A0 (fi) 1995-03-07
US20060189810A1 (en) 2006-08-24
CZ58795A3 (en) 1995-12-13
LT3302B (en) 1995-06-26
US5856353A (en) 1999-01-05
JP3012002B2 (ja) 2000-02-21
SK29395A3 (en) 1995-09-13
FI951059L (fi) 1995-04-18
DK0659181T3 (da) 1999-10-18
HU9500685D0 (en) 1995-04-28
DE10199024I2 (de) 2006-04-06
NZ314376A (en) 1998-10-28
AP390A (en) 1995-08-02
RU95109928A (ru) 1997-03-20
JPH08501299A (ja) 1996-02-13
IS2334B (is) 2008-02-15
ATE178598T1 (de) 1999-04-15
RO118747B1 (ro) 2003-10-30
BG99540A (bg) 1995-11-30
FI120685B (fi) 2010-01-29
MY142901A (en) 2011-01-31
CZ289475B6 (cs) 2002-01-16
NL300039I2 (nl) 2001-09-03
GEP20012579B (en) 2001-11-26
US5585397A (en) 1996-12-17
WO1994005639A1 (en) 1994-03-17
BR1100824A (pt) 1999-08-31
ATE241602T1 (de) 2003-06-15
DE10199024I1 (de) 2001-07-12
DE69333012D1 (de) 2003-07-03
CO4870779A1 (es) 1999-12-27
ES2131589T3 (es) 1999-08-01
RU2135496C1 (ru) 1999-08-27
HUT71892A (en) 1996-02-28
UA44694C2 (uk) 2002-03-15
US6372778B1 (en) 2002-04-16
EP0885887B1 (en) 2003-05-28
IL106927A0 (en) 1993-12-28
CN1087347A (zh) 1994-06-01
PH31251A (en) 1998-05-05
PL185635B1 (pl) 2003-06-30
CN1061339C (zh) 2001-01-31
EP0659181A1 (en) 1995-06-28
LTIP917A (en) 1994-11-25
KR100262056B1 (ko) 2000-07-15
PL307858A1 (en) 1995-06-26
GR3030719T3 (en) 1999-11-30

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