DE69619067T2 - Verfahren zur Herstellung von 3-Amino-2-oxo-1-Halogenpropan-Derivaten - Google Patents
Verfahren zur Herstellung von 3-Amino-2-oxo-1-Halogenpropan-DerivatenInfo
- Publication number
- DE69619067T2 DE69619067T2 DE69619067T DE69619067T DE69619067T2 DE 69619067 T2 DE69619067 T2 DE 69619067T2 DE 69619067 T DE69619067 T DE 69619067T DE 69619067 T DE69619067 T DE 69619067T DE 69619067 T2 DE69619067 T2 DE 69619067T2
- Authority
- DE
- Germany
- Prior art keywords
- halopropane
- oxo
- derivatives
- amino
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C221/00—Preparation of compounds containing amino groups and doubly-bound oxygen atoms bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
- C07C227/16—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions not involving the amino or carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/30—Preparation of optical isomers
- C07C227/32—Preparation of optical isomers by stereospecific synthesis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/22—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated the carbon skeleton being further substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
- C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
- C07C319/20—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by reactions not involving the formation of sulfide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
- C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
- C07C323/39—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton at least one of the nitrogen atoms being part of any of the groups, X being a hetero atom, Y being any atom
- C07C323/43—Y being a hetero atom
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP29982795 | 1995-11-17 |
Publications (2)
Publication Number | Publication Date |
---|---|
DE69619067D1 DE69619067D1 (de) | 2002-03-21 |
DE69619067T2 true DE69619067T2 (de) | 2002-10-02 |
Family
ID=17877407
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE69619067T Expired - Fee Related DE69619067T2 (de) | 1995-11-17 | 1996-11-18 | Verfahren zur Herstellung von 3-Amino-2-oxo-1-Halogenpropan-Derivaten |
Country Status (4)
Country | Link |
---|---|
US (3) | US5767316A (de) |
EP (2) | EP0774453B1 (de) |
CA (1) | CA2190570C (de) |
DE (1) | DE69619067T2 (de) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0774453B1 (de) * | 1995-11-17 | 2002-02-06 | Ajinomoto Co., Inc. | Verfahren zur Herstellung von 3-Amino-2-oxo-1-Halogenpropan-Derivaten |
JPH11100363A (ja) * | 1997-07-29 | 1999-04-13 | Kanegafuchi Chem Ind Co Ltd | アミノ基が保護された(2s,3r)−1−ハロ−2−ヒドロキシ−3−アミノ−4−フェニルチオブタン又はその光学対掌体の精製、単離方法 |
EP1661893A3 (de) * | 1999-01-29 | 2006-06-07 | Kaneka Corporation | Verfahren zur Herstellung von threo-1,2-epoxy-3-amino-4-phenylbutan-Derivaten |
KR100708221B1 (ko) * | 1999-08-31 | 2007-04-17 | 아지노모토 가부시키가이샤 | 에폭사이드 결정의 제조방법 |
EP2319824A3 (de) * | 1999-12-23 | 2012-04-11 | Ampac Fine Chemicals LLC | Verbesserte Herstellung von 2S,3S-N-isobutyl-N-(2-hydroxy-3-amino-4-phenylbutyl)amin |
US6399793B1 (en) * | 2000-08-16 | 2002-06-04 | Bristol-Myers Squibb Company | Process for the preparation of α' chloroketones |
EP1346979A4 (de) * | 2000-11-30 | 2005-11-09 | Ajinomoto Kk | Verfahren zur herstellung von n-geschützten aminoalkoholen und n-geschützten aminoepoxiden |
DE10143742A1 (de) * | 2001-09-06 | 2003-03-27 | Consortium Elektrochem Ind | Verfahren zur Herstellung von alpha-Halogenketonen |
CN1329373C (zh) * | 2003-12-11 | 2007-08-01 | 上海安基生物科技股份有限公司 | (2s.3r)-n-苄氧羰基-3-氨基-1-氯-4-苯硫基-2-丁醇的生产方法 |
EP1700122A4 (de) * | 2003-12-19 | 2008-05-21 | Ark Diagnostics Inc | Immunoassays, haptene, immunogene und antikörper für anti-hiv-therapeutika |
ME01059B (me) | 2003-12-23 | 2012-10-20 | Janssen Sciences Ireland Uc | Proces za pripremanje (3r,3as,6ar)-heksahidrofuro [2,3-b] furan-3-il (1s,2r)-3-[[(4-aminofenil) sulfonil] (izobutil) amino]-1-benzil-2- hidroksipropilkarbamata |
US20100183716A1 (en) * | 2007-06-22 | 2010-07-22 | Bristo-Meyers Squibb Company | Tableted compositions containing atazanavir |
WO2009002823A2 (en) * | 2007-06-22 | 2008-12-31 | Bristol-Myers Squibb Company | Tableted compositions containing atazanavir |
DK2170292T3 (da) * | 2007-06-22 | 2014-04-07 | Bristol Myers Squibb Holdings Ireland | Atazanavirholdige sammensætninger i tabletform |
DE602008005462D1 (de) * | 2007-06-22 | 2011-04-21 | Bristol Myers Squibb Co | Tablettierte atazanavirhaltige zusammensetzungen |
CN101508664B (zh) * | 2009-02-25 | 2012-08-22 | 江阴希迪医药科技有限公司 | N-苄氧羰基-3-氨基-1-氯-4-苯硫基-2-丁醇合成方法 |
DK2380871T3 (da) * | 2010-04-15 | 2013-04-08 | Indena Spa | Fremgangsmåde til fremstilling af isoserin-derivater |
CN106380412A (zh) * | 2016-08-31 | 2017-02-08 | 中国科学院新疆生态与地理研究所 | 一种合成利托那韦中间体的方法 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1529913A (en) | 1976-02-04 | 1978-10-25 | Beecham Group Ltd | Beta-lactam compounds |
CA1340588C (en) | 1988-06-13 | 1999-06-08 | Balraj Krishan Handa | Amino acid derivatives |
DE3820492A1 (de) | 1988-06-16 | 1989-12-28 | Diehl Gmbh & Co | Rohrwaffe mit chemisch-elektrischem hybridantrieb mittels regenerativer treibmitteleinspritzung |
US5021454A (en) * | 1989-10-06 | 1991-06-04 | Rohm And Haas Company | Benzoylaminoalkanoic acids and esters |
US5101068A (en) | 1990-02-16 | 1992-03-31 | Prototek Inc. | Magnesium fluoromalonates |
US5648511A (en) * | 1990-11-19 | 1997-07-15 | G.D. Searle & Co. | Method for making intermediates useful in the synthesis of retroviral protease inhibitors |
EP0641333B1 (de) | 1992-05-20 | 1996-08-14 | G.D. Searle & Co. | Verfahren zur herstellung von intermediaten in der synthese von retroviralen protease inhibitoren |
IS2334B (is) | 1992-09-08 | 2008-02-15 | Vertex Pharmaceuticals Inc., (A Massachusetts Corporation) | Aspartyl próteasi hemjari af nýjum flokki súlfonamíða |
US5461154A (en) | 1994-02-02 | 1995-10-24 | Eli Lilly And Company | Intermediate and process for making |
JP3665343B2 (ja) | 1995-02-03 | 2005-06-29 | 株式会社カネカ | α−ハロケトン、α−ハロヒドリン及びエポキシドの製造法 |
EP0774453B1 (de) * | 1995-11-17 | 2002-02-06 | Ajinomoto Co., Inc. | Verfahren zur Herstellung von 3-Amino-2-oxo-1-Halogenpropan-Derivaten |
-
1996
- 1996-11-18 EP EP96308319A patent/EP0774453B1/de not_active Expired - Lifetime
- 1996-11-18 DE DE69619067T patent/DE69619067T2/de not_active Expired - Fee Related
- 1996-11-18 CA CA002190570A patent/CA2190570C/en not_active Expired - Fee Related
- 1996-11-18 EP EP01100821A patent/EP1097919A3/de not_active Withdrawn
- 1996-11-18 US US08/752,169 patent/US5767316A/en not_active Ceased
-
1998
- 1998-04-14 US US09/059,370 patent/US5902887A/en not_active Expired - Fee Related
-
2000
- 2000-06-16 US US09/595,173 patent/USRE38796E1/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US5902887A (en) | 1999-05-11 |
EP0774453B1 (de) | 2002-02-06 |
CA2190570A1 (en) | 1997-05-18 |
EP1097919A3 (de) | 2003-08-06 |
US5767316A (en) | 1998-06-16 |
EP1097919A2 (de) | 2001-05-09 |
EP0774453A1 (de) | 1997-05-21 |
CA2190570C (en) | 2005-05-03 |
USRE38796E1 (en) | 2005-09-13 |
DE69619067D1 (de) | 2002-03-21 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |