KR20220064369A - Cdk2 저해제로서의 이미다졸릴 피리디미딘일아민 화합물 - Google Patents

Cdk2 저해제로서의 이미다졸릴 피리디미딘일아민 화합물 Download PDF

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KR20220064369A
KR20220064369A KR1020227008392A KR20227008392A KR20220064369A KR 20220064369 A KR20220064369 A KR 20220064369A KR 1020227008392 A KR1020227008392 A KR 1020227008392A KR 20227008392 A KR20227008392 A KR 20227008392A KR 20220064369 A KR20220064369 A KR 20220064369A
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alkyl
trifluoromethyl
imidazol
methylsulfonyl
pyrimidin
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민 예
잉난 천
마가렛 파바타
이본 로
친다 예
징웨이 리
켄 무카이
브랜든 스미스
량싱 우
웬칭 야오
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인사이트 코포레이션
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KR1020227008392A 2019-08-14 2020-08-13 Cdk2 저해제로서의 이미다졸릴 피리디미딘일아민 화합물 Pending KR20220064369A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962886735P 2019-08-14 2019-08-14
US62/886,735 2019-08-14
PCT/US2020/046078 WO2021030537A1 (en) 2019-08-14 2020-08-13 Imidazolyl pyrimidinylamine compounds as cdk2 inhibitors

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KR20220064369A true KR20220064369A (ko) 2022-05-18

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US (3) US11427567B2 (https=)
EP (1) EP4013750A1 (https=)
JP (2) JP7660556B2 (https=)
KR (1) KR20220064369A (https=)
CN (1) CN116348458A (https=)
AR (1) AR119765A1 (https=)
AU (1) AU2020328025A1 (https=)
BR (1) BR112022002698A2 (https=)
CA (1) CA3150681A1 (https=)
CL (1) CL2022000339A1 (https=)
CO (1) CO2022001453A2 (https=)
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IL (1) IL290527B1 (https=)
MX (2) MX2022001940A (https=)
PE (1) PE20221010A1 (https=)
PH (1) PH12022550361A1 (https=)
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CA3150681A1 (en) 2019-08-14 2021-02-18 Incyte Corporation Imidazolyl pyrimidinylamine compounds as cdk2 inhibitors
TWI841768B (zh) 2019-08-14 2024-05-11 美商克林提克斯醫藥股份有限公司 非肽生長抑制素(somatostatin)5型受體激動劑及其用途
US11851426B2 (en) 2019-10-11 2023-12-26 Incyte Corporation Bicyclic amines as CDK2 inhibitors
WO2022113003A1 (en) 2020-11-27 2022-06-02 Rhizen Pharmaceuticals Ag Cdk inhibitors
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WO2022149057A1 (en) 2021-01-05 2022-07-14 Rhizen Pharmaceuticals Ag Cdk inhibitors
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KR20240020735A (ko) 2021-05-07 2024-02-15 카이메라 쎄라퓨틱스 인코포레이티드 Cdk2 분해제 및 그 용도
US11981671B2 (en) 2021-06-21 2024-05-14 Incyte Corporation Bicyclic pyrazolyl amines as CDK2 inhibitors
US11976073B2 (en) 2021-12-10 2024-05-07 Incyte Corporation Bicyclic amines as CDK2 inhibitors
US20240018136A1 (en) * 2022-03-09 2024-01-18 Prelude Therapeutics, Incorporated CDK Inhibitors And Their Use As Pharmaceuticals
US20260034123A1 (en) * 2022-07-28 2026-02-05 Cedilla Therapeutics, Inc. Cdk2 inhibitors and methods of using the same
WO2024027825A1 (zh) * 2022-08-05 2024-02-08 齐鲁制药有限公司 一种cdk抑制剂及其磷酸盐的多晶型
CN119790049A (zh) * 2022-09-30 2025-04-08 楚浦创制（武汉）医药科技有限公司 2-氨基嘧啶类化合物及其应用、药用组合物
US20240247001A1 (en) 2022-12-16 2024-07-25 Astrazeneca Ab 2,6,9-trisubstituted purines
WO2025237337A1 (zh) * 2024-05-14 2025-11-20 浙江扬厉医药技术有限公司 噻唑取代嘧啶胺类化合物、其药物组合物及应用
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