KR100596989B1 - 탁세인의 선택적 유도체화 방법 - Google Patents

탁세인의 선택적 유도체화 방법 Download PDF

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Publication number
KR100596989B1
KR100596989B1 KR1019997003388A KR19997003388A KR100596989B1 KR 100596989 B1 KR100596989 B1 KR 100596989B1 KR 1019997003388 A KR1019997003388 A KR 1019997003388A KR 19997003388 A KR19997003388 A KR 19997003388A KR 100596989 B1 KR100596989 B1 KR 100596989B1
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KR
South Korea
Prior art keywords
hydrocarbyl
hydroxy
hydrogen
heteroaryl
taxane
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Expired - Fee Related
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KR1019997003388A
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English (en)
Korean (ko)
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KR20000068782A (ko
Inventor
홀튼로버트에이.
쟝주밍
클락폴에이.
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플로리다 스테이트 유니버시티
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Publication of KR20000068782A publication Critical patent/KR20000068782A/ko
Application granted granted Critical
Publication of KR100596989B1 publication Critical patent/KR100596989B1/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • C07F7/1872—Preparation; Treatments not provided for in C07F7/20
    • C07F7/1892—Preparation; Treatments not provided for in C07F7/20 by reactions not provided for in C07F7/1876 - C07F7/1888

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epoxy Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Soil Working Implements (AREA)
  • Fats And Perfumes (AREA)
  • Percussion Or Vibration Massage (AREA)
KR1019997003388A 1997-08-18 1998-08-17 탁세인의 선택적 유도체화 방법 Expired - Fee Related KR100596989B1 (ko)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US5600097P 1997-08-18 1997-08-18
US60/056,000 1997-08-18
US8126598P 1998-04-09 1998-04-09
US60/081,265 1998-04-09
US09/063,477 US7288665B1 (en) 1997-08-18 1998-04-20 Process for selective derivatization of taxanes
US9/063,477 1998-04-20
US09/063,477 1998-04-20
PCT/US1998/017016 WO1999009021A1 (en) 1997-08-18 1998-08-17 Process for selective derivatization of taxanes

Publications (2)

Publication Number Publication Date
KR20000068782A KR20000068782A (ko) 2000-11-25
KR100596989B1 true KR100596989B1 (ko) 2006-07-07

Family

ID=27368950

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019997003388A Expired - Fee Related KR100596989B1 (ko) 1997-08-18 1998-08-17 탁세인의 선택적 유도체화 방법

Country Status (25)

Country Link
US (5) US7288665B1 (enExample)
EP (6) EP1671960A2 (enExample)
JP (1) JP2001504864A (enExample)
KR (1) KR100596989B1 (enExample)
CN (3) CN100351246C (enExample)
AT (3) ATE326455T1 (enExample)
AU (1) AU744987B2 (enExample)
BR (1) BR9806145A (enExample)
CA (2) CA2268662A1 (enExample)
CY (1) CY1105399T1 (enExample)
CZ (1) CZ296580B6 (enExample)
DE (3) DE69836072T2 (enExample)
DK (3) DK0956284T3 (enExample)
ES (3) ES2274579T3 (enExample)
HU (1) HUP0300425A3 (enExample)
ID (1) ID21654A (enExample)
IL (3) IL129386A0 (enExample)
NO (4) NO325139B1 (enExample)
NZ (1) NZ335156A (enExample)
PL (3) PL332723A1 (enExample)
PT (3) PT1170293E (enExample)
RU (1) RU2225402C2 (enExample)
SG (1) SG97986A1 (enExample)
WO (1) WO1999009021A1 (enExample)
ZA (1) ZA987394B (enExample)

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