KR100223720B1 - 항종양화합물 및 그 제조방법 - Google Patents

항종양화합물 및 그 제조방법 Download PDF

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Publication number
KR100223720B1
KR100223720B1 KR1019950704147A KR19950704147A KR100223720B1 KR 100223720 B1 KR100223720 B1 KR 100223720B1 KR 1019950704147 A KR1019950704147 A KR 1019950704147A KR 19950704147 A KR19950704147 A KR 19950704147A KR 100223720 B1 KR100223720 B1 KR 100223720B1
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KR
South Korea
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group
radical
hydrogen
substituted
tert
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Expired - Fee Related
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KR1019950704147A
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English (en)
Korean (ko)
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KR960701045A (ko
Inventor
오지마 이와오
봄바델리 에지오
Original Assignee
제임스 알. 데니히
더 리서치 파운데이션 오브 스테이트 유니버시티 오브 뉴욕
팔리안티 쥬세뻬
인데나 에스.피.아
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Application filed by 제임스 알. 데니히, 더 리서치 파운데이션 오브 스테이트 유니버시티 오브 뉴욕, 팔리안티 쥬세뻬, 인데나 에스.피.아 filed Critical 제임스 알. 데니히
Priority to KR1019980709593A priority Critical patent/KR100223114B1/ko
Publication of KR960701045A publication Critical patent/KR960701045A/ko
Application granted granted Critical
Publication of KR100223720B1 publication Critical patent/KR100223720B1/ko
Anticipated expiration legal-status Critical
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
    • C07F7/1804—Compounds having Si-O-C linkages
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
KR1019950704147A 1993-03-26 1994-03-24 항종양화합물 및 그 제조방법 Expired - Fee Related KR100223720B1 (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1019980709593A KR100223114B1 (ko) 1993-03-26 1994-03-24 항종양화합물,그제조방법및용도

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US8/040189 1993-03-26
US08/040,189 US5475011A (en) 1993-03-26 1993-03-26 Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment
PCT/US1994/003215 WO1994022856A1 (en) 1993-03-26 1994-03-24 Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1019980709593A Division KR100223114B1 (ko) 1993-03-26 1994-03-24 항종양화합물,그제조방법및용도

Publications (2)

Publication Number Publication Date
KR960701045A KR960701045A (ko) 1996-02-24
KR100223720B1 true KR100223720B1 (ko) 1999-10-15

Family

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Family Applications (1)

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KR1019950704147A Expired - Fee Related KR100223720B1 (ko) 1993-03-26 1994-03-24 항종양화합물 및 그 제조방법

Country Status (19)

Country Link
US (3) US5475011A (enExample)
EP (1) EP0690856B1 (enExample)
JP (2) JP3157165B2 (enExample)
KR (1) KR100223720B1 (enExample)
CN (1) CN1067682C (enExample)
AT (1) ATE229018T1 (enExample)
AU (1) AU676041B2 (enExample)
CA (1) CA2158147C (enExample)
CZ (1) CZ288924B6 (enExample)
DE (1) DE69431833T2 (enExample)
DK (1) DK0690856T3 (enExample)
ES (1) ES2190440T3 (enExample)
HU (1) HUT73848A (enExample)
NO (1) NO311722B1 (enExample)
PL (2) PL179587B1 (enExample)
PT (1) PT690856E (enExample)
RU (1) RU2137764C1 (enExample)
SK (1) SK282317B6 (enExample)
WO (1) WO1994022856A1 (enExample)

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CN101838281B (zh) * 2010-05-20 2015-02-18 上海博速医药科技有限公司 一种多西他赛手性侧链中间体的制备方法
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Also Published As

Publication number Publication date
JPH08508497A (ja) 1996-09-10
DE69431833T2 (de) 2003-11-06
DE69431833D1 (de) 2003-01-16
CZ248095A3 (en) 1996-03-13
KR960701045A (ko) 1996-02-24
CN1067682C (zh) 2001-06-27
NO953796D0 (no) 1995-09-25
ES2190440T3 (es) 2003-08-01
US5705508A (en) 1998-01-06
CA2158147A1 (en) 1994-10-13
NO953796L (no) 1995-11-15
NO311722B1 (no) 2002-01-14
CZ288924B6 (cs) 2001-09-12
US5599820A (en) 1997-02-04
PL310827A1 (en) 1996-01-08
JP3145993B2 (ja) 2001-03-12
EP0690856B1 (en) 2002-12-04
HU9502642D0 (en) 1995-11-28
PL180708B1 (pl) 2001-03-30
EP0690856A4 (enExample) 1996-02-07
CA2158147C (en) 1999-10-05
JPH11322737A (ja) 1999-11-24
PL179587B1 (pl) 2000-09-29
RU2137764C1 (ru) 1999-09-20
ATE229018T1 (de) 2002-12-15
AU676041B2 (en) 1997-02-27
SK118395A3 (en) 1996-06-05
AU6491694A (en) 1994-10-24
CN1123547A (zh) 1996-05-29
SK282317B6 (sk) 2002-01-07
DK0690856T3 (da) 2003-03-31
HUT73848A (en) 1996-09-30
PT690856E (pt) 2003-04-30
US5475011A (en) 1995-12-12
WO1994022856A1 (en) 1994-10-13
EP0690856A1 (en) 1996-01-10
JP3157165B2 (ja) 2001-04-16

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