JPWO2020068729A5 - - Google Patents

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JPWO2020068729A5
JPWO2020068729A5 JP2021540378A JP2021540378A JPWO2020068729A5 JP WO2020068729 A5 JPWO2020068729 A5 JP WO2020068729A5 JP 2021540378 A JP2021540378 A JP 2021540378A JP 2021540378 A JP2021540378 A JP 2021540378A JP WO2020068729 A5 JPWO2020068729 A5 JP WO2020068729A5
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alkyl
alkylene
membered heterocycloalkyl
cycloalkyl
membered
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JP2021540378A
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JP2022502490A (ja
JP7399968B2 (ja
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Priority claimed from PCT/US2019/052567 external-priority patent/WO2020068729A1/en
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JP2021540378A 2018-09-25 2019-09-24 Ａｌｋ２及び／またはｆｇｆｒ調節剤としてのピラゾロ［４，３－ｄ］ピリミジン化合物 Active JP7399968B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862736121P 2018-09-25 2018-09-25
US62/736,121 2018-09-25
PCT/US2019/052567 WO2020068729A1 (en) 2018-09-25 2019-09-24 Pyrazolo[4,3-d]pyrimidine compounds as alk2 abd/or fgfr modulators

Publications (3)

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JP2022502490A JP2022502490A (ja) 2022-01-11
JPWO2020068729A5 true JPWO2020068729A5 (ru) 2022-06-06
JP7399968B2 JP7399968B2 (ja) 2023-12-18

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JP2021540378A Active JP7399968B2 (ja) 2018-09-25 2019-09-24 Ａｌｋ２及び／またはｆｇｆｒ調節剤としてのピラゾロ［４，３－ｄ］ピリミジン化合物

Country Status (8)

Country Link
US (2) US11111247B2 (ru)
EP (1) EP3856348B1 (ru)
JP (1) JP7399968B2 (ru)
AR (1) AR116507A1 (ru)
ES (1) ES2973117T3 (ru)
MA (1) MA53726A (ru)
TW (1) TW202028207A (ru)
WO (1) WO2020068729A1 (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7504880B2 (ja) 2018-10-26 2024-06-24 ケロス セラピューティクス インコーポレイテッド Ａｌｋ２阻害剤の結晶形
US20230018728A1 (en) * 2019-11-21 2023-01-19 Jiangsu Hengrui Medicine Co., Ltd. Pyrazolo-heteroaryl derivative, preparation method therefor, and medical use thereof
CN112941036B (zh) * 2021-02-08 2023-06-09 吉林惠康生物药业有限公司 一种提高狂犬病毒在人二倍体细胞中复制水平的方法
WO2022199652A1 (en) * 2021-03-24 2022-09-29 Impact Therapeutics (Shanghai) , Inc Five-membered heteroaryl-pyrimidine compounds as usp1 inhibitors and the use thereof
WO2024022519A1 (zh) * 2022-07-28 2024-02-01 先声再明医药有限公司 杂环并嘧啶类化合物及其应用

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