JP4155926B2 - ５ｈｔ２ｃレセプター修飾因子 - Google Patents

５ｈｔ２ｃレセプター修飾因子 Download PDF

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JP4155926B2
JP4155926B2 JP2003583332A JP2003583332A JP4155926B2 JP 4155926 B2 JP4155926 B2 JP 4155926B2 JP 2003583332 A JP2003583332 A JP 2003583332A JP 2003583332 A JP2003583332 A JP 2003583332A JP 4155926 B2 JP4155926 B2 JP 4155926B2
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tetrahydro
benzazepine
methyl
methoxy
bromo
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JP2005527579A5 (cg-RX-API-DMAC10.html
JP2005527579A (ja
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ブライアン スミス，
ジェフリー スミス，
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アリーナ ファーマシューティカルズ， インコーポレイテッド
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
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  • General Health & Medical Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Vascular Medicine (AREA)
  • Anesthesiology (AREA)
JP2003583332A 2002-04-12 2003-04-11 ５ｈｔ２ｃレセプター修飾因子 Expired - Lifetime JP4155926B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US37205802P 2002-04-12 2002-04-12
US40549502P 2002-08-23 2002-08-23
US43460702P 2002-12-18 2002-12-18
US10/410,991 US6953787B2 (en) 2002-04-12 2003-04-10 5HT2C receptor modulators
PCT/US2003/011076 WO2003086306A2 (en) 2002-04-12 2003-04-11 5ht2c receptor modulators

Related Child Applications (1)

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JP2006058747A Division JP4191741B2 (ja) 2002-04-12 2006-03-03 ５ｈｔ２ｃレセプター修飾因子

Publications (3)

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JP2005527579A JP2005527579A (ja) 2005-09-15
JP2005527579A5 JP2005527579A5 (cg-RX-API-DMAC10.html) 2007-03-29
JP4155926B2 true JP4155926B2 (ja) 2008-09-24

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JP2003583332A Expired - Lifetime JP4155926B2 (ja) 2002-04-12 2003-04-11 ５ｈｔ２ｃレセプター修飾因子
JP2006058747A Expired - Lifetime JP4191741B2 (ja) 2002-04-12 2006-03-03 ５ｈｔ２ｃレセプター修飾因子
JP2008202412A Expired - Lifetime JP4966929B2 (ja) 2002-04-12 2008-08-05 ５ｈｔ２ｃレセプター修飾因子
JP2011201117A Expired - Lifetime JP5602116B2 (ja) 2002-04-12 2011-09-14 ５ｈｔ２ｃレセプター修飾因子
JP2012211059A Withdrawn JP2013018780A (ja) 2002-04-12 2012-09-25 ５ｈｔ２ｃレセプター修飾因子

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JP2006058747A Expired - Lifetime JP4191741B2 (ja) 2002-04-12 2006-03-03 ５ｈｔ２ｃレセプター修飾因子
JP2008202412A Expired - Lifetime JP4966929B2 (ja) 2002-04-12 2008-08-05 ５ｈｔ２ｃレセプター修飾因子
JP2011201117A Expired - Lifetime JP5602116B2 (ja) 2002-04-12 2011-09-14 ５ｈｔ２ｃレセプター修飾因子
JP2012211059A Withdrawn JP2013018780A (ja) 2002-04-12 2012-09-25 ５ｈｔ２ｃレセプター修飾因子

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EP (4) EP1557409A1 (cg-RX-API-DMAC10.html)
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KR (3) KR100908166B1 (cg-RX-API-DMAC10.html)
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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007521269A (ja) * 2003-06-17 2007-08-02 アリーナ ファーマシューティカルズ， インコーポレイテッド ３−ベンズアゼピンを調製する方法
JP2012006970A (ja) * 2002-04-12 2012-01-12 Arena Pharmaceuticals Inc ５ｈｔ２ｃレセプター修飾因子

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* Cited by examiner, † Cited by third party
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JP2007521269A (ja) * 2003-06-17 2007-08-02 アリーナ ファーマシューティカルズ， インコーポレイテッド ３−ベンズアゼピンを調製する方法
JP2011116780A (ja) * 2003-06-17 2011-06-16 Arena Pharmaceuticals Inc ３−ベンズアゼピンを調製する方法
JP4920409B2 (ja) * 2003-06-17 2012-04-18 アリーナ ファーマシューティカルズ， インコーポレイテッド ３−ベンズアゼピンを調製する方法
JP2012107067A (ja) * 2003-06-17 2012-06-07 Arena Pharmaceuticals Inc ３−ベンズアゼピンを調製する方法

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