JP2016508136A5 - - Google Patents
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- JP2016508136A5 JP2016508136A5 JP2015549842A JP2015549842A JP2016508136A5 JP 2016508136 A5 JP2016508136 A5 JP 2016508136A5 JP 2015549842 A JP2015549842 A JP 2015549842A JP 2015549842 A JP2015549842 A JP 2015549842A JP 2016508136 A5 JP2016508136 A5 JP 2016508136A5
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- JP
- Japan
- Prior art keywords
- linker
- self
- bond
- compound
- destructing
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 CC(OC(C(N1CCN(*)CC1)=O)c(cc1)ccc1NC)=O Chemical compound CC(OC(C(N1CCN(*)CC1)=O)c(cc1)ccc1NC)=O 0.000 description 2
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261745448P | 2012-12-21 | 2012-12-21 | |
| US61/745,448 | 2012-12-21 | ||
| US201361785027P | 2013-03-14 | 2013-03-14 | |
| US61/785,027 | 2013-03-14 | ||
| PCT/US2013/077306 WO2014100762A1 (en) | 2012-12-21 | 2013-12-20 | Hydrophilic self-immolative linkers and conjugates thereof |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2016508136A JP2016508136A (ja) | 2016-03-17 |
| JP2016508136A5 true JP2016508136A5 (enExample) | 2018-06-14 |
| JP6482471B2 JP6482471B2 (ja) | 2019-03-13 |
Family
ID=50979293
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2015549842A Expired - Fee Related JP6482471B2 (ja) | 2012-12-21 | 2013-12-20 | 親水性の自壊性リンカー及びそのコンジュゲート |
Country Status (23)
| Country | Link |
|---|---|
| US (5) | US9089614B2 (enExample) |
| EP (1) | EP2935259B1 (enExample) |
| JP (1) | JP6482471B2 (enExample) |
| KR (2) | KR20150119848A (enExample) |
| CN (2) | CN108546283A (enExample) |
| AR (1) | AR094280A1 (enExample) |
| AU (1) | AU2013364065B2 (enExample) |
| BR (1) | BR112015014712A2 (enExample) |
| CA (1) | CA2896690A1 (enExample) |
| CL (1) | CL2015001735A1 (enExample) |
| DK (1) | DK2935259T3 (enExample) |
| ES (1) | ES2714951T3 (enExample) |
| IL (1) | IL239506B (enExample) |
| MX (1) | MX379355B (enExample) |
| MY (1) | MY169117A (enExample) |
| NZ (1) | NZ630601A (enExample) |
| PH (1) | PH12015501422A1 (enExample) |
| PT (1) | PT2935259T (enExample) |
| RU (2) | RU2019105549A (enExample) |
| SG (2) | SG11201504887TA (enExample) |
| TW (1) | TWI716339B (enExample) |
| WO (1) | WO2014100762A1 (enExample) |
| ZA (1) | ZA201504941B (enExample) |
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2013
- 2013-12-20 KR KR1020157019681A patent/KR20150119848A/ko not_active Abandoned
- 2013-12-20 WO PCT/US2013/077306 patent/WO2014100762A1/en not_active Ceased
- 2013-12-20 CN CN201810460861.6A patent/CN108546283A/zh active Pending
- 2013-12-20 BR BR112015014712A patent/BR112015014712A2/pt not_active Application Discontinuation
- 2013-12-20 PT PT13865282T patent/PT2935259T/pt unknown
- 2013-12-20 RU RU2019105549A patent/RU2019105549A/ru unknown
- 2013-12-20 JP JP2015549842A patent/JP6482471B2/ja not_active Expired - Fee Related
- 2013-12-20 CN CN201380073519.6A patent/CN105102455B/zh not_active Expired - Fee Related
- 2013-12-20 SG SG11201504887TA patent/SG11201504887TA/en unknown
- 2013-12-20 RU RU2015129800A patent/RU2015129800A/ru unknown
- 2013-12-20 MX MX2015007918A patent/MX379355B/es unknown
- 2013-12-20 US US14/137,799 patent/US9089614B2/en not_active Expired - Fee Related
- 2013-12-20 KR KR1020217034685A patent/KR20210132742A/ko not_active Abandoned
- 2013-12-20 US US14/654,486 patent/US9943610B2/en active Active
- 2013-12-20 MY MYPI2015001576A patent/MY169117A/en unknown
- 2013-12-20 EP EP13865282.1A patent/EP2935259B1/en active Active
- 2013-12-20 TW TW102147572A patent/TWI716339B/zh not_active IP Right Cessation
- 2013-12-20 CA CA2896690A patent/CA2896690A1/en not_active Abandoned
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- 2013-12-20 NZ NZ630601A patent/NZ630601A/en not_active IP Right Cessation
- 2013-12-20 ES ES13865282T patent/ES2714951T3/es active Active
- 2013-12-20 DK DK13865282.1T patent/DK2935259T3/en active
- 2013-12-20 AR ARP130105028A patent/AR094280A1/es unknown
- 2013-12-20 AU AU2013364065A patent/AU2013364065B2/en not_active Ceased
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2015
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- 2015-06-18 IL IL239506A patent/IL239506B/en active IP Right Grant
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- 2015-07-09 ZA ZA2015/04941A patent/ZA201504941B/en unknown
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2018
- 2018-03-13 US US15/920,229 patent/US20180264131A1/en not_active Abandoned
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2020
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