JP2009500424A5 - - Google Patents
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- JP2009500424A5 JP2009500424A5 JP2008520396A JP2008520396A JP2009500424A5 JP 2009500424 A5 JP2009500424 A5 JP 2009500424A5 JP 2008520396 A JP2008520396 A JP 2008520396A JP 2008520396 A JP2008520396 A JP 2008520396A JP 2009500424 A5 JP2009500424 A5 JP 2009500424A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- group
- aryl
- carbocycle
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Links
- 0 C*NCC(Cc1ccccc1)C(O)=O Chemical compound C*NCC(Cc1ccccc1)C(O)=O 0.000 description 3
- QXKFRGBDFPUSEZ-UHFFFAOYSA-N CC(N(C1)C(Cc2ccccc2)CCC1C(O)=O)=C Chemical compound CC(N(C1)C(Cc2ccccc2)CCC1C(O)=O)=C QXKFRGBDFPUSEZ-UHFFFAOYSA-N 0.000 description 1
- ZLIPGCUNOOFZML-UHFFFAOYSA-N CCN(CC(Cc1ccccc1)C1)CC1C(O)=O Chemical compound CCN(CC(Cc1ccccc1)C1)CC1C(O)=O ZLIPGCUNOOFZML-UHFFFAOYSA-N 0.000 description 1
- LXIANNUASSWOKI-UHFFFAOYSA-N CCN(CCC1Cc2ccccc2)CC1C(O)=O Chemical compound CCN(CCC1Cc2ccccc2)CC1C(O)=O LXIANNUASSWOKI-UHFFFAOYSA-N 0.000 description 1
- XWCSUERVLZIHKC-UHFFFAOYSA-N CCNCC(CC(O)=O)Cc1ccccc1 Chemical compound CCNCC(CC(O)=O)Cc1ccccc1 XWCSUERVLZIHKC-UHFFFAOYSA-N 0.000 description 1
- ZWURJJVCFRJQOY-UHFFFAOYSA-N CCNCCC(Cc1ccccc1)C(O)=O Chemical compound CCNCCC(Cc1ccccc1)C(O)=O ZWURJJVCFRJQOY-UHFFFAOYSA-N 0.000 description 1
- AOLLIWDGLAVYML-UHFFFAOYSA-N CN(C1)C(Cc2ccccc2)CC1C(O)=O Chemical compound CN(C1)C(Cc2ccccc2)CC1C(O)=O AOLLIWDGLAVYML-UHFFFAOYSA-N 0.000 description 1
- JEYBSDROLSIJQP-UHFFFAOYSA-N CN(CC1Cc2ccccc2)CC1C(O)=O Chemical compound CN(CC1Cc2ccccc2)CC1C(O)=O JEYBSDROLSIJQP-UHFFFAOYSA-N 0.000 description 1
- XDYCCVBZZUKWFY-UHFFFAOYSA-N CNC(CC(O)=O)Cc1ccccc1 Chemical compound CNC(CC(O)=O)Cc1ccccc1 XDYCCVBZZUKWFY-UHFFFAOYSA-N 0.000 description 1
- BJWPOHOQHOEKSU-UHFFFAOYSA-N CNC(CCC(O)=O)Cc1ccccc1 Chemical compound CNC(CCC(O)=O)Cc1ccccc1 BJWPOHOQHOEKSU-UHFFFAOYSA-N 0.000 description 1
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69776705P | 2005-07-07 | 2005-07-07 | |
| US60/697,767 | 2005-07-07 | ||
| PCT/US2006/026352 WO2007008603A1 (en) | 2005-07-07 | 2006-07-07 | Monomethylvaline compounds having phenylalanine side-chain modifications at the c-terminus |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012104711A Division JP2012144576A (ja) | 2005-07-07 | 2012-05-01 | フェニルアラニン側鎖修飾をｃ末端に有するモノメチルバリン化合物 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009500424A JP2009500424A (ja) | 2009-01-08 |
| JP2009500424A5 true JP2009500424A5 (enExample) | 2009-08-20 |
| JP5171621B2 JP5171621B2 (ja) | 2013-03-27 |
Family
ID=37637475
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2008520396A Expired - Fee Related JP5171621B2 (ja) | 2005-07-07 | 2006-07-07 | フェニルアラニン側鎖修飾をｃ末端に有するモノメチルバリン化合物 |
| JP2012104711A Withdrawn JP2012144576A (ja) | 2005-07-07 | 2012-05-01 | フェニルアラニン側鎖修飾をｃ末端に有するモノメチルバリン化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012104711A Withdrawn JP2012144576A (ja) | 2005-07-07 | 2012-05-01 | フェニルアラニン側鎖修飾をｃ末端に有するモノメチルバリン化合物 |
Country Status (7)
| Country | Link |
|---|---|
| US (3) | US8343928B2 (enExample) |
| EP (3) | EP1917020B1 (enExample) |
| JP (2) | JP5171621B2 (enExample) |
| AU (1) | AU2006269422B2 (enExample) |
| CA (1) | CA2614436C (enExample) |
| ES (2) | ES2708763T3 (enExample) |
| WO (1) | WO2007008603A1 (enExample) |
Families Citing this family (152)
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- 2006-07-07 ES ES13190752T patent/ES2708763T3/es active Active
- 2006-07-07 EP EP13190752.9A patent/EP2722051B1/en active Active
- 2006-07-07 JP JP2008520396A patent/JP5171621B2/ja not_active Expired - Fee Related
- 2006-07-07 US US11/994,809 patent/US8343928B2/en active Active
- 2006-07-07 ES ES06786489.2T patent/ES2585357T3/es active Active
- 2006-07-07 AU AU2006269422A patent/AU2006269422B2/en active Active
-
2012
- 2012-05-01 JP JP2012104711A patent/JP2012144576A/ja not_active Withdrawn
- 2012-11-01 US US13/666,766 patent/US10000555B2/en active Active
-
2018
- 2018-05-24 US US15/988,989 patent/US20180355025A1/en not_active Abandoned
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