JP2012518634A5 - - Google Patents

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Publication number
JP2012518634A5
JP2012518634A5 JP2011551039A JP2011551039A JP2012518634A5 JP 2012518634 A5 JP2012518634 A5 JP 2012518634A5 JP 2011551039 A JP2011551039 A JP 2011551039A JP 2011551039 A JP2011551039 A JP 2011551039A JP 2012518634 A5 JP2012518634 A5 JP 2012518634A5
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JP
Japan
Prior art keywords
benzamide
cyclopropyl
carbonyl
trans
cyclobutyl
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JP2011551039A
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Japanese (ja)
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JP5666480B2 (ja
JP2012518634A (ja
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Priority claimed from PCT/SE2010/050191 external-priority patent/WO2010096011A1/en
Publication of JP2012518634A publication Critical patent/JP2012518634A/ja
Publication of JP2012518634A5 publication Critical patent/JP2012518634A5/ja
Application granted granted Critical
Publication of JP5666480B2 publication Critical patent/JP5666480B2/ja
Expired - Fee Related legal-status Critical Current
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JP2011551039A 2009-02-20 2010-02-19 ヒスタミンｈ３受容体を標的とするシクロプロピルアミド誘導体 Expired - Fee Related JP5666480B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15406709P 2009-02-20 2009-02-20
US61/154,067 2009-02-20
PCT/SE2010/050191 WO2010096011A1 (en) 2009-02-20 2010-02-19 Cyclopropyl amide derivatives targeting the histamine h3 receptor

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014248499A Division JP2015071634A (ja) 2009-02-20 2014-12-09 ヒスタミンｈ３受容体を標的とするシクロプロピルアミド誘導体

Publications (3)

Publication Number Publication Date
JP2012518634A JP2012518634A (ja) 2012-08-16
JP2012518634A5 true JP2012518634A5 (enExample) 2013-04-11
JP5666480B2 JP5666480B2 (ja) 2015-02-12

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Family Applications (2)

Application Number Title Priority Date Filing Date
JP2011551039A Expired - Fee Related JP5666480B2 (ja) 2009-02-20 2010-02-19 ヒスタミンｈ３受容体を標的とするシクロプロピルアミド誘導体
JP2014248499A Pending JP2015071634A (ja) 2009-02-20 2014-12-09 ヒスタミンｈ３受容体を標的とするシクロプロピルアミド誘導体

Family Applications After (1)

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JP2014248499A Pending JP2015071634A (ja) 2009-02-20 2014-12-09 ヒスタミンｈ３受容体を標的とするシクロプロピルアミド誘導体

Country Status (39)

Country Link
US (3) US8993577B2 (enExample)
EP (1) EP2398780B1 (enExample)
JP (2) JP5666480B2 (enExample)
KR (1) KR20110126628A (enExample)
CN (2) CN104398516A (enExample)
AR (1) AR075531A1 (enExample)
AU (1) AU2010216454B2 (enExample)
BR (1) BRPI1007817A2 (enExample)
CA (1) CA2752796A1 (enExample)
CO (1) CO6400219A2 (enExample)
CR (1) CR20110447A (enExample)
CU (2) CU20110161A7 (enExample)
DK (1) DK2398780T3 (enExample)
DO (1) DOP2011000270A (enExample)
EA (2) EA020093B1 (enExample)
EC (1) ECSP11011280A (enExample)
ES (1) ES2416464T3 (enExample)
HK (1) HK1208348A1 (enExample)
HN (1) HN2011002261A (enExample)
HR (1) HRP20130579T1 (enExample)
IL (1) IL214277A (enExample)
ME (1) ME01619B (enExample)
MX (1) MX2011008280A (enExample)
NI (1) NI201100160A (enExample)
NZ (1) NZ595248A (enExample)
PE (2) PE20151281A1 (enExample)
PL (1) PL2398780T3 (enExample)
PT (1) PT2398780E (enExample)
RS (1) RS52851B (enExample)
SA (1) SA110310136B1 (enExample)
SG (1) SG173449A1 (enExample)
SI (1) SI2398780T1 (enExample)
SM (1) SMT201300077B (enExample)
SV (1) SV2011004008A (enExample)
TW (1) TW201039825A (enExample)
UA (1) UA108841C2 (enExample)
UY (1) UY32460A (enExample)
WO (1) WO2010096011A1 (enExample)
ZA (1) ZA201106821B (enExample)

Families Citing this family (11)

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WO2022059779A1 (ja) 2020-09-18 2022-03-24 大日本住友製薬株式会社 アミン誘導体
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