JP2020527175A5 - - Google Patents
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- JP2020527175A5 JP2020527175A5 JP2020524667A JP2020524667A JP2020527175A5 JP 2020527175 A5 JP2020527175 A5 JP 2020527175A5 JP 2020524667 A JP2020524667 A JP 2020524667A JP 2020524667 A JP2020524667 A JP 2020524667A JP 2020527175 A5 JP2020527175 A5 JP 2020527175A5
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- JP
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- compound according
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- Prior art date
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2017/093106 | 2017-07-17 | ||
| CNPCT/CN2017/093106 | 2017-07-17 | ||
| PCT/CN2018/095973 WO2019015583A1 (en) | 2017-07-17 | 2018-07-17 | NOVEL COMPOUNDS AND THEIR USES AS ACC INHIBITORS |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2020527175A JP2020527175A (ja) | 2020-09-03 |
| JP2020527175A5 true JP2020527175A5 (enExample) | 2021-07-26 |
| JP7067725B2 JP7067725B2 (ja) | 2022-05-16 |
Family
ID=65014996
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020524667A Expired - Fee Related JP7067725B2 (ja) | 2017-07-17 | 2018-07-17 | Ａｃｃ阻害剤としての新規な化合物およびそれらの使用 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US10995099B2 (enExample) |
| EP (1) | EP3655409B1 (enExample) |
| JP (1) | JP7067725B2 (enExample) |
| CN (1) | CN111201234A (enExample) |
| WO (2) | WO2019015583A1 (enExample) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA3070525C (en) * | 2017-07-26 | 2022-03-15 | Nanjing Sanhome Pharmaceutical Co., Ltd. | Compound as acc inhibitor and use thereof |
| JP7374233B2 (ja) | 2019-07-02 | 2023-11-06 | ▲広▼▲東▼▲東▼▲陽▼光▲薬▼▲業▼有限公司 | 立体配置を有するチエノピリミジン誘導体及び薬物におけるその応用 |
| AR119594A1 (es) * | 2019-08-09 | 2021-12-29 | Gilead Sciences Inc | Derivados de tienopirimidina como inhibidores acc y usos de los mismos |
| CN114555601B (zh) | 2019-10-15 | 2024-04-02 | 勃林格殷格翰国际有限公司 | 新颖的四唑类 |
| CN112778325A (zh) | 2019-11-07 | 2021-05-11 | 南京瑞捷医药科技有限公司 | 一种acc抑制剂及其用途 |
| CA3193607A1 (en) * | 2020-10-14 | 2022-04-21 | Boehringer Ingelheim International Gmbh | Tetrazole derivatives as trpa1 inhibitors |
| US11661427B2 (en) * | 2020-10-14 | 2023-05-30 | Boehringer Ingelheim International Gmbh | Tetrazole derivatives as TRPA1 inhibitors |
| CN116745299A (zh) * | 2021-02-07 | 2023-09-12 | 正大天晴药业集团股份有限公司 | 噻吩并嘧啶衍生物 |
| JP7565457B2 (ja) | 2021-04-14 | 2024-10-10 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ＴＲＰＡ１阻害剤としての３Ｈ，４Ｈ－チエノ－［２，３－ｄ］ピリミジン－４－オン誘導体 |
| CN114409664B (zh) * | 2021-12-24 | 2023-07-18 | 河北威远生物化工有限公司 | 一种螺杂环四氢吡喃化合物及其制备方法和应用 |
| CN114815020B (zh) * | 2022-04-21 | 2023-09-22 | 岭南师范学院 | 一种高品质因数折射率传感器的设计方法及折射率传感器 |
| CN116747321B (zh) * | 2023-06-14 | 2025-09-05 | 厦门君德医药科技有限公司 | 一种接枝改性的介孔二氧化硅及其制备方法和应用 |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3628320B1 (en) | 2011-11-11 | 2022-03-16 | Gilead Apollo, LLC | Acc inhibitors and uses thereof |
| JP6130909B2 (ja) * | 2012-05-30 | 2017-05-17 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 生物農薬および殺虫剤を含む組成物 |
| HK1221662A1 (zh) | 2013-05-10 | 2017-06-09 | Gilead Apollo, Llc | Acc抑制剂和其用途 |
| WO2015003879A1 (en) * | 2013-07-08 | 2015-01-15 | Syngenta Participations Ag | Microbiocidal heterobicylic derivatives |
| CN105949197A (zh) * | 2014-01-29 | 2016-09-21 | 苏州晶云药物科技有限公司 | 依鲁替尼的新晶型及其制备方法 |
| GB201419102D0 (en) * | 2014-10-27 | 2014-12-10 | Imp Innovations Ltd | Novel compounds |
| CA2972919A1 (en) | 2015-01-09 | 2016-07-14 | Gilead Apollo, Llc | Acc inhibitor combination therapy for the treatment of non-alcoholic fatty liver disease |
| CN205115664U (zh) * | 2015-10-15 | 2016-03-30 | 阳光能源（青海）有限公司 | 一种用于单晶炉的二次填料装置 |
| CN106137971A (zh) * | 2015-11-17 | 2016-11-23 | 南京瑞捷医药科技有限公司 | 一种他克莫司分散体及其缓释组合物及制备方法 |
| CA3005900C (en) | 2015-11-25 | 2023-10-31 | Gilead Apollo, Llc | Triazole acc inhibitors and uses thereof |
| MX2018006286A (es) | 2015-11-25 | 2018-09-07 | Gilead Apollo Llc | Inhibidores de acc pirazolicos y usos de los mismos. |
| CN108699078A (zh) | 2016-03-02 | 2018-10-23 | 吉利德阿波罗公司 | 噻吩并嘧啶二酮acc抑制剂的固体形式及其制备方法 |
| PL3589636T3 (pl) * | 2017-03-03 | 2024-02-19 | Gilead Sciences, Inc. | Sposoby wytwarzania inhibitorów acc i ich form stałych |
| WO2018228369A1 (zh) * | 2017-06-15 | 2018-12-20 | 浙江海正药业股份有限公司 | 杂芳基并嘧啶酮类衍生物、其制备方法及其在医药上用途 |
| CA3070525C (en) * | 2017-07-26 | 2022-03-15 | Nanjing Sanhome Pharmaceutical Co., Ltd. | Compound as acc inhibitor and use thereof |
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2018
- 2018-07-17 EP EP18835671.1A patent/EP3655409B1/en active Active
- 2018-07-17 US US16/631,800 patent/US10995099B2/en active Active
- 2018-07-17 CN CN201880053983.1A patent/CN111201234A/zh active Pending
- 2018-07-17 JP JP2020524667A patent/JP7067725B2/ja not_active Expired - Fee Related
- 2018-07-17 WO PCT/CN2018/095973 patent/WO2019015583A1/en not_active Ceased
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2019
- 2019-01-14 WO PCT/CN2019/071630 patent/WO2020015343A1/en not_active Ceased