IL110802A - Substituted oxazine and thiazine oxazolidinone antimicrobials and pharmaceutical compositions comprising them - Google Patents

Substituted oxazine and thiazine oxazolidinone antimicrobials and pharmaceutical compositions comprising them

Info

Publication number
IL110802A
IL110802A IL11080294A IL11080294A IL110802A IL 110802 A IL110802 A IL 110802A IL 11080294 A IL11080294 A IL 11080294A IL 11080294 A IL11080294 A IL 11080294A IL 110802 A IL110802 A IL 110802A
Authority
IL
Israel
Prior art keywords
c8alkoxy
spp
mycobacterium
hydroxy
amino
Prior art date
Application number
IL11080294A
Other languages
English (en)
Other versions
IL110802A0 (en
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26817181&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL110802(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of IL110802A0 publication Critical patent/IL110802A0/xx
Publication of IL110802A publication Critical patent/IL110802A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL11080294A 1993-09-09 1994-08-29 Substituted oxazine and thiazine oxazolidinone antimicrobials and pharmaceutical compositions comprising them IL110802A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11927993A 1993-09-09 1993-09-09
US22615894A 1994-04-11 1994-04-11

Publications (2)

Publication Number Publication Date
IL110802A0 IL110802A0 (en) 1994-11-11
IL110802A true IL110802A (en) 2000-09-28

Family

ID=26817181

Family Applications (1)

Application Number Title Priority Date Filing Date
IL11080294A IL110802A (en) 1993-09-09 1994-08-29 Substituted oxazine and thiazine oxazolidinone antimicrobials and pharmaceutical compositions comprising them

Country Status (20)

Country Link
EP (1) EP0717738B1 (es)
JP (1) JP3176630B2 (es)
KR (1) KR100301269B1 (es)
CN (1) CN1057087C (es)
AT (1) ATE185804T1 (es)
AU (1) AU687866B2 (es)
CA (1) CA2168560C (es)
DE (2) DE69421285T2 (es)
DK (1) DK0717738T3 (es)
ES (1) ES2139093T3 (es)
GR (1) GR3031809T3 (es)
IL (1) IL110802A (es)
LV (1) LV12605B (es)
MY (1) MY115155A (es)
NL (1) NL300079I1 (es)
NZ (1) NZ271805A (es)
PH (1) PH31634A (es)
SI (1) SI0717738T1 (es)
TW (1) TW293817B (es)
WO (1) WO1995007271A1 (es)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2174935A1 (en) 2004-06-29 2010-04-14 Teva Pharmaceutical Industries Ltd Linezolid Compositions

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