BR112015005743A2 - derivados tricíclicos de quinoxalina e quinolina - Google Patents

derivados tricíclicos de quinoxalina e quinolina

Info

Publication number
BR112015005743A2
BR112015005743A2 BR112015005743A BR112015005743A BR112015005743A2 BR 112015005743 A2 BR112015005743 A2 BR 112015005743A2 BR 112015005743 A BR112015005743 A BR 112015005743A BR 112015005743 A BR112015005743 A BR 112015005743A BR 112015005743 A2 BR112015005743 A2 BR 112015005743A2
Authority
BR
Brazil
Prior art keywords
tricyclic
quinoxaline
quinoline derivatives
ht2c receptor
quinoline
Prior art date
Application number
BR112015005743A
Other languages
English (en)
Inventor
Lucia Relo Ana
Haupt Andreas
Hoft Carolin
Koolman Hannes
Mack Helmut
Drescher Karla
Henrica Maria Bakker Margaretha
Xu Ruxu
Lakics Viktor
Braje Wilfried
Zhao Xiaona
Original Assignee
Abbvie Deutschland
Abbvie Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50275085&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112015005743(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from CN201310410951.1A external-priority patent/CN104418862A/zh
Application filed by Abbvie Deutschland, Abbvie Inc filed Critical Abbvie Deutschland
Publication of BR112015005743A2 publication Critical patent/BR112015005743A2/pt

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
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    • A61P25/00Drugs for disorders of the nervous system
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
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    • A61P25/08Antiepileptics; Anticonvulsants
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16Peri-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Gynecology & Obstetrics (AREA)
  • Cardiology (AREA)
  • Emergency Medicine (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

resumo “derivados tricíclicos de quinoxalina e quinolina” a presente invenção refere-se aos derivados tricíclicos de quinolina e quinoxalina, a uma composição farmacêutica contendo esses compostos, aos seus usos como moduladores, especialmente agonistas ou agonistas parciais do receptor 5-ht2c, ao uso na preparaçao de um medicamento para prevenir ou tratar as condições e doenças que respondem à modulação do receptor 5-ht2c, e a um método para prevenir ou tratar as condições e doenças que respondem à modulação do receptor 5-ht2c.
BR112015005743A 2012-09-14 2013-09-13 derivados tricíclicos de quinoxalina e quinolina BR112015005743A2 (pt)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261701531P 2012-09-14 2012-09-14
US201261701514P 2012-09-14 2012-09-14
US201361793033P 2013-03-15 2013-03-15
CN201310410951.1A CN104418862A (zh) 2013-09-11 2013-09-11 三环喹啉和喹喔啉衍生物
PCT/EP2013/069036 WO2014041131A1 (en) 2012-09-14 2013-09-13 Tricyclic quinoline and quinoxaline derivatives

Publications (1)

Publication Number Publication Date
BR112015005743A2 true BR112015005743A2 (pt) 2017-07-04

Family

ID=50275085

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015005743A BR112015005743A2 (pt) 2012-09-14 2013-09-13 derivados tricíclicos de quinoxalina e quinolina

Country Status (26)

Country Link
US (3) US10118926B2 (pt)
EP (1) EP2895485A1 (pt)
JP (1) JP6290217B2 (pt)
KR (1) KR20150056608A (pt)
CN (1) CN104995191A (pt)
AR (1) AR092568A1 (pt)
AU (2) AU2013314279B2 (pt)
BR (1) BR112015005743A2 (pt)
CA (1) CA2884548A1 (pt)
CL (1) CL2015000628A1 (pt)
CR (1) CR20150186A (pt)
DO (1) DOP2015000058A (pt)
EC (1) ECSP15012766A (pt)
HK (1) HK1212684A1 (pt)
IL (1) IL237726A0 (pt)
IN (1) IN2015DN02070A (pt)
MX (1) MX2015003364A (pt)
NZ (1) NZ631187A (pt)
PE (1) PE20150777A1 (pt)
PH (1) PH12015500551A1 (pt)
RU (1) RU2015113558A (pt)
SG (1) SG11201501894VA (pt)
TW (1) TW201414735A (pt)
UA (1) UA116216C2 (pt)
UY (1) UY35029A (pt)
WO (1) WO2014041131A1 (pt)

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UY35029A (es) 2014-04-30
AR092568A1 (es) 2015-04-22
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AU2013314279B2 (en) 2017-11-02
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JP6290217B2 (ja) 2018-03-07
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UA116216C2 (uk) 2018-02-26
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CR20150186A (es) 2015-08-28

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