KR20150056608A - 트리사이클릭 퀴놀린 및 퀴녹살린 유도체 - Google Patents

트리사이클릭 퀴놀린 및 퀴녹살린 유도체 Download PDF

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Publication number
KR20150056608A
KR20150056608A KR1020157009502A KR20157009502A KR20150056608A KR 20150056608 A KR20150056608 A KR 20150056608A KR 1020157009502 A KR1020157009502 A KR 1020157009502A KR 20157009502 A KR20157009502 A KR 20157009502A KR 20150056608 A KR20150056608 A KR 20150056608A
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South Korea
Prior art keywords
fluorinated
alkyl
alkoxy
ring
diazepino
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KR1020157009502A
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English (en)
Korean (ko)
Inventor
하네스 쿨맨
빌프리트 브라예
헬무트 마크
안드레아스 하우프트
아나 루시아 렐로
카를라 드레쉐
마르가레타 헨리카 마리아 바커
빅토르 라킥스
카롤린 호프트
뤼쉬 쉬
샤오나 자오
Original Assignee
아비에 도이치란트 게엠베하 운트 콤파니 카게
애브비 인코포레이티드
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50275085&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20150056608(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from CN201310410951.1A external-priority patent/CN104418862A/zh
Application filed by 아비에 도이치란트 게엠베하 운트 콤파니 카게, 애브비 인코포레이티드 filed Critical 아비에 도이치란트 게엠베하 운트 콤파니 카게
Publication of KR20150056608A publication Critical patent/KR20150056608A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
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    • A61P3/04—Anorexiants; Antiobesity agents
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    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16—Peri-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Urology & Nephrology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Psychology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Gynecology & Obstetrics (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020157009502A 2012-09-14 2013-09-13 트리사이클릭 퀴놀린 및 퀴녹살린 유도체 KR20150056608A (ko)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US201261701531P 2012-09-14 2012-09-14
US201261701514P 2012-09-14 2012-09-14
US61/701,514 2012-09-14
US61/701,531 2012-09-14
US201361793033P 2013-03-15 2013-03-15
US61/793,033 2013-03-15
CN201310410951.1A CN104418862A (zh) 2013-09-11 2013-09-11 三环喹啉和喹喔啉衍生物
CN201310410951.1 2013-09-11
PCT/EP2013/069036 WO2014041131A1 (en) 2012-09-14 2013-09-13 Tricyclic quinoline and quinoxaline derivatives

Publications (1)

Publication Number Publication Date
KR20150056608A true KR20150056608A (ko) 2015-05-26

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KR1020157009502A KR20150056608A (ko) 2012-09-14 2013-09-13 트리사이클릭 퀴놀린 및 퀴녹살린 유도체

Country Status (26)

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US (3) US10118926B2 (pt)
EP (1) EP2895485A1 (pt)
JP (1) JP6290217B2 (pt)
KR (1) KR20150056608A (pt)
CN (1) CN104995191A (pt)
AR (1) AR092568A1 (pt)
AU (2) AU2013314279B2 (pt)
BR (1) BR112015005743A2 (pt)
CA (1) CA2884548A1 (pt)
CL (1) CL2015000628A1 (pt)
CR (1) CR20150186A (pt)
DO (1) DOP2015000058A (pt)
EC (1) ECSP15012766A (pt)
HK (1) HK1212684A1 (pt)
IL (1) IL237726A0 (pt)
IN (1) IN2015DN02070A (pt)
MX (1) MX2015003364A (pt)
NZ (1) NZ631187A (pt)
PE (1) PE20150777A1 (pt)
PH (1) PH12015500551A1 (pt)
RU (1) RU2015113558A (pt)
SG (1) SG11201501894VA (pt)
TW (1) TW201414735A (pt)
UA (1) UA116216C2 (pt)
UY (1) UY35029A (pt)
WO (1) WO2014041131A1 (pt)

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WO2023068755A1 (ko) * 2021-10-18 2023-04-27 주식회사 사피엔스바이오 신규한 화합물 및 이를 포함하는 약학적 조성물

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US10118926B2 (en) 2018-11-06
US20140080816A1 (en) 2014-03-20
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CA2884548A1 (en) 2014-03-20
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