ID21350A - 2-sianopirolidina n-tersubstitusi - Google Patents

2-sianopirolidina n-tersubstitusi

Info

Publication number
ID21350A
ID21350A IDW990296D ID990296D ID21350A ID 21350 A ID21350 A ID 21350A ID W990296 D IDW990296 D ID W990296D ID 990296 D ID990296 D ID 990296D ID 21350 A ID21350 A ID 21350A
Authority
ID
Indonesia
Prior art keywords
sianopirolidina
substituted
Prior art date
Application number
IDW990296D
Other languages
English (en)
Indonesian (id)
Inventor
Edwin Bernard Villhauer
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25000236&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ID21350(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ID21350A publication Critical patent/ID21350A/id

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IDW990296D 1996-11-07 1997-11-05 2-sianopirolidina n-tersubstitusi ID21350A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US74629596A 1996-11-07 1996-11-07

Publications (1)

Publication Number Publication Date
ID21350A true ID21350A (id) 1999-05-27

Family

ID=25000236

Family Applications (2)

Application Number Title Priority Date Filing Date
IDW990296D ID21350A (id) 1996-11-07 1997-11-05 2-sianopirolidina n-tersubstitusi
IDP973634A ID18331A (id) 1996-11-07 1997-11-10 2-sianopirolidina n-tersubtitusi

Family Applications After (1)

Application Number Title Priority Date Filing Date
IDP973634A ID18331A (id) 1996-11-07 1997-11-10 2-sianopirolidina n-tersubtitusi

Country Status (28)

Country Link
EP (1) EP0937040B1 (fr)
JP (1) JP3217380B2 (fr)
KR (1) KR20000053081A (fr)
CN (1) CN1134412C (fr)
AR (1) AR009605A1 (fr)
AT (1) ATE271543T1 (fr)
AU (1) AU726186B2 (fr)
BR (1) BR9714130B1 (fr)
CA (1) CA2269810C (fr)
CO (1) CO4910126A1 (fr)
CZ (1) CZ296303B6 (fr)
DE (1) DE69729947T2 (fr)
ES (1) ES2226004T3 (fr)
HK (1) HK1022149A1 (fr)
HU (1) HU227125B1 (fr)
ID (2) ID21350A (fr)
IL (3) IL129561A0 (fr)
NO (1) NO312667B1 (fr)
NZ (1) NZ335146A (fr)
PE (1) PE10699A1 (fr)
PL (1) PL190498B1 (fr)
PT (1) PT937040E (fr)
RU (1) RU2180901C2 (fr)
SK (1) SK282904B6 (fr)
TR (1) TR199901004T2 (fr)
TW (1) TW492957B (fr)
WO (1) WO1998019998A2 (fr)
ZA (1) ZA979985B (fr)

Families Citing this family (249)

* Cited by examiner, † Cited by third party
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DE19828113A1 (de) 1998-06-24 2000-01-05 Probiodrug Ges Fuer Arzneim Prodrugs von Inhibitoren der Dipeptidyl Peptidase IV
DE19834591A1 (de) * 1998-07-31 2000-02-03 Probiodrug Ges Fuer Arzneim Verfahren zur Steigerung des Blutglukosespiegels in Säugern
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US7064145B2 (en) * 2000-02-25 2006-06-20 Novo Nordisk A/S Inhibition of beta cell degeneration
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TW583185B (en) * 2000-06-13 2004-04-11 Novartis Ag N-(substituted glycyl)-2-cyanopyrrolidines and pharmaceutical composition for inhibiting dipeptidyl peptidase-IV (DPP-IV) or for the prevention or treatment of diseases or conditions associated with elevated levels of DPP-IV comprising the same
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CA2269810A1 (fr) 1998-05-14
AU726186B2 (en) 2000-11-02
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IL129561A0 (en) 2000-02-29
CZ296303B6 (cs) 2006-02-15
RU2180901C2 (ru) 2002-03-27
CZ161599A3 (cs) 1999-08-11
DE69729947T2 (de) 2005-04-21
NO992028L (no) 1999-04-28
HU227125B1 (en) 2010-07-28
EP0937040A2 (fr) 1999-08-25
BR9714130B1 (pt) 2010-03-23
KR20000053081A (ko) 2000-08-25
IL158020A (en) 2007-03-08
AU5318498A (en) 1998-05-29
IL129561A (en) 2006-10-31
CN1134412C (zh) 2004-01-14
CA2269810C (fr) 2006-07-11
HK1022149A1 (en) 2000-07-28
JP2000511559A (ja) 2000-09-05
WO1998019998A3 (fr) 1998-07-16
BR9714130A (pt) 2000-02-29
CN1236361A (zh) 1999-11-24
AR009605A1 (es) 2000-04-26
HUP0000323A3 (en) 2002-02-28
CO4910126A1 (es) 2000-04-24
SK60899A3 (en) 2000-04-10
ZA979985B (en) 1998-05-07
PT937040E (pt) 2004-11-30
PL332777A1 (en) 1999-10-11
PL190498B1 (pl) 2005-12-30
ID18331A (id) 1998-03-26
SK282904B6 (sk) 2003-01-09
TW492957B (en) 2002-07-01
ES2226004T3 (es) 2005-03-16
EP0937040B1 (fr) 2004-07-21
NO992028D0 (no) 1999-04-28
WO1998019998A2 (fr) 1998-05-14
NO312667B1 (no) 2002-06-17
ATE271543T1 (de) 2004-08-15
PE10699A1 (es) 1999-03-02
HUP0000323A2 (hu) 2000-08-28
JP3217380B2 (ja) 2001-10-09
TR199901004T2 (xx) 1999-07-21

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