ID21350A - 2-sianopirolidina n-tersubstitusi - Google Patents

2-sianopirolidina n-tersubstitusi

Info

Publication number
ID21350A
ID21350A IDW990296D ID990296D ID21350A ID 21350 A ID21350 A ID 21350A ID W990296 D IDW990296 D ID W990296D ID 990296 D ID990296 D ID 990296D ID 21350 A ID21350 A ID 21350A
Authority
ID
Indonesia
Prior art keywords
sianopirolidina
substituted
Prior art date
Application number
IDW990296D
Other languages
English (en)
Indonesian (id)
Inventor
Edwin Bernard Villhauer
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25000236&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ID21350(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of ID21350A publication Critical patent/ID21350A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IDW990296D 1996-11-07 1997-11-05 2-sianopirolidina n-tersubstitusi ID21350A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US74629596A 1996-11-07 1996-11-07

Publications (1)

Publication Number Publication Date
ID21350A true ID21350A (id) 1999-05-27

Family

ID=25000236

Family Applications (2)

Application Number Title Priority Date Filing Date
IDW990296D ID21350A (id) 1996-11-07 1997-11-05 2-sianopirolidina n-tersubstitusi
IDP973634A ID18331A (id) 1996-11-07 1997-11-10 2-sianopirolidina n-tersubtitusi

Family Applications After (1)

Application Number Title Priority Date Filing Date
IDP973634A ID18331A (id) 1996-11-07 1997-11-10 2-sianopirolidina n-tersubtitusi

Country Status (28)

Country Link
EP (1) EP0937040B1 (fr)
JP (1) JP3217380B2 (fr)
KR (1) KR20000053081A (fr)
CN (1) CN1134412C (fr)
AR (1) AR009605A1 (fr)
AT (1) ATE271543T1 (fr)
AU (1) AU726186B2 (fr)
BR (1) BR9714130B1 (fr)
CA (1) CA2269810C (fr)
CO (1) CO4910126A1 (fr)
CZ (1) CZ296303B6 (fr)
DE (1) DE69729947T2 (fr)
ES (1) ES2226004T3 (fr)
HK (1) HK1022149A1 (fr)
HU (1) HU227125B1 (fr)
ID (2) ID21350A (fr)
IL (3) IL129561A0 (fr)
NO (1) NO312667B1 (fr)
NZ (1) NZ335146A (fr)
PE (1) PE10699A1 (fr)
PL (1) PL190498B1 (fr)
PT (1) PT937040E (fr)
RU (1) RU2180901C2 (fr)
SK (1) SK282904B6 (fr)
TR (1) TR199901004T2 (fr)
TW (1) TW492957B (fr)
WO (1) WO1998019998A2 (fr)
ZA (1) ZA979985B (fr)

Families Citing this family (249)

* Cited by examiner, † Cited by third party
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DE19828113A1 (de) 1998-06-24 2000-01-05 Probiodrug Ges Fuer Arzneim Prodrugs von Inhibitoren der Dipeptidyl Peptidase IV
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US7064145B2 (en) * 2000-02-25 2006-06-20 Novo Nordisk A/S Inhibition of beta cell degeneration
US6395767B2 (en) * 2000-03-10 2002-05-28 Bristol-Myers Squibb Company Cyclopropyl-fused pyrrolidine-based inhibitors of dipeptidyl peptidase IV and method
IL151368A0 (en) * 2000-03-31 2003-04-10 Probiodrug Ag Use of a dipeptidyl peptidase iv enzyme activity effector for the production of pharmaceutical compositions
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TW583185B (en) * 2000-06-13 2004-04-11 Novartis Ag N-(substituted glycyl)-2-cyanopyrrolidines and pharmaceutical composition for inhibiting dipeptidyl peptidase-IV (DPP-IV) or for the prevention or treatment of diseases or conditions associated with elevated levels of DPP-IV comprising the same
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US7368421B2 (en) 2001-06-27 2008-05-06 Probiodrug Ag Use of dipeptidyl peptidase IV inhibitors in the treatment of multiple sclerosis
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US6861440B2 (en) 2001-10-26 2005-03-01 Hoffmann-La Roche Inc. DPP IV inhibitors
CA2468192A1 (fr) 2001-11-26 2003-06-05 Trustees Of Tufts College Inhibiteurs peptidomimetiques d'enzymes de clivage post-proline
EP1487471A4 (fr) 2001-11-26 2010-03-10 Tufts College Techniques de traitement de maladies auto-immunes et reactifs associes
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AU2003248259A1 (en) * 2002-07-10 2004-02-02 Yamanouchi Pharmaceutical Co., Ltd. Novel azetidine derivative or salt thereof
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DE69729947D1 (de) 2004-08-26
CA2269810A1 (fr) 1998-05-14
AU726186B2 (en) 2000-11-02
NZ335146A (en) 1999-11-29
IL129561A0 (en) 2000-02-29
CZ296303B6 (cs) 2006-02-15
RU2180901C2 (ru) 2002-03-27
CZ161599A3 (cs) 1999-08-11
DE69729947T2 (de) 2005-04-21
NO992028L (no) 1999-04-28
HU227125B1 (en) 2010-07-28
EP0937040A2 (fr) 1999-08-25
BR9714130B1 (pt) 2010-03-23
KR20000053081A (ko) 2000-08-25
IL158020A (en) 2007-03-08
AU5318498A (en) 1998-05-29
IL129561A (en) 2006-10-31
CN1134412C (zh) 2004-01-14
CA2269810C (fr) 2006-07-11
HK1022149A1 (en) 2000-07-28
JP2000511559A (ja) 2000-09-05
WO1998019998A3 (fr) 1998-07-16
BR9714130A (pt) 2000-02-29
CN1236361A (zh) 1999-11-24
AR009605A1 (es) 2000-04-26
HUP0000323A3 (en) 2002-02-28
CO4910126A1 (es) 2000-04-24
SK60899A3 (en) 2000-04-10
ZA979985B (en) 1998-05-07
PT937040E (pt) 2004-11-30
PL332777A1 (en) 1999-10-11
PL190498B1 (pl) 2005-12-30
ID18331A (id) 1998-03-26
SK282904B6 (sk) 2003-01-09
TW492957B (en) 2002-07-01
ES2226004T3 (es) 2005-03-16
EP0937040B1 (fr) 2004-07-21
NO992028D0 (no) 1999-04-28
WO1998019998A2 (fr) 1998-05-14
NO312667B1 (no) 2002-06-17
ATE271543T1 (de) 2004-08-15
PE10699A1 (es) 1999-03-02
HUP0000323A2 (hu) 2000-08-28
JP3217380B2 (ja) 2001-10-09
TR199901004T2 (xx) 1999-07-21

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