HRP20150945T1 - Postupci za proizvodnju derivata benzil-benzena supstituiranog glukopiranozilom - Google Patents

Postupci za proizvodnju derivata benzil-benzena supstituiranog glukopiranozilom Download PDF

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Publication number
HRP20150945T1
HRP20150945T1 HRP20150945TT HRP20150945T HRP20150945T1 HR P20150945 T1 HRP20150945 T1 HR P20150945T1 HR P20150945T T HRP20150945T T HR P20150945TT HR P20150945 T HRP20150945 T HR P20150945T HR P20150945 T1 HRP20150945 T1 HR P20150945T1
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Croatia
Prior art keywords
alkyl
acid
phenyl
tetrahydrofuran
denotes
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HRP20150945TT
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English (en)
Croatian (hr)
Inventor
Dirk Weber
Tobias Fiedler
Christian Filser
Rainer Hamm
Simone Orlich
Matthias Post
Svenja Renner
Xiao-Jun Wang
Thomas Wirth
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Boehringer Ingelheim International Gmbh
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Application filed by Boehringer Ingelheim International Gmbh filed Critical Boehringer Ingelheim International Gmbh
Publication of HRP20150945T1 publication Critical patent/HRP20150945T1/hr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C07D309/12—Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C07H1/06—Separation; Purification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Packaging Of Annular Or Rod-Shaped Articles, Wearing Apparel, Cassettes, Or The Like (AREA)
  • Wrapping Of Specific Fragile Articles (AREA)
HRP20150945TT 2009-09-30 2010-09-24 Postupci za proizvodnju derivata benzil-benzena supstituiranog glukopiranozilom HRP20150945T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24714409P 2009-09-30 2009-09-30
PCT/EP2010/064120 WO2011039108A2 (en) 2009-09-30 2010-09-24 Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives
EP10762899.2A EP2486029B1 (en) 2009-09-30 2010-09-24 Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives

Publications (1)

Publication Number Publication Date
HRP20150945T1 true HRP20150945T1 (hr) 2015-10-09

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HRP20150945TT HRP20150945T1 (hr) 2009-09-30 2010-09-24 Postupci za proizvodnju derivata benzil-benzena supstituiranog glukopiranozilom

Country Status (25)

Country Link
US (2) US9024010B2 (instruction)
EP (1) EP2486029B1 (instruction)
JP (1) JP5758900B2 (instruction)
KR (1) KR101813025B1 (instruction)
CN (1) CN102574829B (instruction)
AR (1) AR078193A1 (instruction)
AU (1) AU2010303124B2 (instruction)
BR (1) BR112012007085B8 (instruction)
CA (1) CA2775962C (instruction)
CL (1) CL2012000581A1 (instruction)
DK (1) DK2486029T3 (instruction)
EA (1) EA022032B1 (instruction)
ES (1) ES2546762T3 (instruction)
HR (1) HRP20150945T1 (instruction)
HU (1) HUE026133T2 (instruction)
IL (1) IL218101A0 (instruction)
IN (1) IN2012DN02751A (instruction)
MX (1) MX2012003048A (instruction)
NZ (1) NZ598366A (instruction)
PH (1) PH12012500634A1 (instruction)
PL (1) PL2486029T3 (instruction)
PT (1) PT2486029E (instruction)
SI (1) SI2486029T1 (instruction)
TW (1) TWI465458B (instruction)
WO (1) WO2011039108A2 (instruction)

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CN102574829B (zh) 2015-07-01
EP2486029A2 (en) 2012-08-15
SI2486029T1 (sl) 2015-10-30
IL218101A0 (en) 2012-04-30
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