HRP20030647A2 - Isoxazoline derivatives as anti-depressants - Google Patents
Isoxazoline derivatives as anti-depressants Download PDFInfo
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- HRP20030647A2 HRP20030647A2 HR20030647A HRP20030647A HRP20030647A2 HR P20030647 A2 HRP20030647 A2 HR P20030647A2 HR 20030647 A HR20030647 A HR 20030647A HR P20030647 A HRP20030647 A HR P20030647A HR P20030647 A2 HRP20030647 A2 HR P20030647A2
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Child & Adolescent Psychology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP01200611 | 2001-02-21 | ||
EP01201264 | 2001-04-05 | ||
PCT/EP2002/001567 WO2002066484A1 (en) | 2001-02-21 | 2002-02-13 | Isoxazoline derivatives as anti-depressants |
Publications (1)
Publication Number | Publication Date |
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HRP20030647A2 true HRP20030647A2 (en) | 2005-06-30 |
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Family Applications (1)
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HR20030647A HRP20030647A2 (en) | 2001-02-21 | 2003-08-12 | Isoxazoline derivatives as anti-depressants |
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US (1) | US7169786B2 (de) |
EP (1) | EP1368358B1 (de) |
JP (1) | JP3953424B2 (de) |
KR (1) | KR100848898B1 (de) |
CN (1) | CN100400540C (de) |
AR (1) | AR035685A1 (de) |
AT (1) | ATE337322T1 (de) |
AU (1) | AU2002244717B2 (de) |
BG (1) | BG107984A (de) |
BR (1) | BR0207433A (de) |
CA (1) | CA2437505C (de) |
CY (1) | CY1106448T1 (de) |
CZ (1) | CZ20032515A3 (de) |
DE (1) | DE60214138T2 (de) |
DK (1) | DK1368358T3 (de) |
EA (1) | EA006747B1 (de) |
EE (1) | EE200300398A (de) |
EG (1) | EG23929A (de) |
ES (1) | ES2271230T3 (de) |
HK (1) | HK1065537A1 (de) |
HR (1) | HRP20030647A2 (de) |
HU (1) | HUP0303270A3 (de) |
IL (2) | IL157470A0 (de) |
MX (1) | MXPA03007432A (de) |
MY (1) | MY137836A (de) |
NO (1) | NO20033700L (de) |
NZ (1) | NZ526741A (de) |
PL (1) | PL208593B1 (de) |
PT (1) | PT1368358E (de) |
SI (1) | SI1368358T1 (de) |
SK (1) | SK11612003A3 (de) |
TW (1) | TWI257392B (de) |
WO (1) | WO2002066484A1 (de) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0203299D0 (en) * | 2002-02-12 | 2002-03-27 | Glaxo Group Ltd | Novel compounds |
WO2003082878A1 (en) * | 2002-04-02 | 2003-10-09 | Janssen Pharmaceutica N.V. | Substituted amino isoxazoline derivatives and their use as anti-depressants. |
TW200409777A (en) * | 2002-08-12 | 2004-06-16 | Janssen Pharmaceutica Nv | C-substituted tricyclic isoxazoline derivatives and their use as anti-depressants |
EP1554286B1 (de) * | 2002-08-15 | 2010-01-27 | Janssen Pharmaceutica N.V. | Kondensierte heterocyclische isoxazolinderivate und deren verwendung als antidepressiva |
EP1532155B1 (de) * | 2002-08-21 | 2008-02-27 | Janssen Pharmaceutica N.V. | C6- UND C9-SUBSTITUIERTE CHROMENO[4,3-c]ISOXAZOLINE UND IHRE VERWENDUNG ALS ANTI-DEPRESSIVA |
KR20050114641A (ko) | 2003-03-07 | 2005-12-06 | 아스텔라스세이야쿠 가부시키가이샤 | 2,6-이치환된 스티릴을 갖는 질소 함유 헤테로환 유도체 |
ATE420881T1 (de) | 2003-09-17 | 2009-01-15 | Janssen Pharmaceutica Nv | Kondensierte heterocyclische verbindungen als modulatoren des serotoninrezeptors |
EP1905774B1 (de) * | 2003-09-17 | 2013-02-20 | Janssen Pharmaceutica N.V. | Kondensierte heterocyclische Verbindungen als Modulatoren des Serotoninrezeptors |
DE602005016836D1 (de) * | 2004-11-26 | 2009-11-05 | Janssen Pharmaceutica Nv | Chotischer und anxiolytischer aktivität |
MX2009009447A (es) * | 2007-03-09 | 2009-09-14 | Sanofi Aventis | Dihidro y tetrahidro oxazolopirimidinonas sustituidas, preparacion y uso de las mismas. |
US7863266B2 (en) * | 2007-06-08 | 2011-01-04 | Helicon Therapeutics, Inc. | Therapeutic pyrazoloquinoline urea derivatives |
EP2236511A4 (de) | 2007-12-21 | 2011-04-13 | Alla Chem Llc | Liganden von alpha-adrenoceptoren und von dopamin-, histamin-, imidazolin- und serotoninrezeptoren und anwendung davon |
AR078171A1 (es) | 2009-09-15 | 2011-10-19 | Sanofi Aventis | Dihidrobenzocicloalquiloximetil-oxazolopirimidinonas sustituidas, preparacion y uso de las mismas |
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ES2055011T3 (es) | 1988-09-19 | 1994-08-16 | Akzo Nv | Un procedimiento para la preparacion de derivados de tetrahidronaftaleno e indano. |
US5880121A (en) * | 1996-01-05 | 1999-03-09 | Hoechst Marion Roussel Inc. | 4,5-dihydronaphth (1,2-c) isoxazoles and derivatives thereof |
PT892804E (pt) * | 1996-04-12 | 2003-01-31 | Janssen Pharmaceutica Nv | Derivados de isoxazolidina |
HUP9602763A3 (en) * | 1996-10-09 | 1999-05-28 | Egyt Gyogyszervegyeszeti Gyar | 3-phenyl isoxazole derivatives, process for producing them and pharmaceutical compositions containing the same |
EP1119568B1 (de) * | 1998-10-09 | 2004-02-18 | Janssen Pharmaceutica N.V. | 4,5-dehydroisoxazole derivate und ihre pharmazeutische verwendung |
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