EE200300398A - Isoksasoliini derivaat, selle saamine ja kasutamine depresioonivastase ravimi valmistamiseks ning seda sisaldav ravimkompositsioon - Google Patents
Isoksasoliini derivaat, selle saamine ja kasutamine depresioonivastase ravimi valmistamiseks ning seda sisaldav ravimkompositsioonInfo
- Publication number
- EE200300398A EE200300398A EEP200300398A EEP200300398A EE200300398A EE 200300398 A EE200300398 A EE 200300398A EE P200300398 A EEP200300398 A EE P200300398A EE P200300398 A EEP200300398 A EE P200300398A EE 200300398 A EE200300398 A EE 200300398A
- Authority
- EE
- Estonia
- Prior art keywords
- preparation
- pharmaceutical composition
- composition containing
- isoxazoline derivative
- medicament
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Child & Adolescent Psychology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP01200611 | 2001-02-21 | ||
EP01201264 | 2001-04-05 | ||
PCT/EP2002/001567 WO2002066484A1 (en) | 2001-02-21 | 2002-02-13 | Isoxazoline derivatives as anti-depressants |
Publications (1)
Publication Number | Publication Date |
---|---|
EE200300398A true EE200300398A (et) | 2003-12-15 |
Family
ID=26076836
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EEP200300398A EE200300398A (et) | 2001-02-21 | 2002-02-13 | Isoksasoliini derivaat, selle saamine ja kasutamine depresioonivastase ravimi valmistamiseks ning seda sisaldav ravimkompositsioon |
Country Status (33)
Country | Link |
---|---|
US (1) | US7169786B2 (et) |
EP (1) | EP1368358B1 (et) |
JP (1) | JP3953424B2 (et) |
KR (1) | KR100848898B1 (et) |
CN (1) | CN100400540C (et) |
AR (1) | AR035685A1 (et) |
AT (1) | ATE337322T1 (et) |
AU (1) | AU2002244717B2 (et) |
BG (1) | BG107984A (et) |
BR (1) | BR0207433A (et) |
CA (1) | CA2437505C (et) |
CY (1) | CY1106448T1 (et) |
CZ (1) | CZ20032515A3 (et) |
DE (1) | DE60214138T2 (et) |
DK (1) | DK1368358T3 (et) |
EA (1) | EA006747B1 (et) |
EE (1) | EE200300398A (et) |
EG (1) | EG23929A (et) |
ES (1) | ES2271230T3 (et) |
HK (1) | HK1065537A1 (et) |
HR (1) | HRP20030647A2 (et) |
HU (1) | HUP0303270A3 (et) |
IL (2) | IL157470A0 (et) |
MX (1) | MXPA03007432A (et) |
MY (1) | MY137836A (et) |
NO (1) | NO20033700L (et) |
NZ (1) | NZ526741A (et) |
PL (1) | PL208593B1 (et) |
PT (1) | PT1368358E (et) |
SI (1) | SI1368358T1 (et) |
SK (1) | SK11612003A3 (et) |
TW (1) | TWI257392B (et) |
WO (1) | WO2002066484A1 (et) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0203299D0 (en) * | 2002-02-12 | 2002-03-27 | Glaxo Group Ltd | Novel compounds |
EP1492796B1 (en) * | 2002-04-02 | 2007-09-05 | Janssen Pharmaceutica N.V. | Substituted amino isoxazoline derivatives and their use as anti-depressants. |
AR040967A1 (es) * | 2002-08-12 | 2005-04-27 | Janssen Pharmaceutica Nv | Derivados de isoxazolina triciclicos c- sustituidos y su uso como anti- depresivos |
CA2494557C (en) * | 2002-08-15 | 2011-10-18 | Janssen Pharmaceutica N.V. | Fused heterocyclic isoxazoline derivatives and their use as anti-depressants |
WO2004018482A2 (en) * | 2002-08-21 | 2004-03-04 | Janssen Pharmaceutica N.V. | C6- and c9-substituted chromeno[4, 3-c]isoxazoline derivatives and their use as anti-depressants |
WO2004078715A1 (ja) * | 2003-03-07 | 2004-09-16 | Astellas Pharma Inc. | 2,6-ジ置換スチリルを有する含窒素へテロ環誘導体 |
EP1944306A1 (en) * | 2003-09-17 | 2008-07-16 | Janssen Pharmaceutica, N.V. | Fused heterocyclic compounds as serotonin receptor modulators |
EA200801812A1 (ru) | 2003-09-17 | 2009-06-30 | Янссен Фармацевтика Н.В. | Сопряженные гетероциклические соединения |
ES2331144T3 (es) * | 2004-11-26 | 2009-12-22 | Janssen Pharmaceutica Nv | Derivados de isoxazolina-indol con actividad antipsicotica y ansiolitica mejorada. |
AU2008226649B2 (en) * | 2007-03-09 | 2013-08-01 | Sanofi | Substituted dihydro and tetrahydro oxazolopyrimidinones, preparation and use thereof |
JP2010529144A (ja) * | 2007-06-08 | 2010-08-26 | ヘリコン・セラピューティクス・インコーポレーテッド | 治療用ピラゾロキノリン尿素誘導体 |
WO2009082268A2 (ru) | 2007-12-21 | 2009-07-02 | Alla Chem, Llc | ЛИГАНДЫ α-АДРЕНОЦЕПТОРОВ, ДОПАМИНОВЫХ, ГИСТАМИНОВЫХ, ИМИДАЗОЛИНОВЫХ И СЕРОТОНИНОВЫХ РЕЦЕПТОРОВ И ИХ ПРИМЕНЕНИЕ |
AR078171A1 (es) | 2009-09-15 | 2011-10-19 | Sanofi Aventis | Dihidrobenzocicloalquiloximetil-oxazolopirimidinonas sustituidas, preparacion y uso de las mismas |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0361577B1 (en) * | 1988-09-19 | 1993-05-05 | Akzo N.V. | Tetrahydronaphthalene and indane derivatives |
US5880121A (en) * | 1996-01-05 | 1999-03-09 | Hoechst Marion Roussel Inc. | 4,5-dihydronaphth (1,2-c) isoxazoles and derivatives thereof |
NZ329954A (en) * | 1996-04-12 | 1999-07-29 | Janssen Pharmaceutica Nv | Isoxazolidine tetracyclic and tricyclic ring system derivatives and medicaments |
HUP9602763A3 (en) * | 1996-10-09 | 1999-05-28 | Egyt Gyogyszervegyeszeti Gyar | 3-phenyl isoxazole derivatives, process for producing them and pharmaceutical compositions containing the same |
ATE259803T1 (de) * | 1998-10-09 | 2004-03-15 | Janssen Pharmaceutica Nv | 4,5-dehydroisoxazole derivate und ihre pharmazeutische verwendung |
-
2002
- 2002-02-13 JP JP2002565998A patent/JP3953424B2/ja not_active Expired - Lifetime
- 2002-02-13 IL IL15747002A patent/IL157470A0/xx unknown
- 2002-02-13 BR BR0207433-8A patent/BR0207433A/pt not_active IP Right Cessation
- 2002-02-13 EP EP02712909A patent/EP1368358B1/en not_active Expired - Lifetime
- 2002-02-13 NZ NZ526741A patent/NZ526741A/en unknown
- 2002-02-13 ES ES02712909T patent/ES2271230T3/es not_active Expired - Lifetime
- 2002-02-13 CA CA2437505A patent/CA2437505C/en not_active Expired - Lifetime
- 2002-02-13 HU HU0303270A patent/HUP0303270A3/hu unknown
- 2002-02-13 EA EA200300915A patent/EA006747B1/ru not_active IP Right Cessation
- 2002-02-13 WO PCT/EP2002/001567 patent/WO2002066484A1/en active IP Right Grant
- 2002-02-13 DK DK02712909T patent/DK1368358T3/da active
- 2002-02-13 US US10/468,555 patent/US7169786B2/en not_active Expired - Lifetime
- 2002-02-13 KR KR1020037008328A patent/KR100848898B1/ko not_active IP Right Cessation
- 2002-02-13 EE EEP200300398A patent/EE200300398A/et unknown
- 2002-02-13 MX MXPA03007432A patent/MXPA03007432A/es active IP Right Grant
- 2002-02-13 AT AT02712909T patent/ATE337322T1/de not_active IP Right Cessation
- 2002-02-13 SI SI200230433T patent/SI1368358T1/sl unknown
- 2002-02-13 AU AU2002244717A patent/AU2002244717B2/en not_active Expired
- 2002-02-13 SK SK1161-2003A patent/SK11612003A3/sk unknown
- 2002-02-13 PL PL363264A patent/PL208593B1/pl unknown
- 2002-02-13 CZ CZ20032515A patent/CZ20032515A3/cs unknown
- 2002-02-13 CN CNB028052439A patent/CN100400540C/zh not_active Expired - Fee Related
- 2002-02-13 DE DE60214138T patent/DE60214138T2/de not_active Expired - Lifetime
- 2002-02-13 PT PT02712909T patent/PT1368358E/pt unknown
- 2002-02-19 MY MYPI20020548A patent/MY137836A/en unknown
- 2002-02-19 EG EG20020197A patent/EG23929A/xx active
- 2002-02-20 TW TW091102853A patent/TWI257392B/zh not_active IP Right Cessation
- 2002-02-20 AR ARP020100583A patent/AR035685A1/es unknown
-
2003
- 2003-07-08 BG BG107984A patent/BG107984A/bg unknown
- 2003-08-12 HR HR20030647A patent/HRP20030647A2/hr not_active Application Discontinuation
- 2003-08-19 IL IL157470A patent/IL157470A/en unknown
- 2003-08-20 NO NO20033700A patent/NO20033700L/no not_active Application Discontinuation
-
2004
- 2004-10-25 HK HK04108329.1A patent/HK1065537A1/xx not_active IP Right Cessation
-
2006
- 2006-11-22 CY CY20061101693T patent/CY1106448T1/el unknown
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