HK1093429A1 - Compounds effecting glucokinase - Google Patents
Compounds effecting glucokinaseInfo
- Publication number
- HK1093429A1 HK1093429A1 HK06113586.7A HK06113586A HK1093429A1 HK 1093429 A1 HK1093429 A1 HK 1093429A1 HK 06113586 A HK06113586 A HK 06113586A HK 1093429 A1 HK1093429 A1 HK 1093429A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- glucokinase
- compounds effecting
- compounds
- effecting glucokinase
- effecting
- Prior art date
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- Pyridine Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
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Application Number | Priority Date | Filing Date | Title |
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SE0102764A SE0102764D0 (sv) | 2001-08-17 | 2001-08-17 | Compounds |
HK05108225A HK1076042A1 (en) | 2001-08-17 | 2004-09-28 | Compounds affecting glucokinase |
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HK1093429A1 true HK1093429A1 (en) | 2007-03-02 |
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HK06113586.7A HK1093429A1 (en) | 2001-08-17 | 2004-09-28 | Compounds effecting glucokinase |
HK05108225A HK1076042A1 (en) | 2001-08-17 | 2004-09-28 | Compounds affecting glucokinase |
HK05111879A HK1079692A1 (en) | 2001-08-17 | 2004-09-28 | Compounds effecting glucokinase |
HK06110634.5A HK1089958A1 (en) | 2001-08-17 | 2004-09-28 | Compounds effecting glucokinase |
HK04107483A HK1064598A1 (en) | 2001-08-17 | 2004-09-28 | Compounds effecting glucokinase |
HK06110673A HK1089960A1 (en) | 2001-08-17 | 2006-09-25 | Compound effecting glucokinase |
HK06110762.9A HK1089966A1 (en) | 2001-08-17 | 2006-09-27 | Compounds effecting glucokinase |
HK06110988A HK1090291A1 (en) | 2001-08-17 | 2006-10-04 | Compounds effecting glucokinase |
HK06111020.5A HK1090292A1 (en) | 2001-08-17 | 2006-10-05 | Compounds effecting glukokinase |
HK06111482.6A HK1090839A1 (en) | 2001-08-17 | 2006-10-18 | Compounds effecting glucokinase |
Family Applications After (9)
Application Number | Title | Priority Date | Filing Date |
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HK05108225A HK1076042A1 (en) | 2001-08-17 | 2004-09-28 | Compounds affecting glucokinase |
HK05111879A HK1079692A1 (en) | 2001-08-17 | 2004-09-28 | Compounds effecting glucokinase |
HK06110634.5A HK1089958A1 (en) | 2001-08-17 | 2004-09-28 | Compounds effecting glucokinase |
HK04107483A HK1064598A1 (en) | 2001-08-17 | 2004-09-28 | Compounds effecting glucokinase |
HK06110673A HK1089960A1 (en) | 2001-08-17 | 2006-09-25 | Compound effecting glucokinase |
HK06110762.9A HK1089966A1 (en) | 2001-08-17 | 2006-09-27 | Compounds effecting glucokinase |
HK06110988A HK1090291A1 (en) | 2001-08-17 | 2006-10-04 | Compounds effecting glucokinase |
HK06111020.5A HK1090292A1 (en) | 2001-08-17 | 2006-10-05 | Compounds effecting glukokinase |
HK06111482.6A HK1090839A1 (en) | 2001-08-17 | 2006-10-18 | Compounds effecting glucokinase |
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EP (12) | EP1695705B1 (da) |
JP (2) | JP3987829B2 (da) |
KR (1) | KR100920439B1 (da) |
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HK (10) | HK1093429A1 (da) |
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NZ (1) | NZ531193A (da) |
PL (1) | PL368970A1 (da) |
PT (5) | PT1661563E (da) |
RU (1) | RU2329043C9 (da) |
SE (1) | SE0102764D0 (da) |
SI (5) | SI1568367T1 (da) |
TW (1) | TWI333855B (da) |
UA (1) | UA83182C2 (da) |
WO (1) | WO2003015774A1 (da) |
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JPWO2003097824A1 (ja) | 2002-05-16 | 2005-09-15 | 萬有製薬株式会社 | グルコキナーゼタンパク質の結晶、及びその結晶を用いたドラッグデザイン方法 |
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JPWO2004007472A1 (ja) | 2002-07-10 | 2005-11-17 | 小野薬品工業株式会社 | Ccr4アンタゴニストおよびその医薬用途 |
WO2004031179A1 (en) | 2002-10-03 | 2004-04-15 | F. Hoffmann-La Roche Ag | Indole-3-carboxamides as glucokinase (gk) activators |
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MXPA05009059A (es) | 2003-02-26 | 2005-10-19 | Banyu Pharma Co Ltd | Derivados de heteroarilcarbamoilbenceno. |
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US7767670B2 (en) | 2003-11-13 | 2010-08-03 | Ambit Biosciences Corporation | Substituted 3-carboxamido isoxazoles as kinase modulators |
KR20060105872A (ko) | 2003-12-29 | 2006-10-11 | 반유 세이야꾸 가부시끼가이샤 | 신규한 2-헤테로아릴 치환된 벤즈이미다졸 유도체 |
JP5033119B2 (ja) | 2005-04-25 | 2012-09-26 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング | キナーゼ阻害剤としての新規アザ複素環化合物 |
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Effective date: 20120815 |