FI67555C - Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t Download PDF

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Publication number
FI67555C
FI67555C FI791678A FI791678A FI67555C FI 67555 C FI67555 C FI 67555C FI 791678 A FI791678 A FI 791678A FI 791678 A FI791678 A FI 791678A FI 67555 C FI67555 C FI 67555C
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FI
Finland
Prior art keywords
compound
formula
group
acid
cef
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Application number
FI791678A
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English (en)
Finnish (fi)
Other versions
FI67555B (fi
FI791678A (fi
Inventor
Cynthia Hilda O'callaghan
David George Hubert Livermore
Christopher Earle Mewall
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Glaxo Group Ltd
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Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of FI791678A publication Critical patent/FI791678A/fi
Priority to FI801609A priority Critical patent/FI67705C/fi
Publication of FI67555B publication Critical patent/FI67555B/fi
Application granted granted Critical
Publication of FI67555C publication Critical patent/FI67555C/fi

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
FI791678A 1978-05-26 1979-05-25 Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t FI67555C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI801609A FI67705C (fi) 1978-05-26 1980-05-19 Foerfarande foer framstaellning av terapeutiskt anvaendbara (6,7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(substituerad oxiimi noacetamido)-(eventuellt substituerat pyridiniummetyl)cef-3 -e-4-karboxylatfoereningar

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB2291378 1978-05-26
GB2291178 1978-05-26
GB2291178 1978-05-26
GB2291378 1978-05-26

Publications (3)

Publication Number Publication Date
FI791678A FI791678A (fi) 1979-11-27
FI67555B FI67555B (fi) 1984-12-31
FI67555C true FI67555C (fi) 1985-04-10

Family

ID=26256190

Family Applications (2)

Application Number Title Priority Date Filing Date
FI791678A FI67555C (fi) 1978-05-26 1979-05-25 Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t
FI801609A FI67705C (fi) 1978-05-26 1980-05-19 Foerfarande foer framstaellning av terapeutiskt anvaendbara (6,7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(substituerad oxiimi noacetamido)-(eventuellt substituerat pyridiniummetyl)cef-3 -e-4-karboxylatfoereningar

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI801609A FI67705C (fi) 1978-05-26 1980-05-19 Foerfarande foer framstaellning av terapeutiskt anvaendbara (6,7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(substituerad oxiimi noacetamido)-(eventuellt substituerat pyridiniummetyl)cef-3 -e-4-karboxylatfoereningar

Country Status (27)

Country Link
US (2) US4258041A (no)
AR (2) AR228726A1 (no)
AT (1) AT370420B (no)
AU (1) AU524671B2 (no)
CA (1) CA1127633A (no)
CH (2) CH649556A5 (no)
DE (1) DE2921316C2 (no)
DK (1) DK157685C (no)
ES (2) ES480914A1 (no)
FI (2) FI67555C (no)
FR (2) FR2426695A1 (no)
HK (1) HK40183A (no)
IE (2) IE49172B1 (no)
IL (3) IL57400A (no)
IT (1) IT1116198B (no)
KE (1) KE3252A (no)
LU (1) LU81319A1 (no)
MY (1) MY8400017A (no)
NL (2) NL176855C (no)
NO (2) NO155347C (no)
NZ (2) NZ190558A (no)
PH (1) PH16961A (no)
PT (2) PT69669A (no)
SE (2) SE438507B (no)
SG (1) SG58382G (no)
SI (2) SI7911231A8 (no)
YU (2) YU41635B (no)

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IL57400A (en) 1982-08-31
YU223482A (en) 1983-04-30
CH646178A5 (de) 1984-11-15
US4258041A (en) 1981-03-24
IL59793A0 (en) 1980-06-30
NL176855B (nl) 1985-01-16
DK157685C (da) 1990-07-09
AR228726A1 (es) 1983-04-15
FR2426695A1 (fr) 1979-12-21
IE802453L (en) 1979-11-26
ES480915A1 (es) 1980-02-01
FR2445835B1 (no) 1983-06-03
NZ190558A (en) 1982-05-31
YU123179A (en) 1983-01-21
IE49173B1 (en) 1985-08-21
IE791025L (en) 1979-11-26
AU524671B2 (en) 1982-09-30
ATA239281A (de) 1982-08-15
IL57400A0 (en) 1979-09-30
YU41635B (en) 1987-12-31
PH16961A (en) 1984-04-27
FR2445835A1 (fr) 1980-08-01
FI67555B (fi) 1984-12-31
US4600772A (en) 1986-07-15
NL176855C (nl) 1985-06-17
FR2426695B1 (no) 1982-06-11
PT69669A (en) 1979-06-01
NL8001348A (nl) 1980-06-30
NZ193326A (en) 1982-05-31
YU43097B (en) 1989-02-28
IL59793A (en) 1982-08-31
CH649556A5 (de) 1985-05-31
NO155347B (no) 1966-12-08
FI791678A (fi) 1979-11-27
ES480914A1 (es) 1980-02-01
AR229883A1 (es) 1983-12-30
KE3252A (en) 1983-01-28
SE8402887D0 (sv) 1984-05-28
DE2921316A1 (de) 1979-12-06
IE49172B1 (en) 1985-08-21
DK216779A (da) 1979-11-27
SE438507B (sv) 1985-04-22
IT1116198B (it) 1986-02-10
SG58382G (en) 1983-09-02
NL7904122A (nl) 1979-11-28
NO155347C (no) 1987-03-18
SI8212234A8 (en) 1997-06-30
HK40183A (en) 1983-10-21
SE7904576L (sv) 1980-02-11
MY8400017A (en) 1984-12-31
PT69670A (en) 1979-06-01
NO850153L (no) 1979-11-27
FI67705B (fi) 1985-01-31
AT370420B (de) 1983-03-25
CA1127633A (en) 1982-07-13
FI67705C (fi) 1985-05-10
SE8402887L (sv) 1984-05-28
SI7911231A8 (en) 1997-06-30
DE2921316C2 (de) 1982-09-16
NO791731L (no) 1979-11-27
FI801609A (fi) 1980-05-19
LU81319A1 (fr) 1979-09-11
AU4742279A (en) 1979-11-29
DK157685B (da) 1990-02-05

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