FI67555C - Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t - Google Patents

Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t Download PDF

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Publication number
FI67555C
FI67555C FI791678A FI791678A FI67555C FI 67555 C FI67555 C FI 67555C FI 791678 A FI791678 A FI 791678A FI 791678 A FI791678 A FI 791678A FI 67555 C FI67555 C FI 67555C
Authority
FI
Finland
Prior art keywords
compound
formula
group
acid
cef
Prior art date
Application number
FI791678A
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English (en)
Finnish (fi)
Other versions
FI67555B (fi
FI791678A (fi
Inventor
Cynthia Hilda O'callaghan
David George Hubert Livermore
Christopher Earle Mewall
Original Assignee
Glaxo Group Ltd
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Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of FI791678A publication Critical patent/FI791678A/fi
Priority to FI801609A priority Critical patent/FI67705C/fi
Publication of FI67555B publication Critical patent/FI67555B/fi
Application granted granted Critical
Publication of FI67555C publication Critical patent/FI67555C/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
FI791678A 1978-05-26 1979-05-25 Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t FI67555C (fi)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FI801609A FI67705C (fi) 1978-05-26 1980-05-19 Foerfarande foer framstaellning av terapeutiskt anvaendbara (6,7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(substituerad oxiimi noacetamido)-(eventuellt substituerat pyridiniummetyl)cef-3 -e-4-karboxylatfoereningar

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB2291378 1978-05-26
GB2291178 1978-05-26
GB2291178 1978-05-26
GB2291378 1978-05-26

Publications (3)

Publication Number Publication Date
FI791678A FI791678A (fi) 1979-11-27
FI67555B FI67555B (fi) 1984-12-31
FI67555C true FI67555C (fi) 1985-04-10

Family

ID=26256190

Family Applications (2)

Application Number Title Priority Date Filing Date
FI791678A FI67555C (fi) 1978-05-26 1979-05-25 Foerfarande foer framstaellning av terapeutiskt anvaendbart (6 7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(2-karboxiprop-2-oxi imno)-acetamido)-3-(1-pyridiniummetyl)-cef-3-em-4-karboxyla t
FI801609A FI67705C (fi) 1978-05-26 1980-05-19 Foerfarande foer framstaellning av terapeutiskt anvaendbara (6,7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(substituerad oxiimi noacetamido)-(eventuellt substituerat pyridiniummetyl)cef-3 -e-4-karboxylatfoereningar

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI801609A FI67705C (fi) 1978-05-26 1980-05-19 Foerfarande foer framstaellning av terapeutiskt anvaendbara (6,7r)-7-((z)-2-(2-aminotiazol-4-yl)-2-(substituerad oxiimi noacetamido)-(eventuellt substituerat pyridiniummetyl)cef-3 -e-4-karboxylatfoereningar

Country Status (27)

Country Link
US (2) US4258041A (no)
AR (2) AR228726A1 (no)
AT (1) AT370420B (no)
AU (1) AU524671B2 (no)
CA (1) CA1127633A (no)
CH (2) CH649556A5 (no)
DE (1) DE2921316C2 (no)
DK (1) DK157685C (no)
ES (2) ES480914A1 (no)
FI (2) FI67555C (no)
FR (2) FR2426695A1 (no)
HK (1) HK40183A (no)
IE (2) IE49172B1 (no)
IL (3) IL57400A (no)
IT (1) IT1116198B (no)
KE (1) KE3252A (no)
LU (1) LU81319A1 (no)
MY (1) MY8400017A (no)
NL (2) NL176855C (no)
NO (2) NO155347C (no)
NZ (2) NZ190558A (no)
PH (1) PH16961A (no)
PT (2) PT69669A (no)
SE (2) SE438507B (no)
SG (1) SG58382G (no)
SI (2) SI7911231A8 (no)
YU (2) YU41635B (no)

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IL57400A (en) 1982-08-31
YU223482A (en) 1983-04-30
CH646178A5 (de) 1984-11-15
US4258041A (en) 1981-03-24
IL59793A0 (en) 1980-06-30
NL176855B (nl) 1985-01-16
DK157685C (da) 1990-07-09
AR228726A1 (es) 1983-04-15
FR2426695A1 (fr) 1979-12-21
IE802453L (en) 1979-11-26
ES480915A1 (es) 1980-02-01
FR2445835B1 (no) 1983-06-03
NZ190558A (en) 1982-05-31
YU123179A (en) 1983-01-21
IE49173B1 (en) 1985-08-21
IE791025L (en) 1979-11-26
AU524671B2 (en) 1982-09-30
ATA239281A (de) 1982-08-15
IL57400A0 (en) 1979-09-30
YU41635B (en) 1987-12-31
PH16961A (en) 1984-04-27
FR2445835A1 (fr) 1980-08-01
FI67555B (fi) 1984-12-31
US4600772A (en) 1986-07-15
NL176855C (nl) 1985-06-17
FR2426695B1 (no) 1982-06-11
PT69669A (en) 1979-06-01
NL8001348A (nl) 1980-06-30
NZ193326A (en) 1982-05-31
YU43097B (en) 1989-02-28
IL59793A (en) 1982-08-31
CH649556A5 (de) 1985-05-31
NO155347B (no) 1966-12-08
FI791678A (fi) 1979-11-27
ES480914A1 (es) 1980-02-01
AR229883A1 (es) 1983-12-30
KE3252A (en) 1983-01-28
SE8402887D0 (sv) 1984-05-28
DE2921316A1 (de) 1979-12-06
IE49172B1 (en) 1985-08-21
DK216779A (da) 1979-11-27
SE438507B (sv) 1985-04-22
IT1116198B (it) 1986-02-10
SG58382G (en) 1983-09-02
NL7904122A (nl) 1979-11-28
NO155347C (no) 1987-03-18
SI8212234A8 (en) 1997-06-30
HK40183A (en) 1983-10-21
SE7904576L (sv) 1980-02-11
MY8400017A (en) 1984-12-31
PT69670A (en) 1979-06-01
NO850153L (no) 1979-11-27
FI67705B (fi) 1985-01-31
AT370420B (de) 1983-03-25
CA1127633A (en) 1982-07-13
FI67705C (fi) 1985-05-10
SE8402887L (sv) 1984-05-28
SI7911231A8 (en) 1997-06-30
DE2921316C2 (de) 1982-09-16
NO791731L (no) 1979-11-27
FI801609A (fi) 1980-05-19
LU81319A1 (fr) 1979-09-11
AU4742279A (en) 1979-11-29
DK157685B (da) 1990-02-05

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