FR2384782A1 - Nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments - Google Patents
Nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicamentsInfo
- Publication number
- FR2384782A1 FR2384782A1 FR7708988A FR7708988A FR2384782A1 FR 2384782 A1 FR2384782 A1 FR 2384782A1 FR 7708988 A FR7708988 A FR 7708988A FR 7708988 A FR7708988 A FR 7708988A FR 2384782 A1 FR2384782 A1 FR 2384782A1
- Authority
- FR
- France
- Prior art keywords
- acetamido
- thiazolyl
- amino
- cephalosporin
- resistant staphylococci
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/40—Unsubstituted amino or imino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
Les produits de formule générale I :
Priority Applications (36)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7708988A FR2384782A1 (fr) | 1977-03-25 | 1977-03-25 | Nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments |
SE7802833A SE439312B (sv) | 1977-03-25 | 1978-03-13 | Sett att framstella nya oximderivat av 3-acetoximetyl-7-aminotiazolylacetamido cefalosporansyra |
US05/886,421 US4288434A (en) | 1977-03-25 | 1978-03-14 | Cephalosporanic acid derivatives |
ZA00781630A ZA781630B (en) | 1977-03-25 | 1978-03-21 | New oxime derivatives of 3-acetoxy methyl 7-amino thiazolyl acetamido cephalosporanic acid-process for preparing them and pharmaceutical compositions |
ES468169A ES468169A1 (es) | 1977-03-25 | 1978-03-22 | Procedimiento de preparacion de nuevas oximas derivadas del acido 3-acetoximetil-7-aminotiazolil-acetamido-cefalospora- nico. |
DK129578A DK159156C (da) | 1977-03-25 | 1978-03-22 | Analogifremgangsmaade til fremstilling af (2-(2-aminothiazol-4-yl)-2-(0-substitueret)-oxyiminoacetamido)-7-cephalosporan-syre og fysiologisk acceptable salte deraf |
HU78RO972A HU182567B (en) | 1977-03-25 | 1978-03-22 | Prcess for preparing new oxime derivatives of 3-acetoxymethyl-7-amino-thiazolyl-acetamido-cef-3-em-4-carboxylic acid |
DE19782812625 DE2812625A1 (de) | 1977-03-25 | 1978-03-22 | Oximderivate der 3-acetoxymethyl-7- aminothiazolyl-acetamido-cephalosporansaeure, ihre herstellung und pharmazeutische mittel |
DE2858771A DE2858771C2 (fr) | 1977-03-25 | 1978-03-22 | |
CA299,661A CA1125280A (fr) | 1977-03-25 | 1978-03-23 | Procede de preparation de nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique |
CH1361/84A CH648555A5 (fr) | 1977-03-25 | 1978-03-23 | Ester d'un acide thiazolyl acetique. |
GB11613/78A GB1605175A (en) | 1977-03-25 | 1978-03-23 | Oxime derivatives of 7-(amino-thiazolyl-acetamido)-cephalosporanic acid process for preparing them and pharmaceutical compositions containing them |
PT67815A PT67815A (fr) | 1977-03-25 | 1978-03-23 | Procede de preparation de nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-aminothiazolyl acetamido cephalosporanique |
NL7803166A NL192041C (nl) | 1977-03-25 | 1978-03-23 | Geneesmiddel met antibacteriële werking, alsmede 7-£2-(2-aminothiazool-4-yl)-2-(veretherd oxyimino)-aceetamido|-3-cefem -4-carbonzuurderivaten. |
GB16825/80A GB1605176A (en) | 1977-03-25 | 1978-03-23 | Oxime derivatives of 7-amino-thiazolyl-acetic acid and processes for preparing them |
CH322978A CH633292A5 (fr) | 1977-03-25 | 1978-03-23 | Oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique, procede de preparation et compositions pharmaceutiques. |
AU34471/78A AU520657B2 (en) | 1977-03-25 | 1978-03-23 | Oxime Derivatives of 3- acetoxy methyl 7-amino thiazolyl acetamido cephalosporanic acid, process for preparing them and pharmaceutical compositions |
BE186254A BE865298A (fr) | 1977-03-25 | 1978-03-24 | Nouvelles oximes derivees de l'acide 3-acetoxy-methyl 7-amino thiazolyl acetamido cephalosporanique, procede de preparation et compositions pharmaceutiques |
LU79312A LU79312A1 (fr) | 1977-03-25 | 1978-03-24 | Procede de preparation de nouvelles oximes derivees de l'acide 3-acetoxymethyl-7-amino thiazolyl acetamido cephalosporanique |
JP3319378A JPS53119887A (en) | 1977-03-25 | 1978-03-24 | Novel oxime derivative of 33acetoxymethyll 77aminothiazolylacetoamide cephalospolanate process for preparing same and pharmaceutical composition |
IT48604/78A IT1103478B (it) | 1977-03-25 | 1978-03-24 | Ossime derivate dall'acido 3-acetos simetil 7-ammino-tiazolil-acetammido cefalosporanico procedimento per la loro produzione e composizioni farmaceutiche che le contengono come ingrediente attivo |
PH20927A PH15764A (en) | 1977-03-25 | 1978-03-27 | Cephalosporanic acid derivatives |
AT218378A AT360153B (de) | 1977-03-25 | 1978-03-28 | Verfahren zur herstellung von neuen ver- bindungen |
IE604/78A IE47361B1 (en) | 1977-03-25 | 1978-03-29 | New oxime derivatives of (amino-thiazolyl-acetamido)-cephalosporanic acid,processes for preparing them and pharmaceutical compositions containing them |
IE1518/83A IE47362B1 (en) | 1977-03-25 | 1978-03-29 | New oxime derivatives of 7-amino-thiazolyl-acetic acid,and processes for preparing them |
ES477592A ES477592A1 (es) | 1977-03-25 | 1979-02-09 | Procedimiento de preparacion de nuevas oximas derivadas del acido 3-acetoximetil-7-aminotiazolil-acetamido-cefalospora- nico. |
AT331380A AT376215B (de) | 1977-03-25 | 1980-06-24 | Verfahren zur herstellung neuer substituierter 2-(2-amino-4-thiazolyl)-2-hydroxyiminoessigsaeur n |
US06/260,311 US4386210A (en) | 1977-03-25 | 1981-05-04 | 2-(2-Amino-4-thiazolyl)-2-methoxyimino-acetic acid derivatives |
CA379,842A CA1132575A (fr) | 1977-03-25 | 1981-06-16 | Derives de l'acide 2-(2-amino 4-thiazolyl) 2- hydroxyimino acetique et procede pour leur preparation preparation |
CH386882A CH639652A5 (fr) | 1977-03-25 | 1982-06-18 | Acides thiazolyl acetiques, leurs esters et leurs procedes de preparation. |
US06/469,710 US4487937A (en) | 1977-03-25 | 1983-02-25 | 2-(2-Substitutedamino-4-thiazolyl)-2-(1-methoxy-isopropoxyimino)-acetic acids |
SE8304239A SE453192B (sv) | 1977-03-25 | 1983-08-02 | Nya mellanprodukter anvendbara for framstellning av oximderivat av 3-acetoximetyl-7-aminotiazolyl-acetamido-cefalosporinsyra samt forfarande for framstellning av mellanprodukterna |
CH644383A CH646159A5 (fr) | 1977-03-25 | 1983-12-02 | Acides thiazolyl acetiques et leur preparation. |
US06/574,876 US4483981A (en) | 1977-03-25 | 1984-01-30 | Cephalosporanic acid derivatives |
JP61014877A JPS61218580A (ja) | 1977-03-25 | 1986-01-28 | 2−(2−アミノ−4−チアゾリル)−2−メトキシイミノ酢酸誘導体及びその製造法 |
JP63152471A JPS6425768A (en) | 1977-03-25 | 1988-06-22 | 2-(2-amino-4-thiazolyl)-2-methoxyiminoacetic acid derivative and manufacture |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7708988A FR2384782A1 (fr) | 1977-03-25 | 1977-03-25 | Nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2384782A1 true FR2384782A1 (fr) | 1978-10-20 |
FR2384782B1 FR2384782B1 (fr) | 1980-03-14 |
Family
ID=9188585
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7708988A Granted FR2384782A1 (fr) | 1977-03-25 | 1977-03-25 | Nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments |
Country Status (4)
Country | Link |
---|---|
JP (1) | JPS61218580A (fr) |
BE (1) | BE865298A (fr) |
FR (1) | FR2384782A1 (fr) |
ZA (1) | ZA781630B (fr) |
Cited By (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2399418A1 (fr) * | 1977-03-14 | 1979-03-02 | Fujisawa Pharmaceutical Co | Procede de preparation d'acides iminoacetiques et nouveaux produits ainsi obtenus, utilises pour la synthese d'acides cepham- ou cephem-carboxyliques |
EP0009548A2 (fr) * | 1978-07-17 | 1980-04-16 | Fujisawa Pharmaceutical Co., Ltd. | Dérivés de céphalosporine, procédé pour leur préparation, compositions pharmaceutiques les contenant |
FR2476647A2 (fr) * | 1980-02-26 | 1981-08-28 | Roussel Uclaf | Procede de preparation de derives de l'acide 2-(2-amino protege 4-thiazolyl) 2-alkoxyimino acetique isomere syn |
FR2478102A1 (fr) * | 1980-03-13 | 1981-09-18 | Squibb & Sons Inc | Nouveaux derives d'acide hydroxamique de ((amino-2 thiazolyl-4) oximino)-cephalosporines utiles notamment comme medicaments antibacteriens |
FR2506307A1 (fr) * | 1981-05-22 | 1982-11-26 | Roussel Uclaf | Nouveaux derives substitues de l'acide 2-(2-amino 4-thiazolyl) 2-hydroxyimino acetique et leur procede de preparation |
EP0095329A2 (fr) * | 1982-05-20 | 1983-11-30 | Glaxo Group Limited | Céphalosporines antibiotiques |
EP0101265A2 (fr) * | 1982-08-07 | 1984-02-22 | Tanabe Seiyaku Co., Ltd. | Dérivés de céphalosporines et leur préparation |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2714880A1 (de) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | Cephemderivate und verfahren zu ihrer herstellung |
AR228726A1 (es) | 1978-05-26 | 1983-04-15 | Glaxo Group Ltd | Procedimiento para la preparacion del antibiotico(6r,7r)-7-((z)-2-(2-aminotiazol-4-il)-2-(2-carboxiprop-2-oxiimino)acetamido)-3-(1-piridiniometil)cef-3-em-4-carboxilato |
-
1977
- 1977-03-25 FR FR7708988A patent/FR2384782A1/fr active Granted
-
1978
- 1978-03-21 ZA ZA00781630A patent/ZA781630B/xx unknown
- 1978-03-24 BE BE186254A patent/BE865298A/fr not_active IP Right Cessation
-
1986
- 1986-01-28 JP JP61014877A patent/JPS61218580A/ja active Pending
Cited By (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2399418A1 (fr) * | 1977-03-14 | 1979-03-02 | Fujisawa Pharmaceutical Co | Procede de preparation d'acides iminoacetiques et nouveaux produits ainsi obtenus, utilises pour la synthese d'acides cepham- ou cephem-carboxyliques |
EP0009548A2 (fr) * | 1978-07-17 | 1980-04-16 | Fujisawa Pharmaceutical Co., Ltd. | Dérivés de céphalosporine, procédé pour leur préparation, compositions pharmaceutiques les contenant |
EP0009548A3 (en) * | 1978-07-17 | 1980-06-25 | Fujisawa Pharmaceutical Co. Ltd. | Cephalosporin derivatives, process for their preparation and pharmaceutical compositions containing them, and their starting derivatives and their preparation |
EP0059486A1 (fr) * | 1978-07-17 | 1982-09-08 | Fujisawa Pharmaceutical Co., Ltd. | Produits de départ pour la préparation des composés céphalosporiniques et procédé de préparation |
FR2476647A2 (fr) * | 1980-02-26 | 1981-08-28 | Roussel Uclaf | Procede de preparation de derives de l'acide 2-(2-amino protege 4-thiazolyl) 2-alkoxyimino acetique isomere syn |
FR2478102A1 (fr) * | 1980-03-13 | 1981-09-18 | Squibb & Sons Inc | Nouveaux derives d'acide hydroxamique de ((amino-2 thiazolyl-4) oximino)-cephalosporines utiles notamment comme medicaments antibacteriens |
FR2506307A1 (fr) * | 1981-05-22 | 1982-11-26 | Roussel Uclaf | Nouveaux derives substitues de l'acide 2-(2-amino 4-thiazolyl) 2-hydroxyimino acetique et leur procede de preparation |
EP0095329A2 (fr) * | 1982-05-20 | 1983-11-30 | Glaxo Group Limited | Céphalosporines antibiotiques |
EP0095329A3 (fr) * | 1982-05-20 | 1984-11-28 | Glaxo Group Limited | Céphalosporines antibiotiques |
EP0101265A2 (fr) * | 1982-08-07 | 1984-02-22 | Tanabe Seiyaku Co., Ltd. | Dérivés de céphalosporines et leur préparation |
EP0101265A3 (en) * | 1982-08-07 | 1985-04-10 | Tanabe Seiyaku Co., Ltd. | Novel cephalosporin compounds and preparation thereof |
US4598075A (en) * | 1982-08-07 | 1986-07-01 | Tanabe Seiyaku Co., Ltd. | Cephalosporin compounds |
Also Published As
Publication number | Publication date |
---|---|
JPS61218580A (ja) | 1986-09-29 |
ZA781630B (en) | 1979-04-25 |
BE865298A (fr) | 1978-09-25 |
FR2384782B1 (fr) | 1980-03-14 |
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