FI105478B - Menetelmä valmistaa terapeuttisesti vaikuttavaa 2-deoksi-2,3-didehydro-N-asetyylineuramiinihapon johdannaisia ja niiden analogeja - Google Patents

Menetelmä valmistaa terapeuttisesti vaikuttavaa 2-deoksi-2,3-didehydro-N-asetyylineuramiinihapon johdannaisia ja niiden analogeja Download PDF

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Publication number
FI105478B
FI105478B FI924790A FI924790A FI105478B FI 105478 B FI105478 B FI 105478B FI 924790 A FI924790 A FI 924790A FI 924790 A FI924790 A FI 924790A FI 105478 B FI105478 B FI 105478B
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FI
Finland
Prior art keywords
compound
tetradeoxy
acetamido
glycero
formula
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FI924790A
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English (en)
Finnish (fi)
Swedish (sv)
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FI924790A (fi
FI924790A0 (fi
Inventor
Betty Jin
Wen Yang Wu
Basil Danylec
Itzstein Laurence Mark Von
Phan Tho Van
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Biota Scient Management
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Publication of FI924790A0 publication Critical patent/FI924790A0/fi
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI924790A 1990-04-24 1992-10-22 Menetelmä valmistaa terapeuttisesti vaikuttavaa 2-deoksi-2,3-didehydro-N-asetyylineuramiinihapon johdannaisia ja niiden analogeja FI105478B (fi)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
AUPJ980090 1990-04-24
AUPJ980090 1990-04-24
AUPK289690 1990-10-19
AUPK289690 1990-10-19
AUPK453791 1991-02-11
AUPK453791 1991-02-11
AU9100161 1991-04-24
PCT/AU1991/000161 WO1991016320A1 (en) 1990-04-24 1991-04-24 Derivatives and analogues of 2-deoxy-2,3-didehydro-n-acetyl neuraminic acid and their use as antiviral agents

Publications (3)

Publication Number Publication Date
FI924790A FI924790A (fi) 1992-10-22
FI924790A0 FI924790A0 (fi) 1992-10-22
FI105478B true FI105478B (fi) 2000-08-31

Family

ID=27157556

Family Applications (2)

Application Number Title Priority Date Filing Date
FI924790A FI105478B (fi) 1990-04-24 1992-10-22 Menetelmä valmistaa terapeuttisesti vaikuttavaa 2-deoksi-2,3-didehydro-N-asetyylineuramiinihapon johdannaisia ja niiden analogeja
FI20001231A FI20001231A (fi) 1990-04-24 2000-05-23 2-Deoksi-2,3-didehydro-N-asetyylineuramiinihapon johdannaisia ja niiden analogeja ja niiden käyttö antiviraalisina aineina

Family Applications After (1)

Application Number Title Priority Date Filing Date
FI20001231A FI20001231A (fi) 1990-04-24 2000-05-23 2-Deoksi-2,3-didehydro-N-asetyylineuramiinihapon johdannaisia ja niiden analogeja ja niiden käyttö antiviraalisina aineina

Country Status (37)

Country Link
US (2) US5360817A (pl)
EP (2) EP0526543B1 (pl)
JP (1) JP2944750B2 (pl)
KR (1) KR0169496B1 (pl)
CN (3) CN1036849C (pl)
AP (1) AP249A (pl)
AT (2) ATE406358T1 (pl)
AU (2) AU654815B2 (pl)
BG (1) BG62092B1 (pl)
CA (2) CA2291994C (pl)
CY (1) CY2186B1 (pl)
CZ (1) CZ288492B6 (pl)
DE (3) DE69128469T2 (pl)
DK (1) DK0526543T3 (pl)
ES (2) ES2313730T3 (pl)
FI (2) FI105478B (pl)
GR (1) GR3026225T3 (pl)
HK (2) HK1003834A1 (pl)
HU (2) HU219355B (pl)
IE (2) IE911372A1 (pl)
IL (1) IL97936A (pl)
LU (1) LU90468I2 (pl)
MY (1) MY107843A (pl)
NL (1) NL990030I2 (pl)
NO (3) NO302751B1 (pl)
NZ (1) NZ237936A (pl)
OA (1) OA09679A (pl)
PL (3) PL166918B1 (pl)
PT (1) PT97460B (pl)
RU (1) RU2119487C1 (pl)
SG (1) SG43170A1 (pl)
SI (1) SI9110745B (pl)
SK (1) SK282950B6 (pl)
UA (1) UA41252C2 (pl)
WO (1) WO1991016320A1 (pl)
YU (1) YU48741B (pl)
ZA (1) ZA913086B (pl)

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