ES2546762T3 - Procedimientos para preparar derivados de bencil-benceno sustituidos con glucopiranosilo - Google Patents

Procedimientos para preparar derivados de bencil-benceno sustituidos con glucopiranosilo Download PDF

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Publication number
ES2546762T3
ES2546762T3 ES10762899.2T ES10762899T ES2546762T3 ES 2546762 T3 ES2546762 T3 ES 2546762T3 ES 10762899 T ES10762899 T ES 10762899T ES 2546762 T3 ES2546762 T3 ES 2546762T3
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Prior art keywords
alkyl
acid
organic
process according
phenyl
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ES10762899.2T
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English (en)
Spanish (es)
Inventor
Dirk Weber
Tobias Fiedler
Christian Filser
Rainer Hamm
Simone Orlich
Matthias Post
Svenja Renner
Xiao-Jun Wang
Thomas Wirth
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Boehringer Ingelheim International GmbH
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Boehringer Ingelheim International GmbH
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C07D309/12—Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C07H1/06—Separation; Purification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Packaging Of Annular Or Rod-Shaped Articles, Wearing Apparel, Cassettes, Or The Like (AREA)
  • Wrapping Of Specific Fragile Articles (AREA)
ES10762899.2T 2009-09-30 2010-09-24 Procedimientos para preparar derivados de bencil-benceno sustituidos con glucopiranosilo Active ES2546762T3 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24714409P 2009-09-30 2009-09-30
US247144P 2009-09-30
PCT/EP2010/064120 WO2011039108A2 (en) 2009-09-30 2010-09-24 Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives

Publications (1)

Publication Number Publication Date
ES2546762T3 true ES2546762T3 (es) 2015-09-28

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ES10762899.2T Active ES2546762T3 (es) 2009-09-30 2010-09-24 Procedimientos para preparar derivados de bencil-benceno sustituidos con glucopiranosilo

Country Status (25)

Country Link
US (2) US9024010B2 (show.php)
EP (1) EP2486029B1 (show.php)
JP (1) JP5758900B2 (show.php)
KR (1) KR101813025B1 (show.php)
CN (1) CN102574829B (show.php)
AR (1) AR078193A1 (show.php)
AU (1) AU2010303124B2 (show.php)
BR (1) BR112012007085B8 (show.php)
CA (1) CA2775962C (show.php)
CL (1) CL2012000581A1 (show.php)
DK (1) DK2486029T3 (show.php)
EA (1) EA022032B1 (show.php)
ES (1) ES2546762T3 (show.php)
HR (1) HRP20150945T1 (show.php)
HU (1) HUE026133T2 (show.php)
IL (1) IL218101A0 (show.php)
IN (1) IN2012DN02751A (show.php)
MX (1) MX2012003048A (show.php)
NZ (1) NZ598366A (show.php)
PH (1) PH12012500634A1 (show.php)
PL (1) PL2486029T3 (show.php)
PT (1) PT2486029E (show.php)
SI (1) SI2486029T1 (show.php)
TW (1) TWI465458B (show.php)
WO (1) WO2011039108A2 (show.php)

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EA033286B1 (ru) 2013-04-18 2019-09-30 Бёрингер Ингельхайм Интернациональ Гмбх Способ лечения или отсрочки развития хронической болезни почек
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