EA201001554A1 - Ингибиторы модуляторов воспаления: производные олеанолевой кислоты, гомологированные с-17 - Google Patents

Ингибиторы модуляторов воспаления: производные олеанолевой кислоты, гомологированные с-17

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Publication number
EA201001554A1
EA201001554A1 EA201001554A EA201001554A EA201001554A1 EA 201001554 A1 EA201001554 A1 EA 201001554A1 EA 201001554 A EA201001554 A EA 201001554A EA 201001554 A EA201001554 A EA 201001554A EA 201001554 A1 EA201001554 A1 EA 201001554A1
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EA
Eurasian Patent Office
Prior art keywords
oleanolic acid
homologous
inhibitors
acid derivatives
inflammation modulators
Prior art date
Application number
EA201001554A
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English (en)
Other versions
EA020156B1 (ru
Inventor
Зин Джайэнг
Зиофен Лайу
Джек Грейнер
Стивен С. Сзакс
Мелеэн Висник
Original Assignee
Ритэ Фамэсутикл, Инк.
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Application filed by Ритэ Фамэсутикл, Инк. filed Critical Ритэ Фамэсутикл, Инк.
Publication of EA201001554A1 publication Critical patent/EA201001554A1/ru
Publication of EA020156B1 publication Critical patent/EA020156B1/ru

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Abstract

Настоящее изобретение направлено, среди прочего, на создание новых производных олеанолевой кислоты, имеющих формулув которой все переменные такие, как определено в данном описании. Предлагается также фармацевтическая композиция, комплекты и изделия, содержащие такие соединения, способы и промежуточные вещества, применяемые при приготовлении соединений, а также способы применения соединений и композиций.
EA201001554A 2008-04-18 2009-04-20 Антиоксидативные модуляторы воспаления: гомологизированные по с-17 производные олеанолевой кислоты EA020156B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4636608P 2008-04-18 2008-04-18
US11129408P 2008-11-04 2008-11-04
PCT/US2009/041176 WO2009129548A1 (en) 2008-04-18 2009-04-20 Antioxidant inflammation modulators: c-17 homologated oleanolic acid derivatives

Publications (2)

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EA201001554A1 true EA201001554A1 (ru) 2011-06-30
EA020156B1 EA020156B1 (ru) 2014-09-30

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