CY1118475T1 - Αντιοξειδωτικοι ρυθμιστες φλεγμονης: c-17 ομολογοποιημενα παραγωγα ολεανολικου οξεος - Google Patents

Αντιοξειδωτικοι ρυθμιστες φλεγμονης: c-17 ομολογοποιημενα παραγωγα ολεανολικου οξεος

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Publication number
CY1118475T1
CY1118475T1 CY20171100090T CY171100090T CY1118475T1 CY 1118475 T1 CY1118475 T1 CY 1118475T1 CY 20171100090 T CY20171100090 T CY 20171100090T CY 171100090 T CY171100090 T CY 171100090T CY 1118475 T1 CY1118475 T1 CY 1118475T1
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CY
Cyprus
Prior art keywords
olanolic
oxygen
acid producers
inflammatory regulators
compounds
Prior art date
Application number
CY20171100090T
Other languages
English (en)
Inventor
Xin Jiang
Melean Visnick
Jack Greiner
Xiaofeng Liu
Stephen S Szucs
Original Assignee
Reata Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reata Pharmaceuticals, Inc. filed Critical Reata Pharmaceuticals, Inc.
Publication of CY1118475T1 publication Critical patent/CY1118475T1/el

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Abstract

Η εφεύρεση παρέχει, αλλά δεν περιορίζεται σε αυτά, καινοτόμα παράγωγα ολεανολικού οξέος που έχουν τον τύπο (1) με τις μεταβλητές να ορίζονται στο παρόν. Επίσης παρέχονται φαρμακευτικές συνθέσεις, κιτ και προϊόντα (articles of manufacture) που περιλαμβάνουν τέτοιες ενώσεις, μέθοδοι και ενδιάμεσα χρήσιμα για την παραγωγή των ενώσεων, και μέθοδοι χρήσης των ενώσεων και συνθέσεων.
CY20171100090T 2008-04-18 2017-01-23 Αντιοξειδωτικοι ρυθμιστες φλεγμονης: c-17 ομολογοποιημενα παραγωγα ολεανολικου οξεος CY1118475T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US4636608P 2008-04-18 2008-04-18
US11129408P 2008-11-04 2008-11-04
PCT/US2009/041176 WO2009129548A1 (en) 2008-04-18 2009-04-20 Antioxidant inflammation modulators: c-17 homologated oleanolic acid derivatives

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CY1118475T1 true CY1118475T1 (el) 2017-07-12

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KR101354828B1 (ko) 2005-11-04 2014-02-18 와이어쓰 엘엘씨 ｍＴＯＲ 저해자, 헤르셉틴, 및/또는 ＨＫＩ-272의항신생물성 조합
US8022216B2 (en) 2007-10-17 2011-09-20 Wyeth Llc Maleate salts of (E)-N-{4-[3-chloro-4-(2-pyridinylmethoxy)anilino]-3-cyano-7-ethoxy-6-quinolinyl}-4-(dimethylamino)-2-butenamide and crystalline forms thereof
MX356760B (es) 2008-01-11 2018-06-12 Dartmouth College Triterpenoides sinteticos y metodos de uso en el tratamiento de enfermedad.
US7915402B2 (en) 2008-04-18 2011-03-29 Reata Pharmaceuticals, Inc. Antioxidant inflammation modulators: oleanolic acid derivatives with saturation in the C-ring
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