CY2186B1 - Derivatives and analogues of 2-deoxy-2,3-didehydro-n-acetyl neuraminic acid and their use as antiviral agents - Google Patents

Derivatives and analogues of 2-deoxy-2,3-didehydro-n-acetyl neuraminic acid and their use as antiviral agents

Info

Publication number
CY2186B1
CY2186B1 CY9900009A CY9900009A CY2186B1 CY 2186 B1 CY2186 B1 CY 2186B1 CY 9900009 A CY9900009 A CY 9900009A CY 9900009 A CY9900009 A CY 9900009A CY 2186 B1 CY2186 B1 CY 2186B1
Authority
CY
Cyprus
Prior art keywords
didehydro
deoxy
analogues
derivatives
antiviral agents
Prior art date
Application number
CY9900009A
Other languages
English (en)
Inventor
Von Laurence Mark Itzstein
Wen-Yang Wu
Van Tho Phan
Basil Danylec
Betty Jin
Original Assignee
Biota Scient Man
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biota Scient Man filed Critical Biota Scient Man
Publication of CY2186B1 publication Critical patent/CY2186B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
CY9900009A 1990-04-24 1999-03-02 Derivatives and analogues of 2-deoxy-2,3-didehydro-n-acetyl neuraminic acid and their use as antiviral agents CY2186B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AUPJ980090 1990-04-24
AUPK289690 1990-10-19
AUPK453791 1991-02-11

Publications (1)

Publication Number Publication Date
CY2186B1 true CY2186B1 (en) 2002-11-08

Family

ID=27157556

Family Applications (1)

Application Number Title Priority Date Filing Date
CY9900009A CY2186B1 (en) 1990-04-24 1999-03-02 Derivatives and analogues of 2-deoxy-2,3-didehydro-n-acetyl neuraminic acid and their use as antiviral agents

Country Status (37)

Country Link
US (2) US5360817A (bg)
EP (2) EP0526543B1 (bg)
JP (1) JP2944750B2 (bg)
KR (1) KR0169496B1 (bg)
CN (3) CN1036849C (bg)
AP (1) AP249A (bg)
AT (2) ATE406358T1 (bg)
AU (2) AU654815B2 (bg)
BG (1) BG62092B1 (bg)
CA (2) CA2291994C (bg)
CY (1) CY2186B1 (bg)
CZ (1) CZ288492B6 (bg)
DE (3) DE69128469T2 (bg)
DK (1) DK0526543T3 (bg)
ES (2) ES2313730T3 (bg)
FI (2) FI105478B (bg)
GR (1) GR3026225T3 (bg)
HK (2) HK1003834A1 (bg)
HU (2) HU219355B (bg)
IE (2) IE911372A1 (bg)
IL (1) IL97936A (bg)
LU (1) LU90468I2 (bg)
MY (1) MY107843A (bg)
NL (1) NL990030I2 (bg)
NO (3) NO302751B1 (bg)
NZ (1) NZ237936A (bg)
OA (1) OA09679A (bg)
PL (3) PL166918B1 (bg)
PT (1) PT97460B (bg)
RU (1) RU2119487C1 (bg)
SG (1) SG43170A1 (bg)
SI (1) SI9110745B (bg)
SK (1) SK282950B6 (bg)
UA (1) UA41252C2 (bg)
WO (1) WO1991016320A1 (bg)
YU (1) YU48741B (bg)
ZA (1) ZA913086B (bg)

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NL287642A (bg) 1962-01-18

Also Published As

Publication number Publication date
FI924790A (fi) 1992-10-22
AU7533891A (en) 1991-12-12
NO302751B1 (no) 1998-04-20
FI105478B (fi) 2000-08-31
NO974670L (no) 1992-12-18
CZ288492B6 (en) 2001-06-13
NL990030I1 (nl) 1999-12-01
CN1036849C (zh) 1997-12-31
MY107843A (en) 1996-06-29
SI9110745A (en) 1997-04-30
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PL167630B1 (pl) 1995-10-31
DE69128469T2 (de) 1998-06-04
RU2119487C1 (ru) 1998-09-27
AU654815B2 (en) 1994-11-24
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IE911372A1 (en) 1991-11-06
PL166918B1 (pl) 1995-07-31
CA2291994C (en) 2003-10-14
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ES2313730T3 (es) 2009-03-01
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DE69128469D1 (de) 1998-01-29
EP0526543A1 (en) 1993-02-10
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YU74591A (sh) 1994-06-24
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KR0169496B1 (ko) 1999-01-15
HU210717A9 (en) 1995-06-28
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AP249A (en) 1993-03-17
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UA41252C2 (uk) 2001-09-17
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US5648379A (en) 1997-07-15
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OA09679A (en) 1993-05-15
HU9203180D0 (en) 1992-12-28
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SK282950B6 (sk) 2003-01-09
LU90468I2 (fr) 2000-01-03
NO923944D0 (no) 1992-10-09
PL167192B1 (pl) 1995-08-31
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US5360817A (en) 1994-11-01
ZA913086B (en) 1992-12-30

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