CY1114563T1 - Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα - Google Patents

Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα

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Publication number
CY1114563T1
CY1114563T1 CY20131100819T CY131100819T CY1114563T1 CY 1114563 T1 CY1114563 T1 CY 1114563T1 CY 20131100819 T CY20131100819 T CY 20131100819T CY 131100819 T CY131100819 T CY 131100819T CY 1114563 T1 CY1114563 T1 CY 1114563T1
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CY
Cyprus
Prior art keywords
methyl
butin
pyridin
hydrates
cyano
Prior art date
Application number
CY20131100819T
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English (en)
Inventor
Waldemar Pfrengle
Peter Sieger
Original Assignee
Boehringer Ingelheim International Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37102454&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1114563(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim International Gmbh filed Critical Boehringer Ingelheim International Gmbh
Publication of CY1114563T1 publication Critical patent/CY1114563T1/el

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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
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Abstract

Η εφεύρεση σχετίζεται με άλατα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-[3-αμινο-πιπεριδιν-1-υλο]-ξανθίνης με υδροχλωρικό οξύ, καθώς και με τα εναντιομερή αυτών, μείγματα αυτών και ένυδρα συμπλέγματα αυτών.
CY20131100819T 2005-07-30 2013-09-18 Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα CY1114563T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005035891A DE102005035891A1 (de) 2005-07-30 2005-07-30 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP06777973.6A EP1912990B1 (de) 2005-07-30 2006-07-26 Hydrochloride und hydrate von 1-[(3-cyano-pyridin-2-yl) methyl]-3-methyl-7-(2-butin-1-yl)-8-(3-amino-piperidin-1-yl)-xanthin, deren herstellung und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
CY1114563T1 true CY1114563T1 (el) 2016-10-05

Family

ID=37102454

Family Applications (1)

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CY20131100819T CY1114563T1 (el) 2005-07-30 2013-09-18 Υδροχλωριδια και ενυδρα συμπλεγματα της 1-[(3-κυανο-πυριδιν-2-υλο)μεθυλο]-3-μεθυλο-7-(2-βουτιν-1-υλο)-8-(3-αμινο-πιπεριδιν-1-υλο)ξανθινης, η παραγωγη αυτων και η χρηση αυτων ως φαρμακευτικα μεσα

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US (2) US8106060B2 (el)
EP (2) EP2540724B1 (el)
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