CN1610547A - 用作5-ht6受体拮抗剂的n-(2-芳乙基)苄胺 - Google Patents

用作5-ht6受体拮抗剂的n-(2-芳乙基)苄胺 Download PDF

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Publication number
CN1610547A
CN1610547A CNA028105435A CN02810543A CN1610547A CN 1610547 A CN1610547 A CN 1610547A CN A028105435 A CNA028105435 A CN A028105435A CN 02810543 A CN02810543 A CN 02810543A CN 1610547 A CN1610547 A CN 1610547A
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ethyl
indol
benzylamine
propoxy
ethoxy
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Chinese (zh)
Inventor
Z·陈
M·P·科肯
M·J·菲谢
B·吉特伦
J·R·吉里格
J·R·麦科旺
S·C·米勒
J·M·肖斯
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Eli Lilly and Co
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Eli Lilly and Co
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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CN104220421A (zh) * 2012-03-20 2014-12-17 阿达梅德公司 用于治疗中枢神经系统疾病的苄胺的磺酰胺衍生物
CN102746211A (zh) * 2012-06-27 2012-10-24 上海泰坦化学有限公司 一种取代吲哚-3-甲醛类化合物的制备方法
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CN104619344A (zh) * 2012-09-09 2015-05-13 H.隆德贝克有限公司 治疗阿尔茨海默病的方法及其药物组合物
CN104725249A (zh) * 2013-12-20 2015-06-24 广东东阳光药业有限公司 苄胺类衍生物及其在药物上的应用
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CN105175307A (zh) * 2014-11-18 2015-12-23 苏州晶云药物科技有限公司 Lu AE58054的盐酸盐晶型A及其制备方法和用途
CN104529865B (zh) * 2014-12-12 2017-02-01 广东东阳光药业有限公司 苄胺类衍生物及其在药物上的应用
CN104529865A (zh) * 2014-12-12 2015-04-22 广东东阳光药业有限公司 苄胺类衍生物及其在药物上的应用
CN108884034A (zh) * 2016-04-08 2018-11-23 H.隆德贝克有限公司 经由亚胺的氢化制造艾达鲁吡啶的方法
CN109069650A (zh) * 2016-04-26 2018-12-21 H.隆德贝克有限公司 乙酰胆碱酯酶抑制剂和艾达鲁吡啶用于减少帕金森氏病患者跌倒的用途
CN106632303A (zh) * 2017-01-09 2017-05-10 湖南华腾制药有限公司 一种6‑噻唑基吲哚衍生物的制备方法
CN109942527A (zh) * 2019-04-26 2019-06-28 新乡市润宇新材料科技有限公司 一种3-溴二苯并呋喃的合成方法
CN116782896A (zh) * 2020-09-02 2023-09-19 恩维瑞克生物科学加拿大公司 硝化裸盖菇素衍生物及其用于调节5-ht2a受体和治疗精神障碍的用途

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