CN100486967C - 5HT2c受体调节剂 - Google Patents

5HT2c受体调节剂 Download PDF

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Publication number
CN100486967C
CN100486967C CNB038082721A CN03808272A CN100486967C CN 100486967 C CN100486967 C CN 100486967C CN B038082721 A CNB038082721 A CN B038082721A CN 03808272 A CN03808272 A CN 03808272A CN 100486967 C CN100486967 C CN 100486967C
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Prior art keywords
tetrahydro
benzazepine
methyl
mmol
trifluoroacetyl
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Expired - Lifetime
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CNB038082721A
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English (en)
Chinese (zh)
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CN1646493A (zh
Inventor
B·史密斯
J·史密斯
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Eisai Co Ltd
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Arena Pharmaceuticals Inc
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Application filed by Arena Pharmaceuticals Inc filed Critical Arena Pharmaceuticals Inc
Priority to CN200910000191.0A priority Critical patent/CN101486678B/zh
Publication of CN1646493A publication Critical patent/CN1646493A/zh
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Publication of CN100486967C publication Critical patent/CN100486967C/zh
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  • Addiction (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
  • Pregnancy & Childbirth (AREA)
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CNB038082721A 2002-04-12 2003-04-11 5HT2c受体调节剂 Expired - Lifetime CN100486967C (zh)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN200910000191.0A CN101486678B (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US37205802P 2002-04-12 2002-04-12
US60/372,058 2002-04-12
US40549502P 2002-08-23 2002-08-23
US60/405,495 2002-08-23
US43460702P 2002-12-18 2002-12-18
US60/434,607 2002-12-18
US10/410,991 2003-04-10
US10/410,991 US6953787B2 (en) 2002-04-12 2003-04-10 5HT2C receptor modulators

Related Child Applications (4)

Application Number Title Priority Date Filing Date
CNA200910000193XA Division CN101485664A (zh) 2002-04-12 2003-04-11 5HT2c受体调节剂
CN200910000191.0A Division CN101486678B (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂
CN2009100001906A Division CN101486677B (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂
CNA2009100001925A Division CN101486679A (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂

Publications (2)

Publication Number Publication Date
CN1646493A CN1646493A (zh) 2005-07-27
CN100486967C true CN100486967C (zh) 2009-05-13

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Family Applications (5)

Application Number Title Priority Date Filing Date
CNB038082721A Expired - Lifetime CN100486967C (zh) 2002-04-12 2003-04-11 5HT2c受体调节剂
CN2009100001906A Expired - Lifetime CN101486677B (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂
CNA200910000193XA Withdrawn CN101485664A (zh) 2002-04-12 2003-04-11 5HT2c受体调节剂
CN200910000191.0A Expired - Lifetime CN101486678B (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂
CNA2009100001925A Pending CN101486679A (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂

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Application Number Title Priority Date Filing Date
CN2009100001906A Expired - Lifetime CN101486677B (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂
CNA200910000193XA Withdrawn CN101485664A (zh) 2002-04-12 2003-04-11 5HT2c受体调节剂
CN200910000191.0A Expired - Lifetime CN101486678B (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂
CNA2009100001925A Pending CN101486679A (zh) 2002-04-12 2003-04-11 5ht2c受体调节剂

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US (11) US6953787B2 (enExample)
EP (4) EP1557409A1 (enExample)
JP (5) JP4155926B2 (enExample)
KR (3) KR100908166B1 (enExample)
CN (5) CN100486967C (enExample)
AT (1) ATE294781T1 (enExample)
AU (1) AU2003221866B2 (enExample)
BR (2) BR122017023795B8 (enExample)
CA (1) CA2481723C (enExample)
CR (2) CR7503A (enExample)
DE (1) DE60300610T2 (enExample)
DK (1) DK1411881T3 (enExample)
ES (2) ES2242165T3 (enExample)
GE (1) GEP20074197B (enExample)
IL (1) IL164162A0 (enExample)
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NZ (1) NZ535381A (enExample)
PL (4) PL219017B1 (enExample)
PT (1) PT1411881E (enExample)
RU (1) RU2317982C2 (enExample)
SI (1) SI1411881T1 (enExample)
TW (1) TWI252105B (enExample)
UA (1) UA77788C2 (enExample)
WO (1) WO2003086306A2 (enExample)
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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101486677B (zh) * 2002-04-12 2012-12-12 阿伦纳药品公司 5ht2c受体调节剂
CN105555769A (zh) * 2013-07-19 2016-05-04 斯洛文尼亚莱柯制药股份有限公司 不需要的对映异构体的外消旋化方法

Families Citing this family (82)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8478824B2 (en) * 2002-02-05 2013-07-02 Portauthority Technologies Inc. Apparatus and method for controlling unauthorized dissemination of electronic mail
SE0200968D0 (sv) * 2002-03-26 2002-03-26 Lars Baltzer Novel polypeptide scaffolds and use thereof
TWI329111B (en) 2002-05-24 2010-08-21 X Ceptor Therapeutics Inc Azepinoindole and pyridoindole derivatives as pharmaceutical agents
US7595311B2 (en) 2002-05-24 2009-09-29 Exelixis, Inc. Azepinoindole derivatives as pharmaceutical agents
ATE441417T1 (de) 2002-12-20 2009-09-15 Glaxo Group Ltd Benzoädüazepinderivate für die behandlung von neurologischen krankheiten
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CN101486678B (zh) * 2002-04-12 2015-09-09 阿伦纳药品公司 5ht2c受体调节剂
CN105555769A (zh) * 2013-07-19 2016-05-04 斯洛文尼亚莱柯制药股份有限公司 不需要的对映异构体的外消旋化方法

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