CA2945746A1 - Compounds useful as immunomodulators - Google Patents

Compounds useful as immunomodulators Download PDF

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Publication number
CA2945746A1
CA2945746A1 CA2945746A CA2945746A CA2945746A1 CA 2945746 A1 CA2945746 A1 CA 2945746A1 CA 2945746 A CA2945746 A CA 2945746A CA 2945746 A CA2945746 A CA 2945746A CA 2945746 A1 CA2945746 A1 CA 2945746A1
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Canada
Prior art keywords
oxy
benzyl
dihydrobenzo
dioxin
amino
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Abandoned
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CA2945746A
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English (en)
French (fr)
Inventor
Louis S. Chupak
Min Ding
Scott W. Martin
Xiaofan Zheng
Piyasena Hewawasam
Timothy P. Connolly
Ningning Xu
Kap-Sun Yeung
Juliang Zhu
David R. Langley
Daniel J. TENNEY
Paul Michael Scola
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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Publication of CA2945746A1 publication Critical patent/CA2945746A1/en
Abandoned legal-status Critical Current

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
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