EA201990221A1 - 1,3-дигидроксифенильные производные, применимые в качестве иммуномодуляторов - Google Patents

1,3-дигидроксифенильные производные, применимые в качестве иммуномодуляторов

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Publication number
EA201990221A1
EA201990221A1 EA201990221A EA201990221A EA201990221A1 EA 201990221 A1 EA201990221 A1 EA 201990221A1 EA 201990221 A EA201990221 A EA 201990221A EA 201990221 A EA201990221 A EA 201990221A EA 201990221 A1 EA201990221 A1 EA 201990221A1
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EA
Eurasian Patent Office
Prior art keywords
immunomodulators
dihydroxiphenyl
compounds
applicable
derivatives applicable
Prior art date
Application number
EA201990221A
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English (en)
Inventor
Кап-сун Еюн
Катрин А. Грант-Янг
Цзюйлян Чжу
Марк Г. Саулниер
Дэвид Б. Френнессон
Чжаосин Мэн
Пол Майкл Скола
Original Assignee
Бристол-Маерс Сквибб Компани
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Application filed by Бристол-Маерс Сквибб Компани filed Critical Бристол-Маерс Сквибб Компани
Publication of EA201990221A1 publication Critical patent/EA201990221A1/ru

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Настоящее изобретение в общем относится к соединениям, применимым в качестве иммуномодуляторов. Оно предусматривает соединения, композиции, содержащие такие соединения, и способы их применения. Изобретение также предусматривает фармацевтические композиции, содержащие по меньшей мере одно соединение по изобретению, которое подходит для лечения различных заболеваний, включая рак и инфекционные заболевания.
EA201990221A 2016-07-08 2017-07-05 1,3-дигидроксифенильные производные, применимые в качестве иммуномодуляторов EA201990221A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662359971P 2016-07-08 2016-07-08
PCT/US2017/040663 WO2018009505A1 (en) 2016-07-08 2017-07-05 1,3-dihydroxy-phenyl derivatives useful as immunomodulators

Publications (1)

Publication Number Publication Date
EA201990221A1 true EA201990221A1 (ru) 2019-06-28

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EA201990221A EA201990221A1 (ru) 2016-07-08 2017-07-05 1,3-дигидроксифенильные производные, применимые в качестве иммуномодуляторов

Country Status (15)

Country Link
US (1) US10590105B2 (ru)
EP (1) EP3481815B1 (ru)
JP (1) JP7168551B2 (ru)
KR (1) KR102491992B1 (ru)
CN (1) CN109689640B (ru)
AU (1) AU2017292758A1 (ru)
BR (1) BR112019000247A2 (ru)
CA (1) CA3029991A1 (ru)
EA (1) EA201990221A1 (ru)
ES (1) ES2895066T3 (ru)
IL (1) IL264092A (ru)
MA (1) MA45591A (ru)
MX (1) MX2019000123A (ru)
SG (1) SG11201900077QA (ru)
WO (1) WO2018009505A1 (ru)

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