CA2777245A1 - Compositions for treatment of cystic fibrosis and other chronic diseases - Google Patents

Compositions for treatment of cystic fibrosis and other chronic diseases Download PDF

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Publication number
CA2777245A1
CA2777245A1 CA2777245A CA2777245A CA2777245A1 CA 2777245 A1 CA2777245 A1 CA 2777245A1 CA 2777245 A CA2777245 A CA 2777245A CA 2777245 A CA2777245 A CA 2777245A CA 2777245 A1 CA2777245 A1 CA 2777245A1
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CA
Canada
Prior art keywords
compound
formula
alkyl
pharmaceutical composition
optionally substituted
Prior art date
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Abandoned
Application number
CA2777245A
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English (en)
French (fr)
Inventor
Fredrick F. Van Goor
William Lawrence Burton
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Vertex Pharmaceuticals Inc
Original Assignee
Vertex Pharmaceuticals Inc
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Filing date
Publication date
Application filed by Vertex Pharmaceuticals Inc filed Critical Vertex Pharmaceuticals Inc
Publication of CA2777245A1 publication Critical patent/CA2777245A1/en
Abandoned legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
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  • Immunology (AREA)
  • Pulmonology (AREA)
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  • Gynecology & Obstetrics (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
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CA2777245A 2009-10-22 2010-10-22 Compositions for treatment of cystic fibrosis and other chronic diseases Abandoned CA2777245A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25418009P 2009-10-22 2009-10-22
US61/254,180 2009-10-22
PCT/US2010/053852 WO2011050325A1 (en) 2009-10-22 2010-10-22 Compositions for treatment of cystic fibrosis and other chronic diseases

Publications (1)

Publication Number Publication Date
CA2777245A1 true CA2777245A1 (en) 2011-04-28

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Family Applications (1)

Application Number Title Priority Date Filing Date
CA2777245A Abandoned CA2777245A1 (en) 2009-10-22 2010-10-22 Compositions for treatment of cystic fibrosis and other chronic diseases

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US (3) US20110098311A1 (enExample)
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US20140329814A2 (en) 2014-11-06
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EP2490687A1 (en) 2012-08-29

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